ES2294641T3 - Nuevos derivados de eritromicina. - Google Patents

Nuevos derivados de eritromicina. Download PDF

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Publication number
ES2294641T3
ES2294641T3 ES05106836T ES05106836T ES2294641T3 ES 2294641 T3 ES2294641 T3 ES 2294641T3 ES 05106836 T ES05106836 T ES 05106836T ES 05106836 T ES05106836 T ES 05106836T ES 2294641 T3 ES2294641 T3 ES 2294641T3
Authority
ES
Spain
Prior art keywords
propyl
formula
compound
imidazol
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES05106836T
Other languages
English (en)
Spanish (es)
Inventor
Yong-Jin Wu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Application granted granted Critical
Publication of ES2294641T3 publication Critical patent/ES2294641T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
ES05106836T 1998-01-02 1998-12-21 Nuevos derivados de eritromicina. Expired - Lifetime ES2294641T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7035898P 1998-01-02 1998-01-02
US70358P 1998-01-02

Publications (1)

Publication Number Publication Date
ES2294641T3 true ES2294641T3 (es) 2008-04-01

Family

ID=22094819

Family Applications (1)

Application Number Title Priority Date Filing Date
ES05106836T Expired - Lifetime ES2294641T3 (es) 1998-01-02 1998-12-21 Nuevos derivados de eritromicina.

Country Status (36)

Country Link
US (1) US6825171B2 (ko)
EP (2) EP1642901B1 (ko)
JP (1) JP2002500231A (ko)
KR (1) KR20010033822A (ko)
CN (1) CN1285841A (ko)
AP (1) AP1060A (ko)
AR (5) AR012764A1 (ko)
AT (1) ATE377018T1 (ko)
AU (1) AU759019B2 (ko)
BG (1) BG104640A (ko)
BR (1) BR9812992A (ko)
CA (1) CA2317131C (ko)
CO (1) CO4970773A1 (ko)
CZ (1) CZ20002456A3 (ko)
DE (1) DE69838651T9 (ko)
DZ (1) DZ2699A1 (ko)
EA (1) EA200000600A1 (ko)
ES (1) ES2294641T3 (ko)
GT (1) GT199800207A (ko)
HR (1) HRP20000444A2 (ko)
HU (1) HUP0100566A3 (ko)
IL (1) IL136721A0 (ko)
IS (1) IS5527A (ko)
MA (1) MA26588A1 (ko)
NO (1) NO20003346L (ko)
NZ (1) NZ504987A (ko)
OA (1) OA11440A (ko)
PA (1) PA8465901A1 (ko)
PE (1) PE20000119A1 (ko)
PL (1) PL341647A1 (ko)
SK (1) SK9772000A3 (ko)
TN (1) TNSN98236A1 (ko)
UY (2) UY25331A1 (ko)
WO (1) WO1999035157A1 (ko)
YU (1) YU40900A (ko)
ZA (1) ZA9811940B (ko)

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EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
ATE344269T1 (de) 1998-12-10 2006-11-15 Pfizer Prod Inc Carbamat und carbazat ketolid antibiotika
EP1749832A3 (en) * 1998-12-10 2008-03-26 Pfizer Products Incorporated Carbamate and carbazate ketolide antibiotics
EP1754700A3 (en) 1999-01-27 2007-05-09 Kosan Biosciences, Inc. Synthesis of oligoketides
BR9916969A (pt) 1999-01-27 2001-11-06 Pfizer Prod Inc Antibióticos cetólidos
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US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
US6514944B2 (en) 1999-04-16 2003-02-04 Kosan Biosciences, Inc. Macrolide antiinfective agents
ES2272273T3 (es) 1999-04-16 2007-05-01 Kosan Biosciences, Inc. Agentes antiinfecciosos macrolidos.
US6939861B2 (en) 1999-04-16 2005-09-06 Kosan Biosciences, Inc. Amido macrolides
AU4354900A (en) 1999-04-16 2000-11-02 Kosan Biosciences, Inc. Ketolide antibacterials
WO2000071557A1 (en) * 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
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EP1114826A3 (en) * 1999-12-29 2001-10-31 Pfizer Products Inc. Novel antibacterial and prokinetic macrolides
US6562795B2 (en) 2000-02-18 2003-05-13 Kosan Biosciences, Inc. Motilide compounds
US20020115621A1 (en) 2000-08-07 2002-08-22 Wei-Gu Su Macrolide antibiotics
US6472372B1 (en) 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
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WO2003024986A1 (en) 2001-09-17 2003-03-27 Ortho-Mcneil Pharmaceutical, Inc. 6-o-carbamate-11,12-lacto-ketolide antimicrobials
BR0214748A (pt) 2001-12-05 2004-11-23 Ortho Mcneil Pharm Inc Derivados 6-oacil-cetolidas de eritromicina, úteis como antibacterianos
US6825172B2 (en) 2002-05-31 2004-11-30 Janssen Pharmaceutica, Nv 3-descladinosyl-6-O-carbamoyl and 6-O-carbonoyl macrolide antibacterial agents
US7163924B2 (en) 2003-04-25 2007-01-16 Chiron Corporation Ketolide derivatives
EP1836211B1 (en) * 2004-12-21 2010-03-03 Pfizer Products Inc. Macrolides
ATE468119T1 (de) 2006-06-12 2010-06-15 Univ Ramot Verfahren zur behandlung von krebs
EA201500699A1 (ru) 2012-12-24 2015-12-30 Рамот Эт Тель-Авив Юниверсити Лтд. Агенты для лечения генетических заболеваний, возникающих в результате нонсенс-мутаций, и способы идентификации этих агентов

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Also Published As

Publication number Publication date
IS5527A (is) 2000-06-09
YU40900A (sh) 2003-01-31
AP9801421A0 (en) 1998-12-31
AR019789A2 (es) 2002-03-13
EP1044208A1 (en) 2000-10-18
AR012764A1 (es) 2000-11-08
IL136721A0 (en) 2001-06-14
PE20000119A1 (es) 2000-02-17
UY25331A1 (es) 2000-12-29
ZA9811940B (en) 2000-06-30
NZ504987A (en) 2002-11-26
EP1642901B1 (en) 2007-10-31
AU759019B2 (en) 2003-04-03
ATE377018T1 (de) 2007-11-15
AR020016A2 (es) 2002-03-27
DE69838651D1 (de) 2007-12-13
AR019790A2 (es) 2002-03-13
HRP20000444A2 (en) 2001-04-30
EP1642901A1 (en) 2006-04-05
AP1060A (en) 2002-04-23
CA2317131C (en) 2004-11-02
PL341647A1 (en) 2001-04-23
SK9772000A3 (en) 2002-09-10
CO4970773A1 (es) 2000-11-07
WO1999035157B1 (en) 1999-10-14
GT199800207A (es) 2000-06-22
BG104640A (en) 2001-09-28
KR20010033822A (ko) 2001-04-25
DZ2699A1 (fr) 2003-03-29
AR019788A2 (es) 2002-03-13
CN1285841A (zh) 2001-02-28
AU1501599A (en) 1999-07-26
DE69838651T9 (de) 2008-06-12
UY25587A1 (es) 1999-09-27
HUP0100566A3 (en) 2003-07-28
US20040067897A1 (en) 2004-04-08
DE69838651T2 (de) 2008-03-06
EA200000600A1 (ru) 2001-02-26
JP2002500231A (ja) 2002-01-08
NO20003346L (no) 2000-08-29
NO20003346D0 (no) 2000-06-27
US6825171B2 (en) 2004-11-30
PA8465901A1 (es) 2000-09-29
MA26588A1 (fr) 2004-12-20
OA11440A (en) 2004-04-28
CA2317131A1 (en) 1999-07-15
CZ20002456A3 (cs) 2001-09-12
TNSN98236A1 (fr) 2005-03-15
BR9812992A (pt) 2000-10-17
HUP0100566A2 (hu) 2001-07-30
WO1999035157A1 (en) 1999-07-15

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