ES2250689T3 - 1h-pirido(4,3-b)indoles terapeuticos. - Google Patents

1h-pirido(4,3-b)indoles terapeuticos.

Info

Publication number
ES2250689T3
ES2250689T3 ES02757023T ES02757023T ES2250689T3 ES 2250689 T3 ES2250689 T3 ES 2250689T3 ES 02757023 T ES02757023 T ES 02757023T ES 02757023 T ES02757023 T ES 02757023T ES 2250689 T3 ES2250689 T3 ES 2250689T3
Authority
ES
Spain
Prior art keywords
pyrido
indole
hexahydro
compound
dichlorophenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES02757023T
Other languages
English (en)
Spanish (es)
Inventor
Michael D. Ennis
Kristine E. Frank
Robert L. Hoffman
Jian-Min Fu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co LLC
Original Assignee
Pharmacia and Upjohn Co LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn Co LLC filed Critical Pharmacia and Upjohn Co LLC
Application granted granted Critical
Publication of ES2250689T3 publication Critical patent/ES2250689T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ES02757023T 2001-08-08 2002-08-06 1h-pirido(4,3-b)indoles terapeuticos. Expired - Lifetime ES2250689T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31089001P 2001-08-08 2001-08-08
US310890P 2001-08-08

Publications (1)

Publication Number Publication Date
ES2250689T3 true ES2250689T3 (es) 2006-04-16

Family

ID=23204521

Family Applications (1)

Application Number Title Priority Date Filing Date
ES02757023T Expired - Lifetime ES2250689T3 (es) 2001-08-08 2002-08-06 1h-pirido(4,3-b)indoles terapeuticos.

Country Status (10)

Country Link
US (1) US6849640B2 (https=)
EP (1) EP1414819B1 (https=)
JP (1) JP2005526691A (https=)
AT (1) ATE306486T1 (https=)
BR (1) BR0211608A (https=)
CA (1) CA2453537A1 (https=)
DE (1) DE60206636T2 (https=)
ES (1) ES2250689T3 (https=)
MX (1) MXPA04001203A (https=)
WO (1) WO2003014118A1 (https=)

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US7592454B2 (en) 2004-04-14 2009-09-22 Bristol-Myers Squibb Company Substituted hexahydro-pyridoindole derivatives as serotonin receptor agonists and antagonists
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WO2007041697A2 (en) * 2005-10-04 2007-04-12 Medivation, Inc. Hydrogenated pyrido-indole compounds for the treatment of huntington ' s disease
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RU2329044C1 (ru) * 2006-11-16 2008-07-20 Андрей Александрович Иващенко Лиганды 5-ht6 рецепторов, фармацевтическая композиция, способ ее получения и лекарственное средство
KR102065319B1 (ko) * 2007-03-12 2020-01-10 인트라-셀룰라 써래피스, 인코퍼레이티드. 치환된 헤테로환 융합 감마-카르볼린 합성
RU2338745C1 (ru) * 2007-03-21 2008-11-20 Андрей Александрович Иващенко ЗАМЕЩЕННЫЕ 2,3,4,5-ТЕТРАГИДРО-1Н-ПИРИДО[4,3-b]ИНДОЛЫ, СПОСОБЫ ИХ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ
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Also Published As

Publication number Publication date
DE60206636D1 (de) 2006-02-23
WO2003014118A1 (en) 2003-02-20
EP1414819A1 (en) 2004-05-06
EP1414819B1 (en) 2005-10-12
CA2453537A1 (en) 2003-02-20
MXPA04001203A (es) 2004-05-20
DE60206636T2 (de) 2006-06-22
US20030060464A1 (en) 2003-03-27
BR0211608A (pt) 2006-04-04
JP2005526691A (ja) 2005-09-08
ATE306486T1 (de) 2005-10-15
US6849640B2 (en) 2005-02-01

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