ECSP12012097A - Derivados de fumarato de ácido graso y sus usos - Google Patents

Derivados de fumarato de ácido graso y sus usos

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Publication number
ECSP12012097A
ECSP12012097A ECSP12012097A ECSP12012097A EC SP12012097 A ECSP12012097 A EC SP12012097A EC SP12012097 A ECSP12012097 A EC SP12012097A EC SP12012097 A ECSP12012097 A EC SP12012097A
Authority
EC
Ecuador
Prior art keywords
fatty acid
derivatives
fumarate
acid fumarate
derivative
Prior art date
Application number
Other languages
English (en)
Inventor
Michael Robert Jirousek
Jean E Bemis
Jesse J Smith
Jill C Milne
Chi B Vu
Original Assignee
Catabasis Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44258993&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP12012097(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Catabasis Pharmaceuticals Inc filed Critical Catabasis Pharmaceuticals Inc
Publication of ECSP12012097A publication Critical patent/ECSP12012097A/es

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    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
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    • C07C235/70Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/72Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atoms of the carboxamide groups bound to acyclic carbon atoms
    • C07C235/76Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton
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    • C07D339/00Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
    • C07D339/02Five-membered rings
    • C07D339/04Five-membered rings having the hetero atoms in positions 1 and 2, e.g. lipoic acid

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Abstract

La invención se refiere a derivados de fumarato de ácido graso, a composiciones que comprenden una cantidad efectiva de un derivado de fumarato de ácido graso y a métodos para tratar o prevenir cáncer, un trastorno metabólico o trastorno neurodegenerativo que comprende la administración de una cantidad efectiva de un derivado de fumarato de ácido graso.
ECSP12012097 2010-01-08 2012-08-08 Derivados de fumarato de ácido graso y sus usos ECSP12012097A (es)

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KR101828616B1 (ko) 2018-02-12
MX337605B (es) 2016-03-10
JP5771627B2 (ja) 2015-09-02
IL244858A0 (en) 2016-05-31
US20160340294A1 (en) 2016-11-24
WO2011085211A1 (en) 2011-07-14
US8969354B2 (en) 2015-03-03
RU2012134069A (ru) 2014-02-20
NI201200120A (es) 2013-06-12
US20150238618A1 (en) 2015-08-27
US20110172240A1 (en) 2011-07-14
DK2521447T3 (en) 2017-09-18
US20130065909A1 (en) 2013-03-14
MX2012007981A (es) 2012-08-23
EP2521447B1 (en) 2017-06-14
CR20120413A (es) 2012-12-18
TWI508725B (zh) 2015-11-21
AU2011204277A1 (en) 2012-08-30
AR080357A1 (es) 2012-04-04
CO6571913A2 (es) 2012-11-30
US9289503B2 (en) 2016-03-22
NZ601698A (en) 2015-04-24
BR112012016879A2 (pt) 2015-09-01
EP2521447A4 (en) 2014-04-30
JP2013516486A (ja) 2013-05-13
CA2786605A1 (en) 2011-07-14
SG182414A1 (en) 2012-08-30
AU2011204277B2 (en) 2015-12-24
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TW201141471A (en) 2011-12-01
CN102821602B (zh) 2016-04-20
EP2521447A1 (en) 2012-11-14
CL2012001911A1 (es) 2012-10-26
MY160249A (en) 2017-02-28
IL244858A (en) 2016-12-29
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