ECSP10010698A - Derivados de dibenzotiazepina y sus usos - Google Patents

Derivados de dibenzotiazepina y sus usos

Info

Publication number
ECSP10010698A
ECSP10010698A EC2010010698A ECSP10010698A ECSP10010698A EC SP10010698 A ECSP10010698 A EC SP10010698A EC 2010010698 A EC2010010698 A EC 2010010698A EC SP10010698 A ECSP10010698 A EC SP10010698A EC SP10010698 A ECSP10010698 A EC SP10010698A
Authority
EC
Ecuador
Prior art keywords
disorder
dibenzotiazepina
derivatives
compounds
schizophrenia
Prior art date
Application number
EC2010010698A
Other languages
English (en)
Spanish (es)
Inventor
Michael R Wood
Dean G Brown
Phil Edwards
Steven Wesolowski
James Hulsizer
James R Damewood
James Campbell Muir
Jr M Edward Pierson
Ashokkumar Bhikkappa Shenvi
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41431860&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP10010698(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ECSP10010698A publication Critical patent/ECSP10010698A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/16—[b, f]-condensed

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
EC2010010698A 2008-06-20 2010-12-20 Derivados de dibenzotiazepina y sus usos ECSP10010698A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US7441708P 2008-06-20 2008-06-20

Publications (1)

Publication Number Publication Date
ECSP10010698A true ECSP10010698A (es) 2011-01-31

Family

ID=41431860

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2010010698A ECSP10010698A (es) 2008-06-20 2010-12-20 Derivados de dibenzotiazepina y sus usos

Country Status (37)

Country Link
US (3) US20110160184A1 (https=)
EP (1) EP2307389B1 (https=)
JP (2) JP5468068B2 (https=)
KR (1) KR20110019781A (https=)
CN (1) CN102131791B (https=)
AR (1) AR072200A1 (https=)
AU (1) AU2009260905B2 (https=)
BR (1) BRPI0914231A2 (https=)
CA (1) CA2728675A1 (https=)
CL (1) CL2010001471A1 (https=)
CR (1) CR11860A (https=)
CU (1) CU23884B1 (https=)
CY (1) CY1113845T1 (https=)
DK (1) DK2307389T3 (https=)
DO (1) DOP2010000393A (https=)
EA (1) EA201001889A1 (https=)
EC (1) ECSP10010698A (https=)
ES (1) ES2402084T3 (https=)
HN (1) HN2010002683A (https=)
HR (1) HRP20130234T1 (https=)
IL (2) IL210081A (https=)
ME (1) ME01516B (https=)
MX (1) MX2010014203A (https=)
MY (1) MY157518A (https=)
NI (1) NI201000224A (https=)
NZ (1) NZ590616A (https=)
PE (1) PE20110029A1 (https=)
PL (1) PL2307389T3 (https=)
PT (1) PT2307389E (https=)
RS (1) RS52703B (https=)
SI (1) SI2307389T1 (https=)
SV (1) SV2010003769A (https=)
TW (1) TWI488854B (https=)
UA (1) UA105903C2 (https=)
UY (1) UY31919A (https=)
WO (1) WO2009154563A1 (https=)
ZA (1) ZA201100488B (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102131791B (zh) * 2008-06-20 2014-12-24 阿斯利康(瑞典)有限公司 二苯并硫杂氮杂*衍生物及其用途
CN105981027A (zh) * 2013-08-12 2016-09-28 哥莱菲特软件公司 安全认证并切换至加密域
CN103524455A (zh) * 2013-10-30 2014-01-22 苏州敬业医药化工有限公司 一种制备2-氯-二苯并[b,f][1,4]硫氮杂卓-11-[10H]酮的方法
CA2931289C (en) 2013-11-21 2023-10-17 Graphite Software Corporation Managed domains for remote content and configuration control on mobile information devices
CN104447615A (zh) * 2014-02-28 2015-03-25 广东东阳光药业有限公司 喹硫平中间体的制备方法
EP4428132A1 (en) * 2023-03-08 2024-09-11 Johann-Wolfgang-Goethe-Universität Frankfurt am Main Slack-activating compounds and their medical use
JP2026509430A (ja) * 2023-03-08 2026-03-19 ヨハン ヴォルフガング ゲーテ－ウニベルジテート フランクフルト アム マイン Ｓｌａｃｋ活性化化合物及びその医学的用途

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Also Published As

Publication number Publication date
AR072200A1 (es) 2010-08-11
TW201002702A (en) 2010-01-16
ZA201100488B (en) 2011-10-26
JP2014098006A (ja) 2014-05-29
AU2009260905B2 (en) 2012-08-23
IL210081A0 (en) 2011-02-28
CN102131791B (zh) 2014-12-24
DK2307389T3 (da) 2013-04-02
SI2307389T1 (sl) 2013-04-30
US20110160184A1 (en) 2011-06-30
CL2010001471A1 (es) 2011-05-06
JP2011524898A (ja) 2011-09-08
JP5468068B2 (ja) 2014-04-09
PE20110029A1 (es) 2011-02-11
PT2307389E (pt) 2013-03-28
EP2307389A1 (en) 2011-04-13
EA201001889A1 (ru) 2011-08-30
MX2010014203A (es) 2011-02-22
DOP2010000393A (es) 2011-01-31
HN2010002683A (es) 2013-01-15
CU23884B1 (es) 2013-04-19
ME01516B (me) 2014-04-20
US8653257B2 (en) 2014-02-18
RS52703B (sr) 2013-08-30
HK1156308A1 (en) 2012-06-08
CN102131791A (zh) 2011-07-20
CR11860A (es) 2011-02-25
CA2728675A1 (en) 2009-12-23
EP2307389A4 (en) 2012-04-11
IL229560A (en) 2015-07-30
CY1113845T1 (el) 2016-07-27
MY157518A (en) 2016-06-15
IL210081A (en) 2013-12-31
US8158618B2 (en) 2012-04-17
BRPI0914231A2 (pt) 2015-11-03
ES2402084T3 (es) 2013-04-26
EP2307389B1 (en) 2013-01-23
KR20110019781A (ko) 2011-02-28
UY31919A (es) 2010-01-29
HRP20130234T1 (hr) 2013-04-30
CU20100252A7 (es) 2011-11-15
NI201000224A (es) 2012-03-19
WO2009154563A1 (en) 2009-12-23
US20090318415A1 (en) 2009-12-24
IL229560A0 (en) 2014-01-30
TWI488854B (zh) 2015-06-21
PL2307389T3 (pl) 2013-05-31
AU2009260905A1 (en) 2009-12-23
SV2010003769A (es) 2011-05-20
NZ590616A (en) 2012-09-28
UA105903C2 (uk) 2014-07-10
US20120202991A1 (en) 2012-08-09

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