EA201490673A1 - Производные пирролопиримидина и пурина - Google Patents

Производные пирролопиримидина и пурина

Info

Publication number
EA201490673A1
EA201490673A1 EA201490673A EA201490673A EA201490673A1 EA 201490673 A1 EA201490673 A1 EA 201490673A1 EA 201490673 A EA201490673 A EA 201490673A EA 201490673 A EA201490673 A EA 201490673A EA 201490673 A1 EA201490673 A1 EA 201490673A1
Authority
EA
Eurasian Patent Office
Prior art keywords
compounds
pyrrolopyrimidine
derivatives
mammals
purin
Prior art date
Application number
EA201490673A
Other languages
English (en)
Russian (ru)
Inventor
Хенгмиао Ченг
Теодор Отто мл. Джонсон
Джон Чарльз Кэт
Кевин Кун-Чин Лиу
Элизабет Энн Ланни
Асако Нагата
Саджив Кришнан Наир
Саймон Пол Планкен
Скотт Чаннинг Саттон
Original Assignee
Пфайзер Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47116127&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201490673(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Пфайзер Инк. filed Critical Пфайзер Инк.
Publication of EA201490673A1 publication Critical patent/EA201490673A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
EA201490673A 2011-09-22 2012-09-10 Производные пирролопиримидина и пурина EA201490673A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161538103P 2011-09-22 2011-09-22
US201261639639P 2012-04-27 2012-04-27
PCT/IB2012/054702 WO2013042006A1 (en) 2011-09-22 2012-09-10 Pyrrolopyrimidine and purine derivatives

Publications (1)

Publication Number Publication Date
EA201490673A1 true EA201490673A1 (ru) 2014-06-30

Family

ID=47116127

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201490673A EA201490673A1 (ru) 2011-09-22 2012-09-10 Производные пирролопиримидина и пурина

Country Status (29)

Country Link
US (2) US9040547B2 (enExample)
EP (1) EP2758402B9 (enExample)
JP (1) JP5914667B2 (enExample)
KR (1) KR20140059246A (enExample)
CN (1) CN103814030A (enExample)
AP (1) AP2014007475A0 (enExample)
AR (1) AR088760A1 (enExample)
AU (1) AU2012311184A1 (enExample)
BR (1) BR112014006840A2 (enExample)
CA (1) CA2847540C (enExample)
CL (2) CL2014002726A1 (enExample)
CO (1) CO6910196A2 (enExample)
CR (1) CR20140132A (enExample)
DO (1) DOP2014000055A (enExample)
EA (1) EA201490673A1 (enExample)
ES (1) ES2575710T3 (enExample)
IL (1) IL231592A0 (enExample)
MA (1) MA35451B1 (enExample)
MD (1) MD20140023A2 (enExample)
MX (1) MX2014003501A (enExample)
NI (1) NI201400023A (enExample)
PE (1) PE20141228A1 (enExample)
PH (1) PH12014500638A1 (enExample)
SG (1) SG2014014450A (enExample)
TN (1) TN2014000115A1 (enExample)
TW (1) TWI492946B (enExample)
UA (1) UA110259C2 (enExample)
UY (1) UY34342A (enExample)
WO (1) WO2013042006A1 (enExample)

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RU2650512C2 (ru) * 2013-09-18 2018-04-16 Бейджин Ханми Фармасьютикал Ко., Лтд. Соединение, ингибирующее активности киназ ВТК и/или JAK3
US11078206B2 (en) 2017-12-28 2021-08-03 Daewoong Pharmaceutical Co., Ltd. Amino-fluoropiperidine derivatives as kinase inhibitor
RU2758370C1 (ru) * 2017-12-28 2021-10-28 Даевунг Фармасьютикал Ко., Лтд. Производные оксифторпиперидина в качестве ингибитора киназы

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RU2585177C2 (ru) * 2010-06-23 2016-05-27 Ханми Сайенс Ко., Лтд. Новые конденсированные пиримидиновые производные для ингибирования тирозинкиназной активности
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