UA93609C2 - 2-amino-5,6-dihydro-6h-pyrrolo[3, 4-d]pyrimidine derivatives as hsp-90 inhibitors for treating cancer - Google Patents

2-amino-5,6-dihydro-6h-pyrrolo[3, 4-d]pyrimidine derivatives as hsp-90 inhibitors for treating cancer

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Publication number
UA93609C2
UA93609C2 UAA200908018A UAA200908018A UA93609C2 UA 93609 C2 UA93609 C2 UA 93609C2 UA A200908018 A UAA200908018 A UA A200908018A UA A200908018 A UAA200908018 A UA A200908018A UA 93609 C2 UA93609 C2 UA 93609C2
Authority
UA
Ukraine
Prior art keywords
hsp
inhibitors
pyrrolo
dihydro
amino
Prior art date
Application number
UAA200908018A
Other languages
Russian (ru)
Inventor
Майкл Джон Беннетт
Люк Реймонд Зегндер
Сача Нинковик
Пей-Пей Кунг
Джерри Джялун Менг
Бювен Гуанг
Original Assignee
Пфайзер Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Пфайзер Инк. filed Critical Пфайзер Инк.
Publication of UA93609C2 publication Critical patent/UA93609C2/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

The present invention is directed to compounds of formula (I), and pharmaceutically acceptable salts thereof, their synthesis, and their use as HSP-90 inhibitors., (І)
UAA200908018A 2007-02-06 2008-01-25 2-amino-5,6-dihydro-6h-pyrrolo[3, 4-d]pyrimidine derivatives as hsp-90 inhibitors for treating cancer UA93609C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US88843307P 2007-02-06 2007-02-06

Publications (1)

Publication Number Publication Date
UA93609C2 true UA93609C2 (en) 2011-02-25

Family

ID=41790615

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200908018A UA93609C2 (en) 2007-02-06 2008-01-25 2-amino-5,6-dihydro-6h-pyrrolo[3, 4-d]pyrimidine derivatives as hsp-90 inhibitors for treating cancer

Country Status (3)

Country Link
CN (1) CN101663305A (en)
UA (1) UA93609C2 (en)
ZA (1) ZA200906166B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2575710T3 (en) * 2011-09-22 2016-06-30 Pfizer Inc Pyrrolopyrimidine and purine derivatives
CN102816792B (en) * 2012-08-17 2018-02-02 南京大学 A kind of regulating heat shock protein 70 is expressed, the method and its application of quantity and activity
CN105237533B (en) * 2015-10-26 2017-03-22 中国药科大学 Tetrahydropyridine [4,3-d] miazines Hsp90 inhibitor and medical application thereof
CN108863886A (en) * 2018-08-01 2018-11-23 江苏八巨药业有限公司 It is a kind of to prepare 3-（3- chloropropyl）The method of -4- oxo-pyrrolidine -1- carboxylic acid, ethyl ester

Also Published As

Publication number Publication date
CN101663305A (en) 2010-03-03
ZA200906166B (en) 2010-06-30

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