EA200870079A1 - Замещенные имидазолы и их применение в качестве пестицидов - Google Patents

Замещенные имидазолы и их применение в качестве пестицидов

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Publication number
EA200870079A1
EA200870079A1 EA200870079A EA200870079A EA200870079A1 EA 200870079 A1 EA200870079 A1 EA 200870079A1 EA 200870079 A EA200870079 A EA 200870079A EA 200870079 A EA200870079 A EA 200870079A EA 200870079 A1 EA200870079 A1 EA 200870079A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pesticides
application
substituted imidazoles
substituted
compounds
Prior art date
Application number
EA200870079A
Other languages
English (en)
Other versions
EA015738B1 (ru
Inventor
Натан Энтони Логан Чабб
Марк Роджер Кокс
Жером Себастьян Довернь
Ричард Эндрю Эвин
Кристель Лоре
Original Assignee
Пфайзер Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Пфайзер Лимитед filed Critical Пфайзер Лимитед
Publication of EA200870079A1 publication Critical patent/EA200870079A1/ru
Publication of EA015738B1 publication Critical patent/EA015738B1/ru

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Данное изобретение относится к ряду альфа-замещенных 2-бензилзамещенных имидазольных соединений и их фармацевтически приемлемых солей и сольватов, к композициям, содержащим такие соединения, способам их синтеза и их применению в качестве противопаразитных средств.
EA200870079A 2006-01-19 2007-01-08 Замещенные имидазолы и их применение в качестве пестицидов EA015738B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US76076506P 2006-01-19 2006-01-19
PCT/IB2007/000071 WO2007083207A1 (en) 2006-01-19 2007-01-08 Substituted imidazoles and their use as pesticides

Publications (2)

Publication Number Publication Date
EA200870079A1 true EA200870079A1 (ru) 2009-02-27
EA015738B1 EA015738B1 (ru) 2011-10-31

Family

ID=38038547

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200870079A EA015738B1 (ru) 2006-01-19 2007-01-08 Замещенные имидазолы и их применение в качестве пестицидов

Country Status (32)

Country Link
US (4) US7592362B2 (ru)
EP (2) EP2423199A1 (ru)
JP (1) JP4463317B2 (ru)
KR (1) KR101044494B1 (ru)
CN (1) CN101370786B (ru)
AR (1) AR059055A1 (ru)
AT (1) ATE505461T1 (ru)
AU (1) AU2007206698B2 (ru)
BR (1) BRPI0707185B8 (ru)
CA (1) CA2632771C (ru)
CY (1) CY1111473T1 (ru)
DE (1) DE602007013869D1 (ru)
DK (1) DK1981853T3 (ru)
EA (1) EA015738B1 (ru)
ES (1) ES2362935T3 (ru)
HK (1) HK1127919A1 (ru)
IL (1) IL192063A0 (ru)
MA (1) MA30166B1 (ru)
ME (2) ME00044B (ru)
MY (1) MY145812A (ru)
NO (1) NO341141B1 (ru)
NZ (1) NZ569209A (ru)
PL (1) PL1981853T3 (ru)
PT (1) PT1981853E (ru)
RS (1) RS53512B1 (ru)
SI (1) SI1981853T1 (ru)
TN (1) TNSN08306A1 (ru)
TW (1) TWI337998B (ru)
UA (1) UA93696C2 (ru)
UY (1) UY30096A1 (ru)
WO (1) WO2007083207A1 (ru)
ZA (1) ZA200805565B (ru)

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CN102127066B (zh) * 2010-12-10 2013-08-14 邵阳学院 4-(7-甲氧基-2,2-二甲基-2,3-二氢苯并呋喃-5-基)-2-(3,4-二甲苯氨基)噻唑手性晶体
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CN108349953B (zh) * 2015-11-18 2022-06-17 孟山都技术公司 杀虫组合物和方法
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Also Published As

Publication number Publication date
EP1981853B1 (en) 2011-04-13
CY1111473T1 (el) 2015-08-05
US7547718B2 (en) 2009-06-16
RS53512B1 (en) 2015-02-27
CA2632771C (en) 2011-03-22
MEP4208A (en) 2010-06-10
CA2632771A1 (en) 2007-07-26
EA015738B1 (ru) 2011-10-31
SI1981853T1 (sl) 2011-08-31
EP1981853A1 (en) 2008-10-22
TW200738644A (en) 2007-10-16
CN101370786A (zh) 2009-02-18
UY30096A1 (es) 2007-08-31
US7592362B2 (en) 2009-09-22
BRPI0707185A2 (pt) 2011-04-26
RS20080304A (en) 2009-05-06
DK1981853T3 (da) 2011-06-20
AU2007206698A1 (en) 2007-07-26
MY145812A (en) 2012-04-30
KR101044494B1 (ko) 2011-06-27
AR059055A1 (es) 2008-03-12
BRPI0707185B1 (pt) 2020-03-17
MA30166B1 (fr) 2009-01-02
WO2007083207A1 (en) 2007-07-26
AU2007206698B2 (en) 2011-11-03
TWI337998B (en) 2011-03-01
JP2009528979A (ja) 2009-08-13
US20080119536A1 (en) 2008-05-22
US20070167506A1 (en) 2007-07-19
PT1981853E (pt) 2011-06-27
EP2423199A1 (en) 2012-02-29
PL1981853T3 (pl) 2011-08-31
US7825149B2 (en) 2010-11-02
NO20083404L (no) 2008-08-04
TNSN08306A1 (fr) 2009-12-29
KR20080085046A (ko) 2008-09-22
ZA200805565B (en) 2009-12-30
ES2362935T3 (es) 2011-07-15
CN101370786B (zh) 2012-01-11
DE602007013869D1 (de) 2011-05-26
US20090312326A1 (en) 2009-12-17
NZ569209A (en) 2010-09-30
HK1127919A1 (en) 2009-10-09
ME00044B (me) 2010-06-10
IL192063A0 (en) 2008-12-29
NO341141B1 (no) 2017-08-28
ATE505461T1 (de) 2011-04-15
US20080125473A1 (en) 2008-05-29
BRPI0707185B8 (pt) 2021-05-25
JP4463317B2 (ja) 2010-05-19
UA93696C2 (ru) 2011-03-10
US7544706B2 (en) 2009-06-09

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