UY30096A1 - Imidazoles sustituidos - Google Patents

Imidazoles sustituidos

Info

Publication number
UY30096A1
UY30096A1 UY30096A UY30096A UY30096A1 UY 30096 A1 UY30096 A1 UY 30096A1 UY 30096 A UY30096 A UY 30096A UY 30096 A UY30096 A UY 30096A UY 30096 A1 UY30096 A1 UY 30096A1
Authority
UY
Uruguay
Prior art keywords
imidazols
replaced
substituted
compounds
parasiticides
Prior art date
Application number
UY30096A
Other languages
English (en)
Inventor
Christelle Lauret
Richard Andrew Ewin
Jerome Sebastien Dauvergne
Mark Roger Cox
Nathan Anthony Logan Chubb
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of UY30096A1 publication Critical patent/UY30096A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Esta invención se refiere a una gama de compuestos de imidazol 2-bencil sustituido alfa sustituido y las sales y los solvatos farmacéuticamente aceptables de los mismos, a composiciones que comprenden tales compuestos, procedimientos para sus síntesis y su uso como parasiticidas,
UY30096A 2006-01-19 2007-01-17 Imidazoles sustituidos UY30096A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76076506P 2006-01-19 2006-01-19

Publications (1)

Publication Number Publication Date
UY30096A1 true UY30096A1 (es) 2007-08-31

Family

ID=38038547

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30096A UY30096A1 (es) 2006-01-19 2007-01-17 Imidazoles sustituidos

Country Status (32)

Country Link
US (4) US7592362B2 (es)
EP (2) EP1981853B1 (es)
JP (1) JP4463317B2 (es)
KR (1) KR101044494B1 (es)
CN (1) CN101370786B (es)
AR (1) AR059055A1 (es)
AT (1) ATE505461T1 (es)
AU (1) AU2007206698B2 (es)
BR (1) BRPI0707185B8 (es)
CA (1) CA2632771C (es)
CY (1) CY1111473T1 (es)
DE (1) DE602007013869D1 (es)
DK (1) DK1981853T3 (es)
EA (1) EA015738B1 (es)
ES (1) ES2362935T3 (es)
HK (1) HK1127919A1 (es)
IL (1) IL192063A0 (es)
MA (1) MA30166B1 (es)
ME (2) ME00044B (es)
MY (1) MY145812A (es)
NO (1) NO341141B1 (es)
NZ (1) NZ569209A (es)
PL (1) PL1981853T3 (es)
PT (1) PT1981853E (es)
RS (1) RS53512B1 (es)
SI (1) SI1981853T1 (es)
TN (1) TNSN08306A1 (es)
TW (1) TWI337998B (es)
UA (1) UA93696C2 (es)
UY (1) UY30096A1 (es)
WO (1) WO2007083207A1 (es)
ZA (1) ZA200805565B (es)

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US7592362B2 (en) * 2006-01-19 2009-09-22 Pfizer Limited Substituted imidazoles
US20100041712A1 (en) * 2008-08-18 2010-02-18 Pfizer Inc. Substituted imidazole combinations
AU2009331253B2 (en) 2008-12-24 2012-03-08 Daiichi Sankyo Company, Limited Indanyl compounds
SG172140A1 (en) 2008-12-24 2011-07-28 Daiichi Sankyo Co Ltd Cyclic amine compounds
MX2011008816A (es) * 2009-02-23 2011-09-15 Wyeth Llc Formulacion ectoparasiticida con esencia mejorada.
KR101751085B1 (ko) * 2009-07-16 2017-07-11 솔베이 플루오르 게엠베하 플루오로알킬 (플루오로)알킬 카보네이트의 제조 방법
AU2010339691B2 (en) * 2010-01-07 2015-04-02 Alkermes Pharma Ireland Limited Prodrugs of heteraromatic compounds
MX2012008799A (es) 2010-01-29 2012-08-23 Pfizer Formulaciones antiparasitarias topicas.
CN102127066B (zh) * 2010-12-10 2013-08-14 邵阳学院 4-(7-甲氧基-2,2-二甲基-2,3-二氢苯并呋喃-5-基)-2-(3,4-二甲苯氨基)噻唑手性晶体
WO2012139010A1 (en) * 2011-04-08 2012-10-11 University Of Kansas Grp94 inhibitors
US9295623B2 (en) * 2011-10-03 2016-03-29 Eq Ag Solutions Methods of preventing the transmission of communicable diseases in livestock
US9173404B2 (en) 2011-11-17 2015-11-03 Merial, Inc. Compositions comprising an aryl pyrazole and a substituted imidazole, methods and uses thereof
SG11201403980VA (en) * 2012-01-13 2014-08-28 Gen Hospital Corp Anesthetic compounds and related methods of use
CN102987824A (zh) * 2012-11-29 2013-03-27 张敏 一种防螨虫被
CN104844459B (zh) * 2014-02-18 2016-08-24 扬州三友合成化工有限公司 一种氯甲基异丙基碳酸酯的制备方法
WO2017087218A1 (en) * 2015-11-18 2017-05-26 Monsanto Technology Llc Insecticidal compositions and methods
US10550089B2 (en) 2016-05-12 2020-02-04 Heptares Therapeutics Limited Inhibitors of protease-activated receptor-2
US10766866B2 (en) 2017-10-30 2020-09-08 University Of North Texas Health Science Center At Fort Worth Deterrents for arthropods and marine organisms
CN115073298A (zh) * 2022-05-31 2022-09-20 湖南华腾制药有限公司 连续流微反应器合成2-甲基-3-三氟甲基苯胺的方法

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Also Published As

Publication number Publication date
MEP4208A (en) 2010-06-10
SI1981853T1 (sl) 2011-08-31
US7544706B2 (en) 2009-06-09
NO341141B1 (no) 2017-08-28
RS53512B1 (en) 2015-02-27
CN101370786A (zh) 2009-02-18
AU2007206698B2 (en) 2011-11-03
US20080125473A1 (en) 2008-05-29
US20070167506A1 (en) 2007-07-19
US20090312326A1 (en) 2009-12-17
KR20080085046A (ko) 2008-09-22
WO2007083207A1 (en) 2007-07-26
MY145812A (en) 2012-04-30
DE602007013869D1 (de) 2011-05-26
EP2423199A1 (en) 2012-02-29
IL192063A0 (en) 2008-12-29
CA2632771A1 (en) 2007-07-26
EA015738B1 (ru) 2011-10-31
US7547718B2 (en) 2009-06-16
CA2632771C (en) 2011-03-22
BRPI0707185B8 (pt) 2021-05-25
PT1981853E (pt) 2011-06-27
KR101044494B1 (ko) 2011-06-27
RS20080304A (en) 2009-05-06
EA200870079A1 (ru) 2009-02-27
AU2007206698A1 (en) 2007-07-26
AR059055A1 (es) 2008-03-12
BRPI0707185B1 (pt) 2020-03-17
ME00044B (me) 2010-06-10
TW200738644A (en) 2007-10-16
NO20083404L (no) 2008-08-04
TNSN08306A1 (fr) 2009-12-29
JP2009528979A (ja) 2009-08-13
CN101370786B (zh) 2012-01-11
MA30166B1 (fr) 2009-01-02
HK1127919A1 (en) 2009-10-09
ATE505461T1 (de) 2011-04-15
US20080119536A1 (en) 2008-05-22
DK1981853T3 (da) 2011-06-20
EP1981853B1 (en) 2011-04-13
US7592362B2 (en) 2009-09-22
PL1981853T3 (pl) 2011-08-31
EP1981853A1 (en) 2008-10-22
CY1111473T1 (el) 2015-08-05
NZ569209A (en) 2010-09-30
US7825149B2 (en) 2010-11-02
TWI337998B (en) 2011-03-01
ES2362935T3 (es) 2011-07-15
UA93696C2 (ru) 2011-03-10
BRPI0707185A2 (pt) 2011-04-26
ZA200805565B (en) 2009-12-30
JP4463317B2 (ja) 2010-05-19

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Effective date: 20180809