DK2621916T3 - Benzazole derivatives as histamine H 4 receptor ligands - Google Patents

Benzazole derivatives as histamine H 4 receptor ligands Download PDF

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Publication number
DK2621916T3
DK2621916T3 DK11761383.6T DK11761383T DK2621916T3 DK 2621916 T3 DK2621916 T3 DK 2621916T3 DK 11761383 T DK11761383 T DK 11761383T DK 2621916 T3 DK2621916 T3 DK 2621916T3
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Prior art keywords
methyl
methylpiperidin
yloxy
benzimidazol
phenyl
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DK11761383.6T
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Danish (da)
English (en)
Inventor
Isabelle Berrebi-Bertrand
Xavier Billot
Thierry Calmels
Marc Capet
Denis Danvy
Stéphane Krief
Olivier Labeeuw
Jeanne-Marie Lecomte
Nicolas Levoin
Xavier Ligneau
Philippe Robert
Jean-Charles Schwartz
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Bioprojet Soc Civ
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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DK11761383.6T 2010-09-27 2011-09-27 Benzazole derivatives as histamine H 4 receptor ligands DK2621916T3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20100306038 EP2447263A1 (en) 2010-09-27 2010-09-27 Benzazole derivatives as histamine H4 receptor ligands
PCT/EP2011/066782 WO2012041860A1 (en) 2010-09-27 2011-09-27 Benzazole derivatives as histamine h4 receptor ligands

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DK2621916T3 true DK2621916T3 (en) 2016-04-18

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DK11761383.6T DK2621916T3 (en) 2010-09-27 2011-09-27 Benzazole derivatives as histamine H 4 receptor ligands

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US (2) US8802664B2 (Direct)
EP (2) EP2447263A1 (Direct)
JP (1) JP5922128B2 (Direct)
CN (1) CN103228643B (Direct)
CA (1) CA2812686C (Direct)
CY (1) CY1117416T1 (Direct)
DK (1) DK2621916T3 (Direct)
ES (1) ES2571335T3 (Direct)
HR (1) HRP20160398T1 (Direct)
HU (1) HUE027252T2 (Direct)
MX (1) MX339460B (Direct)
PL (1) PL2621916T3 (Direct)
RS (1) RS54737B1 (Direct)
SI (1) SI2621916T1 (Direct)
SM (1) SMT201600262B (Direct)
WO (1) WO2012041860A1 (Direct)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103648639B (zh) 2011-04-19 2016-10-12 沙特基础工业公司 碳负载的钴和钼催化剂
JP6180514B2 (ja) * 2012-05-04 2017-08-16 ノバルティス アーゲー 補体経路モジュレーターおよびその使用
EP2671870A1 (en) * 2012-06-05 2013-12-11 Bioprojet Novel (aza)benzhydryl ether derivatives, their process of preparation and their use as H4-receptor ligands for therapeutical applications
PL2858647T3 (pl) 2012-06-08 2018-10-31 Sensorion Inhibitory receptora h4 do leczenia szumów usznych
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