DK1948661T3 - Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer - Google Patents

Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer

Info

Publication number
DK1948661T3
DK1948661T3 DK06809195T DK06809195T DK1948661T3 DK 1948661 T3 DK1948661 T3 DK 1948661T3 DK 06809195 T DK06809195 T DK 06809195T DK 06809195 T DK06809195 T DK 06809195T DK 1948661 T3 DK1948661 T3 DK 1948661T3
Authority
DK
Denmark
Prior art keywords
pyrazolo
pyrimidin
derivative used
pde5 inhibitors
pde5
Prior art date
Application number
DK06809195T
Other languages
Danish (da)
English (en)
Inventor
Michael Brent Tollefson
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of DK1948661T3 publication Critical patent/DK1948661T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
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DK06809195T 2005-11-10 2006-10-31 Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer DK1948661T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73532005P 2005-11-10 2005-11-10
PCT/IB2006/003132 WO2007054778A1 (en) 2005-11-10 2006-10-31 Pyrazolo[4,3-d]pyrimidin-5-yl)derivative used as pde5 inhibitors

Publications (1)

Publication Number Publication Date
DK1948661T3 true DK1948661T3 (da) 2009-09-07

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
DK06809195T DK1948661T3 (da) 2005-11-10 2006-10-31 Pyrazolo[4,3-D]pyrimidin-5-YL)-derivat anvendt som PDE5-inhibitorer

Country Status (30)

Country Link
US (2) US20090156618A1 (no)
EP (1) EP1948661B1 (no)
JP (1) JP4208959B1 (no)
KR (1) KR101012592B1 (no)
CN (1) CN101305007B (no)
AP (1) AP2008004437A0 (no)
AR (1) AR057885A1 (no)
AT (1) ATE435865T1 (no)
AU (1) AU2006313486B2 (no)
BR (1) BRPI0618284A2 (no)
CA (1) CA2629339C (no)
CR (1) CR9966A (no)
DE (1) DE602006007728D1 (no)
DK (1) DK1948661T3 (no)
DO (1) DOP2006000248A (no)
EA (1) EA200800920A1 (no)
EC (1) ECSP088441A (no)
ES (1) ES2326919T3 (no)
HK (1) HK1120803A1 (no)
IL (1) IL190456A (no)
MA (1) MA29943B1 (no)
NL (1) NL2000291C2 (no)
NO (1) NO20082593L (no)
PE (1) PE20070764A1 (no)
RS (1) RS20080197A (no)
TN (1) TNSN08209A1 (no)
TW (1) TW200738723A (no)
UY (1) UY29909A1 (no)
WO (1) WO2007054778A1 (no)
ZA (1) ZA200803173B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20110050654A (ko) * 2008-08-01 2011-05-16 바이오크리스트 파마수티컬즈, 인코퍼레이티드 Ｊａｋ3 억제제로서의 피페리딘 유도체
WO2010043633A1 (en) * 2008-10-15 2010-04-22 Palau Pharma, S. A. 2h-pyrazolo [4,3-d]pyrimidin-5-amine derivatives as h4 histamine receptor antagonists for the treatment of allergic, immunological and inflammatory diseases
EP2556820A4 (en) * 2010-04-05 2015-01-21 Sk Chemicals Co Ltd COMPOSITION CONTAINING PDE5 INHIBITOR FOR MITIGATION OF SKIN WRINKLES
WO2012118042A1 (ja) * 2011-02-28 2012-09-07 独立行政法人国立循環器病研究センター 悪性腫瘍転移抑制用医薬
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WO2014060112A1 (en) 2012-10-19 2014-04-24 Origenis Gmbh Pyrazolo[4,3-d]pyrimidines as kinase inhibitors
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