DK175288B1 - Farmaceutiske midler indeholdende lægemidler, der er ustabile eller sparsomt oplöselige i vand, og fremgangsmåder til deres fremstilling - Google Patents

Farmaceutiske midler indeholdende lægemidler, der er ustabile eller sparsomt oplöselige i vand, og fremgangsmåder til deres fremstilling Download PDF

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Publication number
DK175288B1
DK175288B1 DK198503595A DK359585A DK175288B1 DK 175288 B1 DK175288 B1 DK 175288B1 DK 198503595 A DK198503595 A DK 198503595A DK 359585 A DK359585 A DK 359585A DK 175288 B1 DK175288 B1 DK 175288B1
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Prior art keywords
water
cyclodextrin
drug
agent according
methyl
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DK198503595A
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Danish (da)
English (en)
Other versions
DK359585D0 (da
DK359585A (da
Inventor
Ulrich Brauns
Bernhard Willi Werner Mueller
Original Assignee
Janssen Pharmaceutica Nv
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Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DK359585D0 publication Critical patent/DK359585D0/da
Publication of DK359585A publication Critical patent/DK359585A/da
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Classifications

    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B82—NANOTECHNOLOGY
    • B82Y—SPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00—Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08B—POLYSACCHARIDES; DERIVATIVES THEREOF
    • C08B37/00—Preparation of polysaccharides not provided for in groups C08B1/00 - C08B35/00; Derivatives thereof
    • C08B37/0006—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid
    • C08B37/0009—Homoglycans, i.e. polysaccharides having a main chain consisting of one single sugar, e.g. colominic acid alpha-D-Glucans, e.g. polydextrose, alternan, glycogen; (alpha-1,4)(alpha-1,6)-D-Glucans; (alpha-1,3)(alpha-1,4)-D-Glucans, e.g. isolichenan or nigeran; (alpha-1,4)-D-Glucans; (alpha-1,3)-D-Glucans, e.g. pseudonigeran; Derivatives thereof
    • C08B37/0012—Cyclodextrin [CD], e.g. cycle with 6 units (alpha), with 7 units (beta) and with 8 units (gamma), large-ring cyclodextrin or cycloamylose with 9 units or more; Derivatives thereof
    • C08B37/0015—Inclusion compounds, i.e. host-guest compounds, e.g. polyrotaxanes

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nanotechnology (AREA)
  • Molecular Biology (AREA)
  • General Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • Public Health (AREA)
  • Medical Informatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK198503595A 1983-12-21 1985-08-07 Farmaceutiske midler indeholdende lægemidler, der er ustabile eller sparsomt oplöselige i vand, og fremgangsmåder til deres fremstilling DK175288B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3346123 1983-12-21
DE19833346123 DE3346123A1 (de) 1983-12-21 1983-12-21 Pharmazeutische praeparate von in wasser schwerloeslichen oder instabilen arzneistoffen und verfahren zu ihrer herstellung
PCT/EP1984/000417 WO1985002767A1 (fr) 1983-12-21 1984-12-20 Compositions pharmaceutiques contenant des medicaments instables ou peu solubles dans l'eau et leurs procedes de preparation
EP8400417 1984-12-20

Publications (3)

Publication Number Publication Date
DK359585D0 DK359585D0 (da) 1985-08-07
DK359585A DK359585A (da) 1985-08-07
DK175288B1 true DK175288B1 (da) 2004-08-09

Family

ID=6217510

Family Applications (1)

Application Number Title Priority Date Filing Date
DK198503595A DK175288B1 (da) 1983-12-21 1985-08-07 Farmaceutiske midler indeholdende lægemidler, der er ustabile eller sparsomt oplöselige i vand, og fremgangsmåder til deres fremstilling

Country Status (17)

Country Link
EP (1) EP0149197B2 (fr)
JP (1) JPS61500788A (fr)
AT (1) ATE51145T1 (fr)
AU (1) AU565966B2 (fr)
CA (1) CA1222697A (fr)
CY (1) CY1689A (fr)
DE (2) DE3346123A1 (fr)
DK (1) DK175288B1 (fr)
FI (1) FI86140C (fr)
HK (1) HK131293A (fr)
HU (1) HU200943B (fr)
LU (1) LU90283I2 (fr)
NL (1) NL980009I1 (fr)
NO (1) NO2000007I1 (fr)
SG (1) SG24893G (fr)
WO (1) WO1985002767A1 (fr)
ZA (1) ZA8410042B (fr)

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FI853198L (fi) 1985-08-20
DK359585D0 (da) 1985-08-07
CY1689A (en) 1994-01-14
ZA8410042B (en) 1985-09-25
HK131293A (en) 1993-12-03
FI853198A0 (fi) 1985-08-20
EP0149197A3 (en) 1985-08-14
WO1985002767A1 (fr) 1985-07-04
DE3346123A1 (de) 1985-06-27
AU3835285A (en) 1985-07-12
ATE51145T1 (de) 1990-04-15
LU90283I2 (fr) 1998-11-03
DK359585A (da) 1985-08-07
EP0149197A2 (fr) 1985-07-24
HU200943B (en) 1990-09-28
JPS61500788A (ja) 1986-04-24
JPH0570612B2 (fr) 1993-10-05
EP0149197B2 (fr) 1997-01-08
NO2000007I1 (no) 2000-09-21
CA1222697A (fr) 1987-06-09
FI86140C (fi) 1992-07-27
EP0149197B1 (fr) 1990-03-21
NL980009I1 (nl) 1998-05-06
AU565966B2 (en) 1987-10-01
DE3481680D1 (de) 1990-04-26
HUT40561A (en) 1987-01-28
FI86140B (fi) 1992-04-15
SG24893G (en) 1993-08-06

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