DK1144436T3 - Fremgangsmåde til fremstilling af bicykliske forbindelser og anvendelse af denne fremgangsmåde til fremstilling af en ICE-inhiberende forbindelse - Google Patents
Fremgangsmåde til fremstilling af bicykliske forbindelser og anvendelse af denne fremgangsmåde til fremstilling af en ICE-inhiberende forbindelseInfo
- Publication number
- DK1144436T3 DK1144436T3 DK00900552T DK00900552T DK1144436T3 DK 1144436 T3 DK1144436 T3 DK 1144436T3 DK 00900552 T DK00900552 T DK 00900552T DK 00900552 T DK00900552 T DK 00900552T DK 1144436 T3 DK1144436 T3 DK 1144436T3
- Authority
- DK
- Denmark
- Prior art keywords
- preparing
- inhibitory compound
- bicyclic compounds
- compound
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9900227A FR2788276B1 (fr) | 1999-01-12 | 1999-01-12 | NOUVEAU PROCEDE DE PREPARATION DE COMPOSES BICYCLIQUES ET L'APPLICATION DE CE PROCEDE COMME ETAPE INTERMEDIAIRE POUR LA PREPARATION D'UN COMPOSE INHIBITEUR DE L'ENZYME DE CONVERSION DE L'INTERLEUKINE 1-BETA (ice) |
PCT/FR2000/000041 WO2000042061A1 (fr) | 1999-01-12 | 2000-01-11 | Procede de preparation de composes bicycliques et l'application de ce procede pour la preparation d'un compose inhibiteur de ice |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1144436T3 true DK1144436T3 (da) | 2004-08-02 |
Family
ID=9540778
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK00900552T DK1144436T3 (da) | 1999-01-12 | 2000-01-11 | Fremgangsmåde til fremstilling af bicykliske forbindelser og anvendelse af denne fremgangsmåde til fremstilling af en ICE-inhiberende forbindelse |
Country Status (24)
Country | Link |
---|---|
US (1) | US6512111B1 (zh) |
EP (1) | EP1144436B1 (zh) |
JP (1) | JP4601826B2 (zh) |
KR (1) | KR100797349B1 (zh) |
CN (1) | CN1240710C (zh) |
AT (1) | ATE263780T1 (zh) |
AU (1) | AU774752B2 (zh) |
BR (1) | BR0007810B1 (zh) |
CA (1) | CA2359964C (zh) |
DE (1) | DE60009658T2 (zh) |
DK (1) | DK1144436T3 (zh) |
ES (1) | ES2215020T3 (zh) |
FR (1) | FR2788276B1 (zh) |
HK (1) | HK1045316B (zh) |
HU (1) | HU230062B1 (zh) |
IL (2) | IL144227A0 (zh) |
NO (1) | NO328110B1 (zh) |
NZ (1) | NZ512908A (zh) |
PL (1) | PL196993B1 (zh) |
PT (1) | PT1144436E (zh) |
SI (1) | SI1144436T1 (zh) |
TW (1) | TWI222443B (zh) |
WO (1) | WO2000042061A1 (zh) |
ZA (1) | ZA200105550B (zh) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6559304B1 (en) | 1998-08-19 | 2003-05-06 | Vertex Pharmaceuticals Incorporated | Method for synthesizing caspase inhibitors |
US6703500B2 (en) | 1998-08-19 | 2004-03-09 | Vertex Pharmaceuticals, Incorporated | Method of preparing bicyclic intermediates from piperazic acid or an ester thereof useful in the manufacture of caspase inhibitors |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB2128984B (en) * | 1982-05-12 | 1985-05-22 | Hoffmann La Roche | Diaza-bicyclic compounds |
ZA833214B (en) * | 1982-05-12 | 1983-12-28 | Hoffmann La Roche | Bicyclic compounds |
-
1999
- 1999-01-12 FR FR9900227A patent/FR2788276B1/fr not_active Expired - Fee Related
- 1999-12-10 TW TW088121699A patent/TWI222443B/zh not_active IP Right Cessation
-
2000
- 2000-01-11 ES ES00900552T patent/ES2215020T3/es not_active Expired - Lifetime
- 2000-01-11 US US09/869,950 patent/US6512111B1/en not_active Expired - Lifetime
- 2000-01-11 DK DK00900552T patent/DK1144436T3/da active
- 2000-01-11 CN CNB008048320A patent/CN1240710C/zh not_active Expired - Fee Related
- 2000-01-11 AU AU30524/00A patent/AU774752B2/en not_active Ceased
- 2000-01-11 HU HU0202665A patent/HU230062B1/hu not_active IP Right Cessation
- 2000-01-11 WO PCT/FR2000/000041 patent/WO2000042061A1/fr active IP Right Grant
- 2000-01-11 SI SI200030348T patent/SI1144436T1/xx unknown
- 2000-01-11 CA CA2359964A patent/CA2359964C/fr not_active Expired - Fee Related
- 2000-01-11 IL IL14422700A patent/IL144227A0/xx active IP Right Grant
- 2000-01-11 NZ NZ512908A patent/NZ512908A/en not_active IP Right Cessation
- 2000-01-11 DE DE60009658T patent/DE60009658T2/de not_active Expired - Lifetime
- 2000-01-11 KR KR1020017008755A patent/KR100797349B1/ko not_active IP Right Cessation
- 2000-01-11 AT AT00900552T patent/ATE263780T1/de active
- 2000-01-11 EP EP00900552A patent/EP1144436B1/fr not_active Expired - Lifetime
- 2000-01-11 JP JP2000593628A patent/JP4601826B2/ja not_active Expired - Fee Related
- 2000-01-11 PT PT00900552T patent/PT1144436E/pt unknown
- 2000-01-11 PL PL348919A patent/PL196993B1/pl unknown
- 2000-01-11 BR BRPI0007810-7A patent/BR0007810B1/pt not_active IP Right Cessation
-
2001
- 2001-07-05 ZA ZA200105550A patent/ZA200105550B/en unknown
- 2001-07-10 IL IL144227A patent/IL144227A/en not_active IP Right Cessation
- 2001-07-11 NO NO20013435A patent/NO328110B1/no not_active IP Right Cessation
-
2002
- 2002-09-18 HK HK02106828.3A patent/HK1045316B/zh not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BG101422A (en) | Benzoxazole derivatives as bronchodilating compounds | |
DE69711391T2 (de) | Verbessertes verfahren zum herstellen von geschützten 3,4-dihydroxybuttersäure estern | |
EP1338595A3 (en) | Xanthine derivatives as DPP-IV inhibitors | |
ZA955274B (en) | Compound for and method of inhibiting phosphodiesterase IV | |
DK0567271T3 (da) | Steroidderivater til behandling af prostatahypertrofi, fremgangsmåde til fremstilling heraf og anvendelser heraf | |
EA200100994A1 (ru) | 1-АМИНОТРИАЗОЛО[4,3-а]ХИНАЗОЛИН-5-ОНЫ И/ИЛИ -5-ТИОНЫ, ИНГИБИРУЮЩИЕ ФОСФОДИЭСТЕРАЗУ-IV | |
HUP9903836A2 (hu) | Új eljárás Cox-2 inhibítor hatású fenil-szubsztituált 2(5H)-furanonok előállítására | |
AT380471B (de) | Verfahren zur herstellung von neuen 2-oxoazetidin-derivate | |
AU3749495A (en) | Diazepino-indoles as phosphodiesterase iv inhibitors | |
DK1102765T3 (da) | Fremgangsmåde til syntese af (1H)-benzo[c]quinolizin-3-on-derivater | |
DE60112091D1 (de) | Verfahren zur herstellung von azacycloalkanoylaminothiazolen | |
DK1144436T3 (da) | Fremgangsmåde til fremstilling af bicykliske forbindelser og anvendelse af denne fremgangsmåde til fremstilling af en ICE-inhiberende forbindelse | |
IE781382L (en) | Indole derivatives | |
AP2001002314A0 (en) | Substituted benzolactam compounds. | |
HUP0203543A2 (hu) | Eljárás aril-triazolinonok előállítására és új intermedierek az eljáráshoz | |
CA2377233A1 (en) | Intermediates for the synthesis of benzimidazole compounds and process for the preparation thereof | |
GB9906328D0 (en) | 2-Substituted RNA preparation | |
ZA200702878B (en) | Derivatives of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)alkyl]phosphonic acid and method of making them | |
FI20011154A (fi) | Välituotteena käyttökelpoiset tiatsolo(3,2-a)atsepiinijohdannaiset ja menetelmä niiden valmistamiseksi | |
AU4527996A (en) | Trisubstituted thioxanthines | |
EA199800931A1 (ru) | Способ получения ингибиторов фосфодиэстеразы iv | |
AR029324A1 (es) | Procedimiento de preparacion de compuestos biciclicos y aplicacion de este procedimiento como etapa intermedia para la preparacion de un compuesto inhibidor de la enzima que convierte interleuquina 1-beta (ice) | |
DE69302007T2 (de) | Androst-4-en[4,5-b]-pyrrol-derivate und ein verfahren zu ihrer herstellung | |
DK159650C (da) | 1,1-diphenylpropan-1-ol-derivater, fremgangsmaade til fremstilling heraf, farmaceutiske praeparater indeholdende disse, samt fremgangsmaade til fremstilling af disse farmaceutiske praeparater | |
ES8303327A1 (es) | Un metodo para preparar derivados de 1-sulfo-2-oxoazetidina . |