HUP0203543A2 - Eljárás aril-triazolinonok előállítására és új intermedierek az eljáráshoz - Google Patents

Eljárás aril-triazolinonok előállítására és új intermedierek az eljáráshoz

Info

Publication number
HUP0203543A2
HUP0203543A2 HU0203543A HUP0203543A HUP0203543A2 HU P0203543 A2 HUP0203543 A2 HU P0203543A2 HU 0203543 A HU0203543 A HU 0203543A HU P0203543 A HUP0203543 A HU P0203543A HU P0203543 A2 HUP0203543 A2 HU P0203543A2
Authority
HU
Hungary
Prior art keywords
alkyl
amino
general formula
hydrogen
group
Prior art date
Application number
HU0203543A
Other languages
English (en)
Inventor
Jaidev S. Goudar
Original Assignee
Fmc Corp.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fmc Corp. filed Critical Fmc Corp.
Publication of HUP0203543A2 publication Critical patent/HUP0203543A2/hu
Publication of HUP0203543A3 publication Critical patent/HUP0203543A3/hu
Publication of HU228358B1 publication Critical patent/HU228358B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C257/00—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
    • C07C257/10—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
    • C07C257/22—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having nitrogen atoms of amidino groups further bound to nitrogen atoms, e.g. hydrazidines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

A találmány intermedierekként hasznosítható (I) általános képletű 1-aril-triazolinonok előállítási eljárására vonatkozik, amelynek során(i) egy (A) általános képletű amidrazont - amelynek képletében X és Yjelentése egymástól függetlenül hidrogén-, halogénatom, nitro- vagyaminocsoport; Z jelentése hidrogén-, halogénatom, alkil-,alkoxi-, nitro-, amino- vagy (alkil-szulfonil)-amino-csoport; Wjelentése -NHR általános képletű csoport, amelyben R jelentésehidrogénatom, alkil- vagy halogén-alkil-csoport; és R1 jelentésehidrogénatom, alkil-, halogén-alkil-, alkoxi-, acetil- vagyarilcsoport - legalább egy karbonilezőszerrel karbonileznek, vagy (ii)egy (A) általános képletű hidrazonoil-származékot - amelynekképletében X, Y, Z és R1 jelentése a fentiekben meghatározott; és Wjelentése halogénatom, -NCO, -OSO2CH3, -OSO2CF3 vagy -OSO2(p-CH3Ph)képletű csoport - legalább egy gyűrűképző szerrel kondenzálnak. Atalálmány kiterjed az (A) általános képletű új vegyületekre is,amelyek képletében W jelentése halogénatom, -NCO, -OSO2CH3, -OSO2CF3,-OSO2(p-CH3Ph) képletű csoport vagy -NHR általános képletű csoport,amelyben R jelentése hidrogénatom, alkil- vagy halogén-alkil-csoport;X és Y jelentése egymástól függetlenül hidrogén-, halogénatom, nitro-vagy aminocsoport; Z jelentése hidrogén-, halogénatom, alkil-,alkoxi-, nitro-, amino- vagy (alkil-szulfonil)-amino-csoport; és R1jelentése hidrogénatom, alkil-, halogén-alkil-, alkoxi-, acetil- vagyarilcsoport. Ó
HU0203543A 1999-10-13 2000-10-12 Process to prepare aryltriazolinones and novel intermediates thereto HU228358B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15924799P 1999-10-13 1999-10-13
US09/663,336 US6492527B1 (en) 1999-10-13 2000-09-18 Process to prepare aryltriazolinones and novel intermediates thereto
PCT/US2000/028240 WO2001027092A2 (en) 1999-10-13 2000-10-12 Process to prepare aryltriazolinones and novel intermediates thereto

Publications (3)

Publication Number Publication Date
HUP0203543A2 true HUP0203543A2 (hu) 2003-03-28
HUP0203543A3 HUP0203543A3 (en) 2003-04-28
HU228358B1 HU228358B1 (en) 2013-03-28

Family

ID=26855783

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0203543A HU228358B1 (en) 1999-10-13 2000-10-12 Process to prepare aryltriazolinones and novel intermediates thereto

Country Status (19)

Country Link
US (3) US6492527B1 (hu)
EP (1) EP1240149B1 (hu)
JP (1) JP4954409B2 (hu)
KR (1) KR100722041B1 (hu)
CN (1) CN100349879C (hu)
AT (1) ATE332293T1 (hu)
AU (1) AU784318B2 (hu)
BR (1) BR0014561B1 (hu)
CY (1) CY1106186T1 (hu)
CZ (1) CZ304209B6 (hu)
DE (1) DE60029245T2 (hu)
DK (1) DK1240149T3 (hu)
ES (1) ES2267577T3 (hu)
HU (1) HU228358B1 (hu)
IL (2) IL149063A0 (hu)
PL (1) PL364879A1 (hu)
PT (1) PT1240149E (hu)
TW (1) TWI289140B (hu)
WO (1) WO2001027092A2 (hu)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5167283B2 (ja) * 2008-01-10 2013-03-21 北興化学工業株式会社 フェニルトリアゾリノン類の製造法
CN106986838B (zh) * 2017-05-31 2019-11-15 江苏七洲绿色化工股份有限公司 一种丙硫菌唑的制备方法
CN107043359B (zh) * 2017-05-31 2019-08-09 江苏七洲绿色化工股份有限公司 一种丙硫菌唑中间体的制备方法
CN113072510A (zh) * 2021-03-09 2021-07-06 浙江理工大学 一种1,2,4-三氮唑-3-酮化合物的绿色制备方法

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US3879543A (en) * 1968-03-04 1975-04-22 Upjohn Co Certain benzoyl chloride phenylhydrazones as insecticides and miticides
US3870505A (en) 1969-11-07 1975-03-11 Upjohn Co Weed control with substituted phenylhydrazones
FR2105698A5 (hu) 1970-09-17 1972-04-28 Roussel Uclaf
DE2113997A1 (de) 1971-03-23 1972-10-05 Bayer Ag alpha-Acylcarbonylphenylhydrazonderivate,ein Verfahren zu ihrer Herstellung und ihre Verwendung als Insektizide,Akarizide und Fungizide
US3737533A (en) * 1971-04-28 1973-06-05 Upjohn Co Compositions and methods of combatting insects using 1'-variable-1',1'-dihalohalobenzeneazomethanes
US3935315A (en) * 1972-05-26 1976-01-27 Rhone-Poulenc S.A. Insecticidal and acaricidal phenylhydrazone derivatives
NL7307000A (hu) * 1972-05-26 1973-11-28
DE2436544A1 (de) 1973-08-02 1975-02-13 Montedison Spa Fungizid-wirksame alpha, alphadisubstituierte formylidenphenylhydrazine
US3932662A (en) * 1974-05-20 1976-01-13 The Upjohn Company Method of treating animals and formulations therefor
GB1603407A (en) * 1977-09-05 1981-11-25 Wellcome Found Hydantoin derivatives
DK501077A (da) 1976-11-17 1978-05-18 Montedison Spa Nye phosphorsyreestere afledt af 1,2,4-triazol med insekticid nematodicid og acaricid virkning og fremgangsmaade til fremstilling deraf
JPS5653662A (en) * 1979-10-08 1981-05-13 Nippon Nohyaku Co Ltd Preparation of delta2-1,2,4-triazolin-5-ones
JPS5653664A (en) * 1979-10-08 1981-05-13 Nippon Nohyaku Co Ltd Preparation of delta2-1,2,4-triazolin-5-ones
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DE3901720A1 (de) * 1989-01-21 1990-07-26 Hoechst Ag Substituierte benzo(b)pyrane, verfahren zu ihrer herstellung, ihre verwendung sowie pharmazeutische praeparate auf basis dieser verbindungen
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Also Published As

Publication number Publication date
ATE332293T1 (de) 2006-07-15
BR0014561A (pt) 2003-07-29
HU228358B1 (en) 2013-03-28
TWI289140B (en) 2007-11-01
DK1240149T3 (da) 2006-10-30
AU784318B2 (en) 2006-03-09
PL364879A1 (en) 2004-12-27
KR100722041B1 (ko) 2007-05-25
AU1081801A (en) 2001-04-23
CZ304209B6 (cs) 2014-01-08
US6992221B2 (en) 2006-01-31
IL149063A (en) 2007-05-15
CN1420874A (zh) 2003-05-28
BR0014561B1 (pt) 2012-07-24
DE60029245T2 (de) 2007-05-31
CY1106186T1 (el) 2011-06-08
PT1240149E (pt) 2006-11-30
EP1240149B1 (en) 2006-07-05
CN100349879C (zh) 2007-11-21
HUP0203543A3 (en) 2003-04-28
US20030036657A1 (en) 2003-02-20
WO2001027092A2 (en) 2001-04-19
ES2267577T3 (es) 2007-03-16
JP4954409B2 (ja) 2012-06-13
US6600049B2 (en) 2003-07-29
US6492527B1 (en) 2002-12-10
CZ20021240A3 (cs) 2002-09-11
WO2001027092A3 (en) 2001-10-25
EP1240149A2 (en) 2002-09-18
KR20020035171A (ko) 2002-05-09
US20030144528A1 (en) 2003-07-31
IL149063A0 (en) 2002-11-10
DE60029245D1 (de) 2006-08-17
JP2004500341A (ja) 2004-01-08

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Legal Events

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MM4A Lapse of definitive patent protection due to non-payment of fees