SI1144436T1 - METHOD FOR PREPARING BICYCLIC COMPOUNDS AND USE OF SAID METHOD FOR PREPARING AN INTERLEUKIN-1(Beta) CONVERSION ENZYME (ICE) INHIBITOR - Google Patents

METHOD FOR PREPARING BICYCLIC COMPOUNDS AND USE OF SAID METHOD FOR PREPARING AN INTERLEUKIN-1(Beta) CONVERSION ENZYME (ICE) INHIBITOR

Info

Publication number
SI1144436T1
SI1144436T1 SI200030348T SI200030348T SI1144436T1 SI 1144436 T1 SI1144436 T1 SI 1144436T1 SI 200030348 T SI200030348 T SI 200030348T SI 200030348 T SI200030348 T SI 200030348T SI 1144436 T1 SI1144436 T1 SI 1144436T1
Authority
SI
Slovenia
Prior art keywords
preparing
interleukin
beta
inhibitor
ice
Prior art date
Application number
SI200030348T
Other languages
English (en)
Slovenian (sl)
Inventor
Veronique Crocq
Patrick Roussel
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of SI1144436T1 publication Critical patent/SI1144436T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
SI200030348T 1999-01-12 2000-01-11 METHOD FOR PREPARING BICYCLIC COMPOUNDS AND USE OF SAID METHOD FOR PREPARING AN INTERLEUKIN-1(Beta) CONVERSION ENZYME (ICE) INHIBITOR SI1144436T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9900227A FR2788276B1 (fr) 1999-01-12 1999-01-12 NOUVEAU PROCEDE DE PREPARATION DE COMPOSES BICYCLIQUES ET L'APPLICATION DE CE PROCEDE COMME ETAPE INTERMEDIAIRE POUR LA PREPARATION D'UN COMPOSE INHIBITEUR DE L'ENZYME DE CONVERSION DE L'INTERLEUKINE 1-BETA (ice)
EP00900552A EP1144436B1 (fr) 1999-01-12 2000-01-11 Procede de preparation de composes bicycliques et l'application de ce procede pour la preparation d'un compose inhibiteur de ice
PCT/FR2000/000041 WO2000042061A1 (fr) 1999-01-12 2000-01-11 Procede de preparation de composes bicycliques et l'application de ce procede pour la preparation d'un compose inhibiteur de ice

Publications (1)

Publication Number Publication Date
SI1144436T1 true SI1144436T1 (en) 2004-06-30

Family

ID=9540778

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200030348T SI1144436T1 (en) 1999-01-12 2000-01-11 METHOD FOR PREPARING BICYCLIC COMPOUNDS AND USE OF SAID METHOD FOR PREPARING AN INTERLEUKIN-1(Beta) CONVERSION ENZYME (ICE) INHIBITOR

Country Status (24)

Country Link
US (1) US6512111B1 (xx)
EP (1) EP1144436B1 (xx)
JP (1) JP4601826B2 (xx)
KR (1) KR100797349B1 (xx)
CN (1) CN1240710C (xx)
AT (1) ATE263780T1 (xx)
AU (1) AU774752B2 (xx)
BR (1) BR0007810B1 (xx)
CA (1) CA2359964C (xx)
DE (1) DE60009658T2 (xx)
DK (1) DK1144436T3 (xx)
ES (1) ES2215020T3 (xx)
FR (1) FR2788276B1 (xx)
HK (1) HK1045316B (xx)
HU (1) HU230062B1 (xx)
IL (2) IL144227A0 (xx)
NO (1) NO328110B1 (xx)
NZ (1) NZ512908A (xx)
PL (1) PL196993B1 (xx)
PT (1) PT1144436E (xx)
SI (1) SI1144436T1 (xx)
TW (1) TWI222443B (xx)
WO (1) WO2000042061A1 (xx)
ZA (1) ZA200105550B (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6703500B2 (en) 1998-08-19 2004-03-09 Vertex Pharmaceuticals, Incorporated Method of preparing bicyclic intermediates from piperazic acid or an ester thereof useful in the manufacture of caspase inhibitors
US6559304B1 (en) 1998-08-19 2003-05-06 Vertex Pharmaceuticals Incorporated Method for synthesizing caspase inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2128984B (en) * 1982-05-12 1985-05-22 Hoffmann La Roche Diaza-bicyclic compounds
NZ204130A (en) * 1982-05-12 1986-03-14 Hoffmann La Roche Bicyclic heterocyclic compounds and pharmaceutical compositions

Also Published As

Publication number Publication date
DE60009658T2 (de) 2005-03-24
DK1144436T3 (da) 2004-08-02
CA2359964A1 (fr) 2000-07-20
PT1144436E (pt) 2004-08-31
ES2215020T3 (es) 2004-10-01
KR20010101468A (ko) 2001-11-14
ATE263780T1 (de) 2004-04-15
IL144227A0 (en) 2002-05-23
HK1045316A1 (en) 2002-11-22
AU774752B2 (en) 2004-07-08
BR0007810B1 (pt) 2011-08-23
TWI222443B (en) 2004-10-21
ZA200105550B (en) 2002-07-25
HK1045316B (zh) 2006-09-29
EP1144436B1 (fr) 2004-04-07
EP1144436A1 (fr) 2001-10-17
IL144227A (en) 2006-12-31
US6512111B1 (en) 2003-01-28
JP4601826B2 (ja) 2010-12-22
FR2788276A1 (fr) 2000-07-13
PL348919A1 (en) 2002-06-17
CA2359964C (fr) 2010-04-20
FR2788276B1 (fr) 2001-02-16
NO20013435D0 (no) 2001-07-11
BR0007810A (pt) 2001-11-06
CN1240710C (zh) 2006-02-08
NZ512908A (en) 2003-07-25
PL196993B1 (pl) 2008-02-29
JP2002534533A (ja) 2002-10-15
WO2000042061A1 (fr) 2000-07-20
AU3052400A (en) 2000-08-01
NO328110B1 (no) 2009-12-07
DE60009658D1 (de) 2004-05-13
CN1343218A (zh) 2002-04-03
HU230062B1 (hu) 2015-06-29
HUP0202665A3 (en) 2004-12-28
HUP0202665A2 (hu) 2002-12-28
KR100797349B1 (ko) 2008-01-22
NO20013435L (no) 2001-08-27

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