DK0912535T3 - Konjugater af cis-docosahexaensyre og paclitaxel - Google Patents

Konjugater af cis-docosahexaensyre og paclitaxel

Info

Publication number
DK0912535T3
DK0912535T3 DK97930990T DK97930990T DK0912535T3 DK 0912535 T3 DK0912535 T3 DK 0912535T3 DK 97930990 T DK97930990 T DK 97930990T DK 97930990 T DK97930990 T DK 97930990T DK 0912535 T3 DK0912535 T3 DK 0912535T3
Authority
DK
Denmark
Prior art keywords
conjugates
paclitaxel
cis
docosahexaenoic acid
useful
Prior art date
Application number
DK97930990T
Other languages
English (en)
Inventor
Matthews O Bradley
Victor E Shashoua
Nigel L Webb
Charles S Swindell
Original Assignee
Protarga Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Protarga Inc filed Critical Protarga Inc
Application granted granted Critical
Publication of DK0912535T3 publication Critical patent/DK0912535T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542Carboxylic acids, e.g. a fatty acid or an amino acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
DK97930990T 1996-05-22 1997-05-22 Konjugater af cis-docosahexaensyre og paclitaxel DK0912535T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/653,951 US5919815A (en) 1996-05-22 1996-05-22 Taxane compounds and compositions
PCT/US1997/008792 WO1997044336A1 (en) 1996-05-22 1997-05-22 Conjugates of cis-docosahexaenoic acid and paclitaxel

Publications (1)

Publication Number Publication Date
DK0912535T3 true DK0912535T3 (da) 2002-02-25

Family

ID=24622927

Family Applications (1)

Application Number Title Priority Date Filing Date
DK97930990T DK0912535T3 (da) 1996-05-22 1997-05-22 Konjugater af cis-docosahexaensyre og paclitaxel

Country Status (11)

Country Link
US (1) US5919815A (da)
EP (1) EP0912535B1 (da)
JP (1) JP4172725B2 (da)
AT (1) ATE208382T1 (da)
AU (1) AU720704B2 (da)
CA (1) CA2255637C (da)
DE (1) DE69708100T2 (da)
DK (1) DK0912535T3 (da)
ES (1) ES2162681T3 (da)
HK (1) HK1022301A1 (da)
WO (1) WO1997044336A1 (da)

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Also Published As

Publication number Publication date
HK1022301A1 (en) 2000-08-04
AU720704B2 (en) 2000-06-08
CA2255637A1 (en) 1997-11-27
DE69708100D1 (de) 2001-12-13
CA2255637C (en) 2005-01-04
ATE208382T1 (de) 2001-11-15
AU3473497A (en) 1997-12-09
EP0912535B1 (en) 2001-11-07
ES2162681T3 (es) 2002-01-01
JP2000511187A (ja) 2000-08-29
EP0912535A1 (en) 1999-05-06
US5919815A (en) 1999-07-06
DE69708100T2 (de) 2002-04-11
WO1997044336A1 (en) 1997-11-27
JP4172725B2 (ja) 2008-10-29

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