DK0807112T3 - Antimikrobiel heteroaromatisk ringsubstitueret phenyloxazolidinon - Google Patents

Antimikrobiel heteroaromatisk ringsubstitueret phenyloxazolidinon

Info

Publication number
DK0807112T3
DK0807112T3 DK96905168T DK96905168T DK0807112T3 DK 0807112 T3 DK0807112 T3 DK 0807112T3 DK 96905168 T DK96905168 T DK 96905168T DK 96905168 T DK96905168 T DK 96905168T DK 0807112 T3 DK0807112 T3 DK 0807112T3
Authority
DK
Denmark
Prior art keywords
optionally substituted
alkoxy
pct
acyloxy
hydroxy
Prior art date
Application number
DK96905168T
Other languages
Danish (da)
English (en)
Inventor
Douglas K Hutchinson
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of DK0807112T3 publication Critical patent/DK0807112T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
DK96905168T 1995-02-03 1996-01-29 Antimikrobiel heteroaromatisk ringsubstitueret phenyloxazolidinon DK0807112T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38427895A 1995-02-03 1995-02-03
PCT/US1996/000718 WO1996023788A1 (en) 1995-02-03 1996-01-29 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials

Publications (1)

Publication Number Publication Date
DK0807112T3 true DK0807112T3 (da) 2001-12-17

Family

ID=23516681

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96905168T DK0807112T3 (da) 1995-02-03 1996-01-29 Antimikrobiel heteroaromatisk ringsubstitueret phenyloxazolidinon

Country Status (20)

Country Link
US (1) US5910504A (no)
EP (1) EP0807112B1 (no)
JP (1) JPH10513446A (no)
KR (1) KR100441334B1 (no)
CN (1) CN1075073C (no)
AT (1) ATE205205T1 (no)
BR (1) BR9607017A (no)
CA (1) CA2208603A1 (no)
CZ (1) CZ231497A3 (no)
DE (1) DE69615002T2 (no)
DK (1) DK0807112T3 (no)
ES (1) ES2163004T3 (no)
FI (1) FI973217A0 (no)
HK (1) HK1008898A1 (no)
NO (1) NO309526B1 (no)
NZ (1) NZ302844A (no)
PL (1) PL185872B1 (no)
PT (1) PT807112E (no)
RU (1) RU2154645C2 (no)
WO (1) WO1996023788A1 (no)

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DE19750968A1 (de) * 1997-03-07 1998-09-10 Clariant Gmbh Verfahren zur Herstellung von N-Carboxyalkyl-3-fluor-4-dialkylaminoanilinen
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US6069141A (en) * 1998-02-13 2000-05-30 Pharmacia & Upjohn Company Substituted aminophenyl isoxazoline derivatives useful as antimicrobials
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US6608081B2 (en) 1999-08-12 2003-08-19 Ortho-Mcneil Pharmaceutical, Inc. Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
US6413981B1 (en) * 1999-08-12 2002-07-02 Ortho-Mcneil Pharamceutical, Inc. Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
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DE10355461A1 (de) 2003-11-27 2005-06-23 Bayer Healthcare Ag Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
DE102004062475A1 (de) * 2004-12-24 2006-07-06 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
EP1685841A1 (en) * 2005-01-31 2006-08-02 Bayer Health Care Aktiengesellschaft Prevention and treatment of thromboembolic disorders
WO2006124897A2 (en) * 2005-05-13 2006-11-23 Lexicon Genetics Incorporated Methods and compositions for improving cognition
WO2007024789A1 (en) * 2005-08-24 2007-03-01 Lexicon Genetics Incorporated Pyrrolopyridine, pyrrolopyrimidine and pyrazolopyridine compounds, compositions comprising them, and methods of their use
DE102005045518A1 (de) * 2005-09-23 2007-03-29 Bayer Healthcare Ag 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
DE102005047558A1 (de) * 2005-10-04 2008-02-07 Bayer Healthcare Ag Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
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EP2072514A1 (en) * 2007-12-17 2009-06-24 Ferrer Internacional, S.A. 1(2)H-tetrazol-5-yl-phenyl-oxazolidinones as antibacterial agents
WO2012171479A1 (zh) * 2011-06-17 2012-12-20 四川大学 噁唑烷酮类化合物及其在制备抗生素药物中的用途
EP2602248A1 (en) 2011-12-05 2013-06-12 University Of Leicester Novel pyrrole compounds
CN104364240B (zh) * 2012-06-08 2017-02-22 四川贝力克生物技术有限责任公司 一种用于预防或治疗分支杆菌疾病的药物
CN104873510B (zh) * 2014-02-28 2019-03-19 四川好医生药业集团有限公司 噁唑烷酮类化合物抗生物膜用途
CN103965183B (zh) * 2014-03-17 2017-05-03 上海应用技术学院 一种含氟噁唑烷酮类化合物及其制备方法和应用
CN105272976B (zh) * 2014-07-22 2018-11-20 四川好医生药业集团有限公司 一种噁唑烷酮类化合物
CN105399737B (zh) * 2014-09-10 2018-09-21 四川好医生药业集团有限公司 噁唑烷酮类化合物及其用途
SI3300500T1 (sl) 2015-05-20 2020-07-31 Amgen Inc. Triazolni agonisti receptorja APJ
US9988369B2 (en) 2016-05-03 2018-06-05 Amgen Inc. Heterocyclic triazole compounds as agonists of the APJ receptor
EP3541805B1 (en) 2016-11-16 2020-10-14 Amgen Inc. Heteroaryl-substituted triazoles as apj receptor agonists
EP3541810B1 (en) 2016-11-16 2020-12-23 Amgen Inc. Triazole phenyl compounds as agonists of the apj receptor
WO2018093580A1 (en) 2016-11-16 2018-05-24 Amgen Inc. Triazole pyridyl compounds as agonists of the apj receptor
US10736883B2 (en) 2016-11-16 2020-08-11 Amgen Inc. Triazole furan compounds as agonists of the APJ receptor
EP3541804A1 (en) 2016-11-16 2019-09-25 Amgen Inc. Cycloalkyl substituted triazole compounds as agonists of the apj receptor
WO2018093576A1 (en) 2016-11-16 2018-05-24 Amgen Inc. Alkyl substituted triazole compounds as agonists of the apj receptor
CN106831615B (zh) * 2017-02-15 2019-02-15 南京农业大学 一类1，2，3－三唑－5－酰胺类化合物作为农用杀菌剂的应用
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CN113372276B (zh) * 2021-05-25 2022-04-22 三峡大学 吲唑类衍生物及其应用

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Also Published As

Publication number Publication date
DE69615002D1 (de) 2001-10-11
FI973217A (fi) 1997-08-04
FI973217A0 (fi) 1997-08-04
ES2163004T3 (es) 2002-01-16
EP0807112B1 (en) 2001-09-05
US5910504A (en) 1999-06-08
AU703465B2 (en) 1999-03-25
WO1996023788A1 (en) 1996-08-08
CN1075073C (zh) 2001-11-21
PL185872B1 (pl) 2003-08-29
HK1008898A1 (en) 1999-07-23
CA2208603A1 (en) 1996-08-08
RU2154645C2 (ru) 2000-08-20
EP0807112A1 (en) 1997-11-19
KR100441334B1 (ko) 2004-10-20
ATE205205T1 (de) 2001-09-15
KR19980701908A (ko) 1998-06-25
NO973550D0 (no) 1997-08-01
NO309526B1 (no) 2001-02-12
NZ302844A (en) 1999-06-29
DE69615002T2 (de) 2002-06-13
AU4899896A (en) 1996-08-21
PT807112E (pt) 2002-02-28
JPH10513446A (ja) 1998-12-22
BR9607017A (pt) 1997-10-28
NO973550L (no) 1997-10-03
PL321663A1 (en) 1997-12-22
CN1172484A (zh) 1998-02-04
CZ231497A3 (cs) 1998-08-12

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