FI973217A0 - Heteroaromaattisella renkaalla substituoituja antimikrobiaalisia fenyylioksatsolidinoniyhdisteitä - Google Patents

Heteroaromaattisella renkaalla substituoituja antimikrobiaalisia fenyylioksatsolidinoniyhdisteitä

Info

Publication number
FI973217A0
FI973217A0 FI973217A FI973217A FI973217A0 FI 973217 A0 FI973217 A0 FI 973217A0 FI 973217 A FI973217 A FI 973217A FI 973217 A FI973217 A FI 973217A FI 973217 A0 FI973217 A0 FI 973217A0
Authority
FI
Finland
Prior art keywords
optionally substituted
alkoxy
pct
antimicrobial
acyloxy
Prior art date
Application number
FI973217A
Other languages
English (en)
Swedish (sv)
Other versions
FI973217A (fi
Inventor
Douglas K Hutchinson
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FI973217A publication Critical patent/FI973217A/fi
Publication of FI973217A0 publication Critical patent/FI973217A0/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
FI973217A 1995-02-03 1997-08-04 Heteroaromaattisella renkaalla substituoituja antimikrobiaalisia fenyylioksatsolidinoniyhdisteitä FI973217A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38427895A 1995-02-03 1995-02-03
PCT/US1996/000718 WO1996023788A1 (en) 1995-02-03 1996-01-29 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials

Publications (2)

Publication Number Publication Date
FI973217A FI973217A (fi) 1997-08-04
FI973217A0 true FI973217A0 (fi) 1997-08-04

Family

ID=23516681

Family Applications (1)

Application Number Title Priority Date Filing Date
FI973217A FI973217A0 (fi) 1995-02-03 1997-08-04 Heteroaromaattisella renkaalla substituoituja antimikrobiaalisia fenyylioksatsolidinoniyhdisteitä

Country Status (20)

Country Link
US (1) US5910504A (fi)
EP (1) EP0807112B1 (fi)
JP (1) JPH10513446A (fi)
KR (1) KR100441334B1 (fi)
CN (1) CN1075073C (fi)
AT (1) ATE205205T1 (fi)
BR (1) BR9607017A (fi)
CA (1) CA2208603A1 (fi)
CZ (1) CZ231497A3 (fi)
DE (1) DE69615002T2 (fi)
DK (1) DK0807112T3 (fi)
ES (1) ES2163004T3 (fi)
FI (1) FI973217A0 (fi)
HK (1) HK1008898A1 (fi)
NO (1) NO309526B1 (fi)
NZ (1) NZ302844A (fi)
PL (1) PL185872B1 (fi)
PT (1) PT807112E (fi)
RU (1) RU2154645C2 (fi)
WO (1) WO1996023788A1 (fi)

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US6413981B1 (en) * 1999-08-12 2002-07-02 Ortho-Mcneil Pharamceutical, Inc. Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
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US6861433B2 (en) * 2000-12-15 2005-03-01 Pharmacia & Upjohn Company Oxazolidinone photoaffinity probes
AU2002256995A1 (en) * 2001-02-07 2002-08-28 Ortho-Mcneil Pharmaceutical, Inc. Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods
DE10129725A1 (de) * 2001-06-20 2003-01-02 Bayer Ag Kombinationstherapie substituierter Oxazolidinone
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EP1685841A1 (en) * 2005-01-31 2006-08-02 Bayer Health Care Aktiengesellschaft Prevention and treatment of thromboembolic disorders
WO2006124897A2 (en) * 2005-05-13 2006-11-23 Lexicon Genetics Incorporated Methods and compositions for improving cognition
JP2009506036A (ja) * 2005-08-24 2009-02-12 レキシコン・ファーマシューティカルズ・インコーポレーテッド ピロロピリジン、ピロロピリミジンおよびピラゾロピリジン化合物、それらを含む組成物、ならびにそれらの使用方法
DE102005045518A1 (de) * 2005-09-23 2007-03-29 Bayer Healthcare Ag 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
DE102005047561A1 (de) 2005-10-04 2007-04-05 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
DE102005047558A1 (de) * 2005-10-04 2008-02-07 Bayer Healthcare Ag Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
PL1934208T3 (pl) 2005-10-04 2011-09-30 Bayer Ip Gmbh Nowa polimorficzna postać 5-chloro-N-({ (5S)-2-okso-3-[4-( 3-okso-4-morfolinylo)-fenylo]-1,3-oksazolidyn-5-ylo}-metylo)-2-tiofenokarboksamidu
US7547421B2 (en) * 2006-10-18 2009-06-16 Ecolab Inc. Apparatus and method for making a peroxycarboxylic acid
DE102006051625A1 (de) * 2006-11-02 2008-05-08 Bayer Materialscience Ag Kombinationstherapie substituierter Oxazolidinone
WO2008143649A2 (en) * 2006-12-04 2008-11-27 Dr. Reddy's Laboratories Limited Novel oxazolidinone compounds as antiinfective agents
KR100872059B1 (ko) 2007-02-21 2008-12-05 주식회사 레고켐 바이오사이언스 아미독심 또는 하이드록사마이드 기를 가지는 신규한옥사졸리디논 유도체 및 이를 함유하는 의약 조성물
EP2072514A1 (en) * 2007-12-17 2009-06-24 Ferrer Internacional, S.A. 1(2)H-tetrazol-5-yl-phenyl-oxazolidinones as antibacterial agents
WO2012171479A1 (zh) * 2011-06-17 2012-12-20 四川大学 噁唑烷酮类化合物及其在制备抗生素药物中的用途
EP2602248A1 (en) 2011-12-05 2013-06-12 University Of Leicester Novel pyrrole compounds
CN104364240B (zh) * 2012-06-08 2017-02-22 四川贝力克生物技术有限责任公司 一种用于预防或治疗分支杆菌疾病的药物
CN104873510B (zh) * 2014-02-28 2019-03-19 四川好医生药业集团有限公司 噁唑烷酮类化合物抗生物膜用途
CN103965183B (zh) * 2014-03-17 2017-05-03 上海应用技术学院 一种含氟噁唑烷酮类化合物及其制备方法和应用
CN105272976B (zh) * 2014-07-22 2018-11-20 四川好医生药业集团有限公司 一种噁唑烷酮类化合物
CN105399737B (zh) * 2014-09-10 2018-09-21 四川好医生药业集团有限公司 噁唑烷酮类化合物及其用途
PT3300500T (pt) 2015-05-20 2020-05-19 Amgen Inc Agonistas triazóis do receptor apj
US9988369B2 (en) 2016-05-03 2018-06-05 Amgen Inc. Heterocyclic triazole compounds as agonists of the APJ receptor
MA46827A (fr) 2016-11-16 2019-09-25 Amgen Inc Composés de triazole à substitution cycloalkyle en tant qu'agonistes du récepteur apj
WO2018093580A1 (en) 2016-11-16 2018-05-24 Amgen Inc. Triazole pyridyl compounds as agonists of the apj receptor
EP3541810B1 (en) 2016-11-16 2020-12-23 Amgen Inc. Triazole phenyl compounds as agonists of the apj receptor
US10736883B2 (en) 2016-11-16 2020-08-11 Amgen Inc. Triazole furan compounds as agonists of the APJ receptor
US11191762B2 (en) 2016-11-16 2021-12-07 Amgen Inc. Alkyl substituted triazole compounds as agonists of the APJ Receptor
WO2018097945A1 (en) 2016-11-16 2018-05-31 Amgen Inc. Heteroaryl-substituted triazoles as apj receptor agonists
CN106831615B (zh) * 2017-02-15 2019-02-15 南京农业大学 一类1，2，3－三唑－5－酰胺类化合物作为农用杀菌剂的应用
MA50509A (fr) 2017-11-03 2021-06-02 Amgen Inc Agonistes de triazole fusionnés du récepteur apj
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CN113372276B (zh) * 2021-05-25 2022-04-22 三峡大学 吲唑类衍生物及其应用

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Also Published As

Publication number Publication date
EP0807112B1 (en) 2001-09-05
RU2154645C2 (ru) 2000-08-20
HK1008898A1 (en) 1999-07-23
AU4899896A (en) 1996-08-21
DK0807112T3 (da) 2001-12-17
NO973550L (no) 1997-10-03
CZ231497A3 (cs) 1998-08-12
ATE205205T1 (de) 2001-09-15
NO973550D0 (no) 1997-08-01
CA2208603A1 (en) 1996-08-08
CN1172484A (zh) 1998-02-04
KR19980701908A (ko) 1998-06-25
ES2163004T3 (es) 2002-01-16
US5910504A (en) 1999-06-08
NO309526B1 (no) 2001-02-12
WO1996023788A1 (en) 1996-08-08
PL185872B1 (pl) 2003-08-29
EP0807112A1 (en) 1997-11-19
PL321663A1 (en) 1997-12-22
JPH10513446A (ja) 1998-12-22
DE69615002D1 (de) 2001-10-11
FI973217A (fi) 1997-08-04
PT807112E (pt) 2002-02-28
CN1075073C (zh) 2001-11-21
NZ302844A (en) 1999-06-29
KR100441334B1 (ko) 2004-10-20
BR9607017A (pt) 1997-10-28
AU703465B2 (en) 1999-03-25
DE69615002T2 (de) 2002-06-13

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