DK0787141T3 - Fremgangsmåde til sulfonylering, sulfenylering og phosphorylering af cykliske depsipeptider - Google Patents

Fremgangsmåde til sulfonylering, sulfenylering og phosphorylering af cykliske depsipeptider

Info

Publication number
DK0787141T3
DK0787141T3 DK95935902T DK95935902T DK0787141T3 DK 0787141 T3 DK0787141 T3 DK 0787141T3 DK 95935902 T DK95935902 T DK 95935902T DK 95935902 T DK95935902 T DK 95935902T DK 0787141 T3 DK0787141 T3 DK 0787141T3
Authority
DK
Denmark
Prior art keywords
pct
cyclic depsipeptides
sulfenylation
phosphorylation
sulfonylation
Prior art date
Application number
DK95935902T
Other languages
Danish (da)
English (en)
Inventor
Norbert Mencke
Achim Harder
Juergen Scherkenbeck
Andrew Plant
Peter Jeschke
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Application granted granted Critical
Publication of DK0787141T3 publication Critical patent/DK0787141T3/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D273/00Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6527Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK95935902T 1994-10-18 1995-10-05 Fremgangsmåde til sulfonylering, sulfenylering og phosphorylering af cykliske depsipeptider DK0787141T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4437198A DE4437198A1 (de) 1994-10-18 1994-10-18 Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden
PCT/EP1995/003926 WO1996011945A2 (fr) 1994-10-18 1995-10-05 Procede de sulfonylation, de sulfenylation et de phosphorylation de depsipeptides cycliques

Publications (1)

Publication Number Publication Date
DK0787141T3 true DK0787141T3 (da) 2000-12-11

Family

ID=6531064

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95935902T DK0787141T3 (da) 1994-10-18 1995-10-05 Fremgangsmåde til sulfonylering, sulfenylering og phosphorylering af cykliske depsipeptider

Country Status (17)

Country Link
US (1) US5874530A (fr)
EP (1) EP0787141B1 (fr)
JP (1) JPH10511341A (fr)
AT (1) ATE195952T1 (fr)
AU (1) AU698898B2 (fr)
BR (1) BR9509377A (fr)
CA (1) CA2202751A1 (fr)
CZ (1) CZ112397A3 (fr)
DE (2) DE4437198A1 (fr)
DK (1) DK0787141T3 (fr)
ES (1) ES2149378T3 (fr)
FI (1) FI971610A0 (fr)
HU (1) HU218569B (fr)
NZ (1) NZ294843A (fr)
PL (1) PL319649A1 (fr)
SK (1) SK48697A3 (fr)
WO (1) WO1996011945A2 (fr)

Families Citing this family (174)

* Cited by examiner, † Cited by third party
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US6136838A (en) * 1998-03-19 2000-10-24 Merck & Co., Inc. Sulfurpentafluorophenylpyrazoles for controlling ectoparasitic infestations
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
EP1735284A1 (fr) 2004-03-18 2006-12-27 Pfizer Limited Sulfamides n-(1-arylpyrazol-4l) et leur utilisation en tant qu'anti-parasitaires
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102008022520A1 (de) 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
DE102008030764A1 (de) * 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031284A1 (de) 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
DE102008031283A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
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WO2024100115A1 (fr) 2022-11-09 2024-05-16 Syngenta Crop Protection Ag Dérivés de pyrazole microbiocides
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DE4437198A1 (de) * 1994-10-18 1996-04-25 Bayer Ag Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden

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WO1996011945A3 (fr) 1996-07-25
WO1996011945A2 (fr) 1996-04-25
NZ294843A (en) 1998-11-25
ES2149378T3 (es) 2000-11-01
US5874530A (en) 1999-02-23
FI971610A (fi) 1997-04-16
SK48697A3 (en) 1997-11-05
HUT77019A (hu) 1998-03-02
BR9509377A (pt) 1997-11-18
DE4437198A1 (de) 1996-04-25
PL319649A1 (en) 1997-08-18
DE59508691D1 (de) 2000-10-05
AU3803895A (en) 1996-05-06
MX9702771A (es) 1997-07-31
JPH10511341A (ja) 1998-11-04
CA2202751A1 (fr) 1996-04-25
CZ112397A3 (en) 1997-07-16
ATE195952T1 (de) 2000-09-15
AU698898B2 (en) 1998-11-12
FI971610A0 (fi) 1997-04-16
EP0787141B1 (fr) 2000-08-30
HU218569B (hu) 2000-10-28
EP0787141A2 (fr) 1997-08-06

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