DK0626963T3 - Vinylen-azaindolderivater og fremgangsmåde til fremstilling deraf - Google Patents

Vinylen-azaindolderivater og fremgangsmåde til fremstilling deraf

Info

Publication number
DK0626963T3
DK0626963T3 DK94903774T DK94903774T DK0626963T3 DK 0626963 T3 DK0626963 T3 DK 0626963T3 DK 94903774 T DK94903774 T DK 94903774T DK 94903774 T DK94903774 T DK 94903774T DK 0626963 T3 DK0626963 T3 DK 0626963T3
Authority
DK
Denmark
Prior art keywords
preparation
azaindole derivatives
vinylene
vinylene azaindole
derivatives
Prior art date
Application number
DK94903774T
Other languages
Danish (da)
English (en)
Inventor
Franco Buzetti
Angelo Crugnola
Dario Ballinari
Felicita Greco
Original Assignee
Pharmacia & Upjohn Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Spa filed Critical Pharmacia & Upjohn Spa
Application granted granted Critical
Publication of DK0626963T3 publication Critical patent/DK0626963T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Steroid Compounds (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Investigating Or Analyzing Non-Biological Materials By The Use Of Chemical Means (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK94903774T 1992-12-23 1993-12-15 Vinylen-azaindolderivater og fremgangsmåde til fremstilling deraf DK0626963T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929226855A GB9226855D0 (en) 1992-12-23 1992-12-23 Vinylene-azaindole derivatives and process for their preparation
PCT/EP1993/003536 WO1994014808A1 (fr) 1992-12-23 1993-12-15 Derives vinylene-azaindoliques et leur procede de preparation

Publications (1)

Publication Number Publication Date
DK0626963T3 true DK0626963T3 (da) 1999-12-13

Family

ID=10727139

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94903774T DK0626963T3 (da) 1992-12-23 1993-12-15 Vinylen-azaindolderivater og fremgangsmåde til fremstilling deraf

Country Status (24)

Country Link
US (1) US5397787A (fr)
EP (1) EP0626963B1 (fr)
JP (1) JP3507497B2 (fr)
KR (1) KR950700296A (fr)
CN (1) CN1093707A (fr)
AT (1) ATE181074T1 (fr)
AU (1) AU670488B2 (fr)
CA (1) CA2126228A1 (fr)
DE (1) DE69325262T2 (fr)
DK (1) DK0626963T3 (fr)
ES (1) ES2134926T3 (fr)
FI (1) FI943838A0 (fr)
GB (1) GB9226855D0 (fr)
GR (1) GR3030941T3 (fr)
HU (1) HUT67431A (fr)
IL (1) IL108087A (fr)
MX (1) MX9400206A (fr)
MY (1) MY109695A (fr)
NZ (1) NZ259330A (fr)
PL (1) PL304894A1 (fr)
RU (1) RU94040390A (fr)
TW (1) TW296383B (fr)
WO (1) WO1994014808A1 (fr)
ZA (1) ZA939578B (fr)

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JPH07504208A (ja) 1995-05-11
RU94040390A (ru) 1997-05-27
JP3507497B2 (ja) 2004-03-15
KR950700296A (ko) 1995-01-16
PL304894A1 (en) 1995-01-09
ES2134926T3 (es) 1999-10-16
DE69325262T2 (de) 2000-01-20
FI943838A (fi) 1994-08-19
ZA939578B (en) 1994-08-11
ATE181074T1 (de) 1999-06-15
AU5810594A (en) 1994-07-19
GR3030941T3 (en) 1999-11-30
US5397787A (en) 1995-03-14
FI943838A0 (fi) 1994-08-19
TW296383B (fr) 1997-01-21
WO1994014808A1 (fr) 1994-07-07
AU670488B2 (en) 1996-07-18
IL108087A (en) 1997-09-30
HUT67431A (en) 1995-04-28
DE69325262D1 (de) 1999-07-15
NZ259330A (en) 1995-12-21
CN1093707A (zh) 1994-10-19
IL108087A0 (en) 1994-04-12
HU9401950D0 (en) 1994-09-28
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MX9400206A (es) 1994-07-29

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