DK0603251T3 - 1-substituerede 1H-imidazol(4,5-c)quinolin-4-aminer, mellemprodukter og farmaceutiske sammensætninger - Google Patents

1-substituerede 1H-imidazol(4,5-c)quinolin-4-aminer, mellemprodukter og farmaceutiske sammensætninger

Info

Publication number
DK0603251T3
DK0603251T3 DK92919122T DK92919122T DK0603251T3 DK 0603251 T3 DK0603251 T3 DK 0603251T3 DK 92919122 T DK92919122 T DK 92919122T DK 92919122 T DK92919122 T DK 92919122T DK 0603251 T3 DK0603251 T3 DK 0603251T3
Authority
DK
Denmark
Prior art keywords
intermediates
amines
substituted
pharmaceutical compositions
quinoline
Prior art date
Application number
DK92919122T
Other languages
English (en)
Inventor
John F Gerster
Original Assignee
Minnesota Mining & Mfg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Minnesota Mining & Mfg filed Critical Minnesota Mining & Mfg
Application granted granted Critical
Publication of DK0603251T3 publication Critical patent/DK0603251T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/052—Imidazole radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK92919122T 1991-09-04 1992-08-26 1-substituerede 1H-imidazol(4,5-c)quinolin-4-aminer, mellemprodukter og farmaceutiske sammensætninger DK0603251T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/754,610 US5268376A (en) 1991-09-04 1991-09-04 1-substituted 1H-imidazo[4,5-c]quinolin-4-amines
PCT/US1992/007226 WO1993005042A1 (en) 1991-09-04 1992-08-26 1-substituted 1h-imidazo(4,5-c)quinolin-4-amines; intermediate and pharmaceutical compositions

Publications (1)

Publication Number Publication Date
DK0603251T3 true DK0603251T3 (da) 2001-01-02

Family

ID=25035560

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92919122T DK0603251T3 (da) 1991-09-04 1992-08-26 1-substituerede 1H-imidazol(4,5-c)quinolin-4-aminer, mellemprodukter og farmaceutiske sammensætninger

Country Status (18)

Country Link
US (4) US5268376A (da)
EP (1) EP0603251B1 (da)
JP (1) JP3315983B2 (da)
KR (1) KR100233313B1 (da)
AT (1) ATE197050T1 (da)
AU (1) AU2514792A (da)
CA (1) CA2116782C (da)
CZ (1) CZ281726B6 (da)
DE (1) DE69231522T2 (da)
DK (1) DK0603251T3 (da)
ES (1) ES2150918T3 (da)
HU (4) HU223947B1 (da)
IL (1) IL102951A (da)
MX (1) MX9205046A (da)
NZ (1) NZ244075A (da)
PH (1) PH30132A (da)
WO (1) WO1993005042A1 (da)
ZA (1) ZA926456B (da)

Families Citing this family (266)

* Cited by examiner, † Cited by third party
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