DE69232878D1 - Zwischenprodukte zur Herstellung von 1-substituierten, 2-substituierten-1H-Imidazo[4,5-c]Chinolin-4-Aminen - Google Patents

Zwischenprodukte zur Herstellung von 1-substituierten, 2-substituierten-1H-Imidazo[4,5-c]Chinolin-4-Aminen

Info

Publication number
DE69232878D1
DE69232878D1 DE69232878T DE69232878T DE69232878D1 DE 69232878 D1 DE69232878 D1 DE 69232878D1 DE 69232878 T DE69232878 T DE 69232878T DE 69232878 T DE69232878 T DE 69232878T DE 69232878 D1 DE69232878 D1 DE 69232878D1
Authority
DE
Germany
Prior art keywords
substituted
imidazo
intermediates
amines
quinoline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69232878T
Other languages
English (en)
Other versions
DE69232878T2 (de
Inventor
John F Gerster
Stephen L Crooks
Kyle J Lindstrom
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
3M Co
Original Assignee
Minnesota Mining and Manufacturing Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Minnesota Mining and Manufacturing Co filed Critical Minnesota Mining and Manufacturing Co
Application granted granted Critical
Publication of DE69232878D1 publication Critical patent/DE69232878D1/de
Publication of DE69232878T2 publication Critical patent/DE69232878T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Lubricants (AREA)
DE69232878T 1991-03-01 1992-02-20 Zwischenprodukte zur Herstellung von 1-substituierten, 2-substituierten-1H-Imidazo[4,5-c]Chinolin-4-Aminen Expired - Fee Related DE69232878T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US66292691A 1991-03-01 1991-03-01
US68732691A 1991-04-18 1991-04-18

Publications (2)

Publication Number Publication Date
DE69232878D1 true DE69232878D1 (de) 2003-01-30
DE69232878T2 DE69232878T2 (de) 2003-11-20

Family

ID=27098631

Family Applications (2)

Application Number Title Priority Date Filing Date
DE69229114T Expired - Lifetime DE69229114T2 (de) 1991-03-01 1992-02-20 1,2-substituierte 1h-imidazo[4,5-c]chinolin-4-amine
DE69232878T Expired - Fee Related DE69232878T2 (de) 1991-03-01 1992-02-20 Zwischenprodukte zur Herstellung von 1-substituierten, 2-substituierten-1H-Imidazo[4,5-c]Chinolin-4-Aminen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE69229114T Expired - Lifetime DE69229114T2 (de) 1991-03-01 1992-02-20 1,2-substituierte 1h-imidazo[4,5-c]chinolin-4-amine

Country Status (18)

Country Link
EP (2) EP0582581B1 (de)
JP (1) JP2955019B2 (de)
AT (2) ATE179711T1 (de)
AU (2) AU658621B2 (de)
CA (2) CA2104782C (de)
CZ (1) CZ285050B6 (de)
DE (2) DE69229114T2 (de)
DK (2) DK0872478T3 (de)
ES (2) ES2186034T3 (de)
HU (5) HU222111B1 (de)
IE (1) IE920605A1 (de)
IL (2) IL114570A (de)
NO (1) NO303729B1 (de)
NZ (1) NZ241784A (de)
PH (1) PH31614A (de)
SG (2) SG46492A1 (de)
UA (1) UA32546C2 (de)
WO (1) WO1992015582A1 (de)

Families Citing this family (87)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5266575A (en) * 1991-11-06 1993-11-30 Minnesota Mining And Manufacturing Company 2-ethyl 1H-imidazo[4,5-ciquinolin-4-amines
US5395937A (en) * 1993-01-29 1995-03-07 Minnesota Mining And Manufacturing Company Process for preparing quinoline amines
US5648516A (en) * 1994-07-20 1997-07-15 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
US5352784A (en) * 1993-07-15 1994-10-04 Minnesota Mining And Manufacturing Company Fused cycloalkylimidazopyridines
JPH09500128A (ja) * 1993-07-15 1997-01-07 ミネソタ マイニング アンド マニュファクチャリング カンパニー イミダゾ〔４，５−ｃ〕ピリジン−４−アミン
US5482936A (en) * 1995-01-12 1996-01-09 Minnesota Mining And Manufacturing Company Imidazo[4,5-C]quinoline amines
US6133547A (en) * 1996-09-05 2000-10-17 Medtronic, Inc. Distributed activator for a two-dimensional shape memory alloy
US5939090A (en) * 1996-12-03 1999-08-17 3M Innovative Properties Company Gel formulations for topical drug delivery
JPH10298181A (ja) * 1997-04-25 1998-11-10 Sumitomo Pharmaceut Co Ltd タイプ２ヘルパーｔ細胞選択的免疫応答抑制剤
EP1541572A1 (de) * 2000-12-08 2005-06-15 3M Innovative Properties Company Thioether substituierte Imidazochinoline
UA74852C2 (en) * 2000-12-08 2006-02-15 3M Innovative Properties Co Urea-substituted imidazoquinoline ethers
US6664264B2 (en) * 2000-12-08 2003-12-16 3M Innovative Properties Company Thioether substituted imidazoquinolines
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IL73534A (en) * 1983-11-18 1990-12-23 Riker Laboratories Inc 1h-imidazo(4,5-c)quinoline-4-amines,their preparation and pharmaceutical compositions containing certain such compounds
CA1271477A (en) * 1983-11-18 1990-07-10 John F. Gerster 1h-imidazo[4,5-c]quinolin-4-amines
DK0385630T3 (da) * 1989-02-27 1997-05-12 Riker Laboratories Inc 1H-imidazo(4,5-c)quinolin-4-aminer som antivirale midler

Also Published As

Publication number Publication date
NO933069D0 (no) 1993-08-27
ES2186034T3 (es) 2003-05-01
CZ285050B6 (cs) 1999-05-12
EP0872478A3 (de) 1998-11-04
ES2131070T3 (es) 1999-07-16
CA2104782C (en) 2001-08-07
NO303729B1 (no) 1998-08-24
IE990988A1 (en) 2000-12-13
DK0872478T3 (da) 2003-03-31
IL101110A (en) 1995-12-08
HU222111B1 (hu) 2003-04-28
DK0582581T3 (da) 1999-11-08
DE69229114T2 (de) 1999-11-04
EP0582581A1 (de) 1994-02-16
HU222251B1 (hu) 2003-05-28
SG70625A1 (en) 2000-02-22
AU658621B2 (en) 1995-04-27
JP2955019B2 (ja) 1999-10-04
HU222247B1 (hu) 2003-05-28
SG46492A1 (en) 1998-02-20
HU9701089D0 (en) 1997-08-28
NZ241784A (en) 1995-06-27
HU9701083D0 (en) 1997-08-28
ATE229943T1 (de) 2003-01-15
HUT67026A (en) 1995-01-30
DE69229114D1 (de) 1999-06-10
CZ178893A3 (en) 1995-10-18
HU9701084D0 (en) 1997-08-28
WO1992015582A1 (en) 1992-09-17
IL114570A0 (en) 1995-11-27
CA2104782A1 (en) 1992-09-02
EP0582581B1 (de) 1999-05-06
AU2715795A (en) 1995-09-21
PH31614A (en) 1999-01-12
UA32546C2 (uk) 2001-02-15
IL101110A0 (en) 1992-11-15
HU211242A9 (en) 1995-11-28
CA2289219A1 (en) 1992-09-02
ATE179711T1 (de) 1999-05-15
IE920605A1 (en) 1992-09-09
CA2289219C (en) 2003-05-20
EP0872478A2 (de) 1998-10-21
DE69232878T2 (de) 2003-11-20
HU222250B1 (hu) 2003-05-28
HU9302457D0 (en) 1993-11-29
AU1566992A (en) 1992-10-06
AU673309B2 (en) 1996-10-31
EP0872478B1 (de) 2002-12-18
JPH06504789A (ja) 1994-06-02
NO933069L (no) 1993-11-01
IL114570A (en) 1996-10-31

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