ATE203537T1 - Pyrazol(1,5-a)pyrimidin derivate - Google Patents

Pyrazol(1,5-a)pyrimidin derivate

Info

Publication number
ATE203537T1
ATE203537T1 AT96908369T AT96908369T ATE203537T1 AT E203537 T1 ATE203537 T1 AT E203537T1 AT 96908369 T AT96908369 T AT 96908369T AT 96908369 T AT96908369 T AT 96908369T AT E203537 T1 ATE203537 T1 AT E203537T1
Authority
AT
Austria
Prior art keywords
alkyl
lower alkyl
pyrazole
substituted
pyridyl
Prior art date
Application number
AT96908369T
Other languages
English (en)
Inventor
Makoto Inoue
Takashi Okamura
Yasuo Shoji
Kinji Hashimoto
Masayuki Ohara
Tsuneo Yasuda
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Application granted granted Critical
Publication of ATE203537T1 publication Critical patent/ATE203537T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT96908369T 1995-04-10 1996-04-05 Pyrazol(1,5-a)pyrimidin derivate ATE203537T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP8399095 1995-04-10
JP23642795 1995-09-14
PCT/JP1996/000955 WO1996032394A1 (fr) 1995-04-10 1996-04-05 DERIVES DE PYRAZOLO[1,5-a]PYRIMIDINE

Publications (1)

Publication Number Publication Date
ATE203537T1 true ATE203537T1 (de) 2001-08-15

Family

ID=26425023

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96908369T ATE203537T1 (de) 1995-04-10 1996-04-05 Pyrazol(1,5-a)pyrimidin derivate

Country Status (11)

Country Link
US (1) US5985882A (de)
EP (1) EP0820997B1 (de)
KR (1) KR100271998B1 (de)
CN (1) CN1066450C (de)
AT (1) ATE203537T1 (de)
AU (1) AU691413B2 (de)
CA (1) CA2217728C (de)
DE (1) DE69614102T2 (de)
ES (1) ES2159729T3 (de)
TW (1) TW399054B (de)
WO (1) WO1996032394A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6664261B2 (en) * 1996-02-07 2003-12-16 Neurocrine Biosciences, Inc. Pyrazolopyrimidines as CRF receptor antagonists
WO1999059998A1 (fr) * 1998-05-19 1999-11-25 Otsuka Pharmaceutical Factory, Inc. DERIVES DE PYRAZOLO[1,5-a]PYRIMIDINE
US6245759B1 (en) 1999-03-11 2001-06-12 Merck & Co., Inc. Tyrosine kinase inhibitors
WO2003037900A2 (en) * 2001-11-01 2003-05-08 Icagen, Inc. Pyrazolopyrimidines
CN112921405B (zh) * 2019-12-05 2023-06-27 成都先导药物开发股份有限公司 一种合成On-DNA吡唑并[1,5-a]嘧啶化合物的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6157587A (ja) * 1984-08-29 1986-03-24 Shionogi & Co Ltd 縮合複素環誘導体および抗潰瘍剤
JPH05125079A (ja) * 1991-11-05 1993-05-21 Otsuka Pharmaceut Factory Inc ピラゾロ[1,5−aピリミジン誘導体
JP3252189B2 (ja) * 1994-06-21 2002-01-28 株式会社大塚製薬工場 ピラゾロ〔1,5−a〕ピリミジン誘導体
JP4125079B2 (ja) * 2002-09-06 2008-07-23 キヤノン株式会社 光量調節装置および光学機器

Also Published As

Publication number Publication date
CN1181082A (zh) 1998-05-06
DE69614102T2 (de) 2002-03-21
DE69614102D1 (de) 2001-08-30
CA2217728A1 (en) 1996-10-17
EP0820997B1 (de) 2001-07-25
US5985882A (en) 1999-11-16
AU5162996A (en) 1996-10-30
CA2217728C (en) 2001-09-11
EP0820997A1 (de) 1998-01-28
CN1066450C (zh) 2001-05-30
WO1996032394A1 (fr) 1996-10-17
AU691413B2 (en) 1998-05-14
KR100271998B1 (ko) 2001-02-01
TW399054B (en) 2000-07-21
EP0820997A4 (de) 1998-08-12
KR19980703766A (ko) 1998-12-05
ES2159729T3 (es) 2001-10-16

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Legal Events

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