EA200400413A1 - 3-замещённые пиразолы с инсектицидными и акарицидными свойствами - Google Patents
3-замещённые пиразолы с инсектицидными и акарицидными свойствамиInfo
- Publication number
- EA200400413A1 EA200400413A1 EA200400413A EA200400413A EA200400413A1 EA 200400413 A1 EA200400413 A1 EA 200400413A1 EA 200400413 A EA200400413 A EA 200400413A EA 200400413 A EA200400413 A EA 200400413A EA 200400413 A1 EA200400413 A1 EA 200400413A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- alkyl
- alkoxycarbonyl
- halogen
- alkenyl
- alkoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/28—Two oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
- C07D231/40—Acylated on said nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
Abstract
Соединения формулы Iв которой переменные параметры и индексы имеют следующие значения:R- водород, галоген, C-C-алкил, C-C-галоалкил, C-C-алкенил, C-C-галоалкенил, C-C-алкилтио, C-C-алкокси-C-C-алкил, C-C-алкилтио-C-C-алкил или фенил, который является незамещенным или замещенным 1-3 группами R; R- галоген, нитро, циано, C-C-алкил, C-C-галоалкил, C-C-алкилтио, C-C-галоалкилтио, C-C-алкокси или C-C-галоалкокси;Rводород, галоген, C-C-алкил, C-C-галоалкил, C-C-алкенил, C-C-галоалкенил или фенил, который является незамещенным или замещенным 1-3 группами R;A водород, гидрокси, циано, нитро галоген, родано, C-C-алкокси, C-C-галоалкокси, C-C-алкенилокси, C-C-алкилтио, C-C-галоалкилтио, C-C-алкилсульфинил, C-C-алкилсульфонил, аминотиокарбонил, гидроксикарбонил, C-C-алкоксикарбонил, аминокарбонил;B - водород, гидрокси, амино, циано, нитро галоген, C-C-алкил, незамещенный или замещенный 1-3 группами, выбранными из галогена и циано; C-C-алкокси, незамещенный или замещенный 1-3 группами, выбранными из галогена, циано, C-C-алкенила и C-C-алкоксикарбонил-C-C-алкенила; C-C-алкенил, незамещенный или замещенный 1-3 группами, выбранными из галогена и циано; C-C-алкенилокси, C-C-алкилтио, C-C-галоалкилтио, C-C-алкокситиокарбонилтио, C-C-алкоксикарбонил-C-C-алкокси, C-C-алкоксикарбонил-C-C-алкилтио, C-C-алкилсульфинил, C-C-алкилсульфонил, аминотиокарбонил, NRR, N=CHORили N=CHNR;R, R, каждый независимо, представляют собой водород, C-C-алкил, C-C-алкоксикарбонил-C-C-алкил, [(C-C-алкоксикарбонил)(C-C-алкенил)]C-C-алкил, C-C-алкоксикарбонил-C-C-алкенил, C-C-алкилкарбонил, C-C-циклоалкилкарбонил, C-C-алкиламинокарбонил, ди(C-C-алкил)аминокарбонил, C-C-алкоксикарбонил, C-C-алкоксиаминосульфонил или ди(C-C-алкокси)аминосульфонил;R- C-C-алкил, C-C-галоалкил или фенил-C-C-алкил;Q - водород, нитро, галоген, C-C-галоалкил, C-C-алкиламино, ди(C-C)алкиламино, C-C-алкокси, C-C-галоалкокси, C-C-алкенилокси;X - водород, галоген, C-C-галоалкил,
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US32463301P | 2001-09-25 | 2001-09-25 | |
| PCT/EP2002/010719 WO2003029222A1 (en) | 2001-09-25 | 2002-09-25 | Insecticidal and acaricidal 3-substituted pyrazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA200400413A1 true EA200400413A1 (ru) | 2004-08-26 |
| EA007969B1 EA007969B1 (ru) | 2007-02-27 |
Family
ID=23264427
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA200400413A EA007969B1 (ru) | 2001-09-25 | 2002-09-25 | 3-замещённые пиразолы с инсектицидными и акарицидными свойствами |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20040260097A1 (ru) |
| EP (1) | EP1432688A1 (ru) |
| JP (1) | JP2005512969A (ru) |
| KR (1) | KR20040035846A (ru) |
| CN (1) | CN1305857C (ru) |
| AR (1) | AR036631A1 (ru) |
| BR (1) | BR0212385A (ru) |
| CA (1) | CA2460906A1 (ru) |
| EA (1) | EA007969B1 (ru) |
| HU (1) | HUP0402238A3 (ru) |
| IL (1) | IL160444A0 (ru) |
| MX (1) | MXPA04002040A (ru) |
| PL (1) | PL370353A1 (ru) |
| UA (1) | UA79758C2 (ru) |
| WO (1) | WO2003029222A1 (ru) |
| ZA (1) | ZA200402932B (ru) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2514004C1 (ru) * | 2012-10-25 | 2014-04-27 | Государственное научное учреждение Курский научно-исследовательский институт агропромышленного производства Россельхозакадемии | Способ получения комплексного препарата с иммунометаболической и антгельминтной активностью |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004196795A (ja) * | 2002-12-16 | 2004-07-15 | Wyeth | 外部寄生虫駆除剤としてのｎ−フェニル−３−シクロプロピルピラゾール−４−カルボニトリル |
| FR2848780B1 (fr) * | 2002-12-19 | 2005-05-13 | Solvay | Utilisation d'une poudre acaricide |
| GB0905365D0 (en) | 2009-03-27 | 2009-05-13 | Norbrook Lab Ltd | A topical parasiticide composition |
| EP3068385A4 (en) * | 2013-08-15 | 2017-08-02 | Sylleta Inc. | Compositions and methods for control of marine ectoparasites |
| ES2870038T3 (es) | 2015-12-16 | 2021-10-26 | Nippon Soda Co | Compuesto de arilazol y agente de control de plagas |
| WO2023174397A1 (en) * | 2022-03-18 | 2023-09-21 | Insilico Medicine Ip Limited | Pyrazole membrane-associated tyrosine-and threonine-specific cdc2-inhibitory kinase (pkmyt1) inhibitors and uses thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3509567A1 (de) * | 1985-03-16 | 1986-09-18 | Bayer Ag, 5090 Leverkusen | Herbizide und insektizide mittel auf basis von pyrazolderivaten |
| GB8531485D0 (en) * | 1985-12-20 | 1986-02-05 | May & Baker Ltd | Compositions of matter |
| US5232940A (en) * | 1985-12-20 | 1993-08-03 | Hatton Leslie R | Derivatives of N-phenylpyrazoles |
| US6114334A (en) * | 1995-07-13 | 2000-09-05 | Knoll Aktiengesellschaft | Piperazine derivatives as therapeutic agents |
| DE69627281T2 (de) * | 1995-12-19 | 2003-11-13 | Bayer Cropscience Sa | Neue 1-Aryl Pyrazol Derivate und ihre Verwendung als Schädlingsbekämpfungsmittel |
| US6531477B1 (en) * | 1998-10-13 | 2003-03-11 | Dupont Pharmaceuticals Company | 6-substituted pyrazolo [3,4-d] pyrimidin-4-ones useful as cyclin dependent kinase inhibitors |
-
2002
- 2002-09-25 HU HU0402238A patent/HUP0402238A3/hu unknown
- 2002-09-25 US US10/490,369 patent/US20040260097A1/en not_active Abandoned
- 2002-09-25 BR BR0212385-1A patent/BR0212385A/pt not_active IP Right Cessation
- 2002-09-25 JP JP2003532472A patent/JP2005512969A/ja not_active Withdrawn
- 2002-09-25 EA EA200400413A patent/EA007969B1/ru not_active IP Right Cessation
- 2002-09-25 IL IL16044402A patent/IL160444A0/xx unknown
- 2002-09-25 PL PL02370353A patent/PL370353A1/xx not_active Application Discontinuation
- 2002-09-25 AR ARP020103615A patent/AR036631A1/es not_active Application Discontinuation
- 2002-09-25 WO PCT/EP2002/010719 patent/WO2003029222A1/en not_active Application Discontinuation
- 2002-09-25 KR KR10-2004-7004081A patent/KR20040035846A/ko not_active Application Discontinuation
- 2002-09-25 EP EP02777196A patent/EP1432688A1/en not_active Withdrawn
- 2002-09-25 CA CA002460906A patent/CA2460906A1/en not_active Abandoned
- 2002-09-25 MX MXPA04002040A patent/MXPA04002040A/es unknown
- 2002-09-25 UA UA20040403076A patent/UA79758C2/uk unknown
- 2002-09-25 CN CNB028187547A patent/CN1305857C/zh not_active Expired - Fee Related
-
2004
- 2004-04-19 ZA ZA200402932A patent/ZA200402932B/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2514004C1 (ru) * | 2012-10-25 | 2014-04-27 | Государственное научное учреждение Курский научно-исследовательский институт агропромышленного производства Россельхозакадемии | Способ получения комплексного препарата с иммунометаболической и антгельминтной активностью |
Also Published As
| Publication number | Publication date |
|---|---|
| JP2005512969A (ja) | 2005-05-12 |
| AR036631A1 (es) | 2004-09-22 |
| WO2003029222A1 (en) | 2003-04-10 |
| KR20040035846A (ko) | 2004-04-29 |
| MXPA04002040A (es) | 2004-06-07 |
| EA007969B1 (ru) | 2007-02-27 |
| UA79758C2 (en) | 2007-07-25 |
| CN1305857C (zh) | 2007-03-21 |
| IL160444A0 (en) | 2004-07-25 |
| PL370353A1 (en) | 2005-05-16 |
| CA2460906A1 (en) | 2003-04-10 |
| HUP0402238A2 (hu) | 2005-02-28 |
| US20040260097A1 (en) | 2004-12-23 |
| CN1558902A (zh) | 2004-12-29 |
| HUP0402238A3 (en) | 2008-02-28 |
| EP1432688A1 (en) | 2004-06-30 |
| BR0212385A (pt) | 2004-08-17 |
| ZA200402932B (en) | 2005-04-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): BY RU |