DE60127002D1 - Pharmazeutische zusammensetzung - Google Patents

Pharmazeutische zusammensetzung

Info

Publication number
DE60127002D1
DE60127002D1 DE60127002T DE60127002T DE60127002D1 DE 60127002 D1 DE60127002 D1 DE 60127002D1 DE 60127002 T DE60127002 T DE 60127002T DE 60127002 T DE60127002 T DE 60127002T DE 60127002 D1 DE60127002 D1 DE 60127002D1
Authority
DE
Germany
Prior art keywords
pharmaceutical composition
pharmaceutical
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60127002T
Other languages
English (en)
Other versions
DE60127002T2 (de
Inventor
Giuseppe Alvaro
Fabio Romano Di
Paolo Maragni
Marisa Tampieri
Maria Elvira Tranquillini
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of DE60127002D1 publication Critical patent/DE60127002D1/de
Application granted granted Critical
Publication of DE60127002T2 publication Critical patent/DE60127002T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36—Opioid-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE60127002T 2000-10-17 2001-10-12 Pharmazeutische zusammensetzung Expired - Lifetime DE60127002T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0025354 2000-10-17
GBGB0025354.2A GB0025354D0 (en) 2000-10-17 2000-10-17 Chemical compounds

Publications (2)

Publication Number Publication Date
DE60127002D1 true DE60127002D1 (de) 2007-04-12
DE60127002T2 DE60127002T2 (de) 2007-10-31

Family

ID=9901397

Family Applications (3)

Application Number Title Priority Date Filing Date
DE60127002T Expired - Lifetime DE60127002T2 (de) 2000-10-17 2001-10-12 Pharmazeutische zusammensetzung
DE60142197T Expired - Lifetime DE60142197D1 (de) 2000-10-17 2001-10-12 Pharmazeutische Zusammensetzung
DE60106287T Expired - Lifetime DE60106287T2 (de) 2000-10-17 2001-10-12 Chemische verbindungen

Family Applications After (2)

Application Number Title Priority Date Filing Date
DE60142197T Expired - Lifetime DE60142197D1 (de) 2000-10-17 2001-10-12 Pharmazeutische Zusammensetzung
DE60106287T Expired - Lifetime DE60106287T2 (de) 2000-10-17 2001-10-12 Chemische verbindungen

Country Status (29)

Country Link
US (5) US7119092B2 (de)
EP (4) EP1524266B1 (de)
JP (1) JP3940359B2 (de)
KR (1) KR100847414B1 (de)
CN (1) CN1231468C (de)
AR (1) AR034268A1 (de)
AT (3) ATE468324T1 (de)
AU (4) AU9572301A (de)
BR (1) BR0114637A (de)
CA (1) CA2425876C (de)
CY (1) CY1107634T1 (de)
CZ (1) CZ299824B6 (de)
DE (3) DE60127002T2 (de)
DK (2) DK1326832T3 (de)
ES (3) ES2346108T3 (de)
GB (1) GB0025354D0 (de)
HK (2) HK1058788A1 (de)
HU (1) HU228146B1 (de)
IL (3) IL155165A0 (de)
MX (1) MXPA03003536A (de)
MY (1) MY124957A (de)
NO (1) NO324468B1 (de)
NZ (1) NZ525091A (de)
PL (1) PL203071B1 (de)
PT (2) PT1524266E (de)
SI (2) SI1326832T1 (de)
TW (1) TWI299730B (de)
WO (1) WO2002032867A1 (de)
ZA (1) ZA200302801B (de)

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Also Published As

Publication number Publication date
DE60142197D1 (de) 2010-07-01
KR20030036932A (ko) 2003-05-09
TWI299730B (en) 2008-08-11
MXPA03003536A (es) 2003-08-07
DK1524266T3 (da) 2007-06-25
US20050137208A1 (en) 2005-06-23
PL203071B1 (pl) 2009-08-31
ZA200302801B (en) 2004-04-21
US20080021041A1 (en) 2008-01-24
HUP0301459A2 (en) 2006-09-28
DE60106287T2 (de) 2006-02-23
CA2425876A1 (en) 2002-04-25
EP1524266B1 (de) 2007-02-28
IL155165A0 (en) 2003-10-31
PL361180A1 (en) 2004-09-20
IL191486A0 (en) 2008-11-03
US20040014770A1 (en) 2004-01-22
EP1921064A1 (de) 2008-05-14
BR0114637A (pt) 2003-09-30
US7648990B2 (en) 2010-01-19
ES2282794T3 (es) 2007-10-16
EP1524266A1 (de) 2005-04-20
CN1231468C (zh) 2005-12-14
PT1326832E (pt) 2005-01-31
IL155165A (en) 2008-11-26
JP3940359B2 (ja) 2007-07-04
CN1483025A (zh) 2004-03-17
US20100081667A1 (en) 2010-04-01
CZ299824B6 (cs) 2008-12-03
AU9572301A (en) 2002-04-29
CZ20031082A3 (cs) 2004-08-18
AU2001295723B2 (en) 2005-05-26
ATE468324T1 (de) 2010-06-15
KR100847414B1 (ko) 2008-07-18
US20060142302A1 (en) 2006-06-29
EP1752449A1 (de) 2007-02-14
DK1326832T3 (da) 2005-01-31
NZ525091A (en) 2005-04-29
HUP0301459A3 (en) 2007-11-28
SI1326832T1 (en) 2005-02-28
NO20031561D0 (no) 2003-04-07
AU2005204234B2 (en) 2009-05-07
ATE278669T1 (de) 2004-10-15
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NO324468B1 (no) 2007-10-22
AR034268A1 (es) 2004-02-18
AU2005204234A1 (en) 2005-09-15
AU2009201407A1 (en) 2009-05-07
PT1524266E (pt) 2007-05-31
ES2346108T3 (es) 2010-10-08
CA2425876C (en) 2009-07-07
MY124957A (en) 2006-07-31
SI1524266T1 (sl) 2007-08-31
EP1921064B1 (de) 2010-05-19
EP1326832A1 (de) 2003-07-16
US7119092B2 (en) 2006-10-10
US7060702B2 (en) 2006-06-13
GB0025354D0 (en) 2000-11-29
AU2009201407B2 (en) 2011-12-15
DE60106287D1 (de) 2004-11-11
HK1075889A1 (en) 2005-12-30
WO2002032867A1 (en) 2002-04-25
ATE355271T1 (de) 2006-03-15
JP2004511544A (ja) 2004-04-15
EP1326832B1 (de) 2004-10-06
DE60127002T2 (de) 2007-10-31
US7294630B2 (en) 2007-11-13
HK1058788A1 (en) 2004-06-04
NO20031561L (no) 2003-06-14
ES2227287T3 (es) 2005-04-01
CY1107634T1 (el) 2013-04-18

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