ATE278669T1 - Chemische verbindungen - Google Patents

Chemische verbindungen

Info

Publication number
ATE278669T1
ATE278669T1 AT01976453T AT01976453T ATE278669T1 AT E278669 T1 ATE278669 T1 AT E278669T1 AT 01976453 T AT01976453 T AT 01976453T AT 01976453 T AT01976453 T AT 01976453T AT E278669 T1 ATE278669 T1 AT E278669T1
Authority
AT
Austria
Prior art keywords
chemical compounds
compounds
chemical
Prior art date
Application number
AT01976453T
Other languages
English (en)
Inventor
Giuseppe Alvaro
Fabio Romano Di
Paolo Maragni
Marsia Tampieri
Maria Tranquillini
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE278669T1 publication Critical patent/ATE278669T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36—Opioid-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Hospice & Palliative Care (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT01976453T 2000-10-17 2001-10-12 Chemische verbindungen ATE278669T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0025354.2A GB0025354D0 (en) 2000-10-17 2000-10-17 Chemical compounds
PCT/GB2001/004580 WO2002032867A1 (en) 2000-10-17 2001-10-12 Chemical compounds

Publications (1)

Publication Number Publication Date
ATE278669T1 true ATE278669T1 (de) 2004-10-15

Family

ID=9901397

Family Applications (3)

Application Number Title Priority Date Filing Date
AT01976453T ATE278669T1 (de) 2000-10-17 2001-10-12 Chemische verbindungen
AT08151841T ATE468324T1 (de) 2000-10-17 2001-10-12 Pharmazeutische zusammensetzung
AT04077714T ATE355271T1 (de) 2000-10-17 2001-10-12 Pharmazeutische zusammensetzung

Family Applications After (2)

Application Number Title Priority Date Filing Date
AT08151841T ATE468324T1 (de) 2000-10-17 2001-10-12 Pharmazeutische zusammensetzung
AT04077714T ATE355271T1 (de) 2000-10-17 2001-10-12 Pharmazeutische zusammensetzung

Country Status (29)

Country Link
US (5) US7119092B2 (de)
EP (4) EP1921064B1 (de)
JP (1) JP3940359B2 (de)
KR (1) KR100847414B1 (de)
CN (1) CN1231468C (de)
AR (1) AR034268A1 (de)
AT (3) ATE278669T1 (de)
AU (4) AU9572301A (de)
BR (1) BR0114637A (de)
CA (1) CA2425876C (de)
CY (1) CY1107634T1 (de)
CZ (1) CZ299824B6 (de)
DE (3) DE60127002T2 (de)
DK (2) DK1524266T3 (de)
ES (3) ES2282794T3 (de)
GB (1) GB0025354D0 (de)
HK (2) HK1058788A1 (de)
HU (1) HU228146B1 (de)
IL (3) IL155165A0 (de)
MX (1) MXPA03003536A (de)
MY (1) MY124957A (de)
NO (1) NO324468B1 (de)
NZ (1) NZ525091A (de)
PL (1) PL203071B1 (de)
PT (2) PT1326832E (de)
SI (2) SI1326832T1 (de)
TW (1) TWI299730B (de)
WO (1) WO2002032867A1 (de)
ZA (1) ZA200302801B (de)

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Also Published As

Publication number Publication date
US7294630B2 (en) 2007-11-13
US20050137208A1 (en) 2005-06-23
CY1107634T1 (el) 2013-04-18
ATE468324T1 (de) 2010-06-15
CN1231468C (zh) 2005-12-14
SI1326832T1 (en) 2005-02-28
MXPA03003536A (es) 2003-08-07
CZ299824B6 (cs) 2008-12-03
AR034268A1 (es) 2004-02-18
HUP0301459A3 (en) 2007-11-28
WO2002032867A1 (en) 2002-04-25
PL203071B1 (pl) 2009-08-31
EP1524266B1 (de) 2007-02-28
DE60127002T2 (de) 2007-10-31
US20100081667A1 (en) 2010-04-01
DE60127002D1 (de) 2007-04-12
IL155165A0 (en) 2003-10-31
DE60106287T2 (de) 2006-02-23
NO20031561D0 (no) 2003-04-07
AU9572301A (en) 2002-04-29
NO324468B1 (no) 2007-10-22
ES2282794T3 (es) 2007-10-16
US20040014770A1 (en) 2004-01-22
US20060142302A1 (en) 2006-06-29
US7648990B2 (en) 2010-01-19
ES2227287T3 (es) 2005-04-01
AU2005204234A1 (en) 2005-09-15
DK1524266T3 (da) 2007-06-25
ES2346108T3 (es) 2010-10-08
NZ525091A (en) 2005-04-29
PT1326832E (pt) 2005-01-31
CZ20031082A3 (cs) 2004-08-18
EP1921064B1 (de) 2010-05-19
CA2425876A1 (en) 2002-04-25
CN1483025A (zh) 2004-03-17
GB0025354D0 (en) 2000-11-29
KR20030036932A (ko) 2003-05-09
AU2005204234B2 (en) 2009-05-07
NO20031561L (no) 2003-06-14
HK1058788A1 (en) 2004-06-04
EP1921064A1 (de) 2008-05-14
ZA200302801B (en) 2004-04-21
DE60106287D1 (de) 2004-11-11
HK1075889A1 (en) 2005-12-30
AU2009201407B2 (en) 2011-12-15
US7119092B2 (en) 2006-10-10
US7060702B2 (en) 2006-06-13
EP1326832A1 (de) 2003-07-16
EP1524266A1 (de) 2005-04-20
DK1326832T3 (da) 2005-01-31
TWI299730B (en) 2008-08-11
PL361180A1 (en) 2004-09-20
KR100847414B1 (ko) 2008-07-18
IL191486A0 (en) 2008-11-03
DE60142197D1 (de) 2010-07-01
JP3940359B2 (ja) 2007-07-04
AU2001295723B2 (en) 2005-05-26
CA2425876C (en) 2009-07-07
AU2009201407A1 (en) 2009-05-07
BR0114637A (pt) 2003-09-30
EP1326832B1 (de) 2004-10-06
ATE355271T1 (de) 2006-03-15
HU228146B1 (en) 2012-12-28
JP2004511544A (ja) 2004-04-15
SI1524266T1 (sl) 2007-08-31
PT1524266E (pt) 2007-05-31
HUP0301459A2 (en) 2006-09-28
US20080021041A1 (en) 2008-01-24
IL155165A (en) 2008-11-26
EP1752449A1 (de) 2007-02-14
MY124957A (en) 2006-07-31

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