DE60018040D1 - Polymorphische kristalline formen von celekoxib - Google Patents
Polymorphische kristalline formen von celekoxibInfo
- Publication number
- DE60018040D1 DE60018040D1 DE60018040T DE60018040T DE60018040D1 DE 60018040 D1 DE60018040 D1 DE 60018040D1 DE 60018040 T DE60018040 T DE 60018040T DE 60018040 T DE60018040 T DE 60018040T DE 60018040 D1 DE60018040 D1 DE 60018040D1
- Authority
- DE
- Germany
- Prior art keywords
- crystalline forms
- celecoxib
- cyclooxygenase
- celekoxib
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
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US16985699P | 1999-12-08 | 1999-12-08 | |
US169856P | 1999-12-08 | ||
PCT/US2000/032760 WO2001042222A1 (en) | 1999-12-08 | 2000-12-01 | Polymorphic crystalline forms of celecoxib |
Publications (2)
Publication Number | Publication Date |
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DE60018040D1 true DE60018040D1 (de) | 2005-03-17 |
DE60018040T2 DE60018040T2 (de) | 2006-04-13 |
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DE60018040T Expired - Fee Related DE60018040T2 (de) | 1999-12-08 | 2000-12-01 | Polymorphische kristalline formen von celecoxib |
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US (1) | US7476744B2 (de) |
EP (2) | EP1150960B1 (de) |
JP (1) | JP2003516394A (de) |
AT (1) | ATE288897T1 (de) |
AU (1) | AU750978B2 (de) |
BR (1) | BR0008088A (de) |
CA (1) | CA2362675A1 (de) |
CY (1) | CY1106307T1 (de) |
CZ (1) | CZ20013210A3 (de) |
DE (1) | DE60018040T2 (de) |
DK (1) | DK1150960T3 (de) |
DZ (1) | DZ3140A1 (de) |
EA (1) | EA003464B1 (de) |
EE (1) | EE200100419A (de) |
GE (1) | GEP20043180B (de) |
HK (1) | HK1055297A1 (de) |
HR (1) | HRP20010589A2 (de) |
IL (1) | IL144799A (de) |
IS (1) | IS6042A (de) |
MX (1) | MXPA01008161A (de) |
NO (1) | NO321062B1 (de) |
NZ (1) | NZ514059A (de) |
PL (1) | PL349224A1 (de) |
SI (1) | SI1150960T1 (de) |
SK (1) | SK11522001A3 (de) |
UA (1) | UA74539C2 (de) |
WO (1) | WO2001042222A1 (de) |
ZA (1) | ZA200207445B (de) |
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CA2514733A1 (en) * | 2003-02-28 | 2004-09-16 | Transform Pharmaceuticals, Inc. | Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen |
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EP1833476A1 (de) | 2004-11-23 | 2007-09-19 | PLIVA HRVATSKA d.o.o. | Pharmazeutische zusammensetzung von celecoxib mit verlängerter freisetzung |
WO2006079923A2 (en) * | 2005-01-31 | 2006-08-03 | Pharmacia & Upjohn Company Llc | Form iv crystalline celecoxib |
CN105641686A (zh) * | 2005-09-19 | 2016-06-08 | 爱密斯菲尔科技公司 | N-(5-氯水杨酰基)-8-氨基辛酸的二钠盐的晶形 |
SI2404919T1 (sl) | 2005-11-08 | 2013-12-31 | Vertex Pharmaceuticals Incorporated | Heterocikliäśna spojina uporabna kot modulator za prenaĺ alce z atp-vezavno kaseto |
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KR20150063170A (ko) | 2007-12-07 | 2015-06-08 | 버텍스 파마슈티칼스 인코포레이티드 | 3-(6-(1-(2,2-디플루오로벤조[d][1,3]디옥솔-5-일)사이클로프로판카복스아미도)-3-메틸피리딘-2-일)벤조산의 고체 형태 |
DK2639222T3 (en) | 2007-12-07 | 2016-10-03 | Vertex Pharma | Methods for preparing cycloalkylcarboxamido-pyridinbenzoesyrer |
NZ602030A (en) | 2008-02-28 | 2014-02-28 | Vertex Pharma | Heteroaryl derivatives as cftr modulators |
WO2010003811A1 (en) * | 2008-07-11 | 2010-01-14 | Basf Se | Amphiphilic proteins as morphology modifiers |
AR073709A1 (es) * | 2008-09-29 | 2010-11-24 | Vertex Pharma | Unidades de dosis de acido 3-(6-(1-(2,2-difluorobenzeno (d) (1,3) dioxol-5-il) ciclopropancarboxamido)-3-metilpiridin-2-il) benzoico |
WO2011055233A2 (en) | 2009-11-03 | 2011-05-12 | Actavis Group Ptc Ehf | Improved process for preparing celecoxib polymorph |
US20110213159A1 (en) | 2010-03-01 | 2011-09-01 | Vamsee Krishna Muppidi | Process for preparation of celecoxib crystalline form |
HUE056525T2 (hu) | 2010-04-07 | 2022-02-28 | Vertex Pharma | 3-(6-(1-(2,2-Difluorbenzo[d][1,3]dioxol-5-il)ciklopropánkarboxamido)-3-metilpiridin-2-il)benzoesav gyógyszerészeti készítményei és azok adagolása |
EP2468258A1 (de) * | 2010-12-22 | 2012-06-27 | LEK Pharmaceuticals d.d. | Verfahren zur Herstellung einer pharmazeutischen Zusammensetzung, die einen wenig löslichen, pharmazeutisch wirksamen Bestandteil umfasst |
CN103130684A (zh) * | 2013-03-22 | 2013-06-05 | 南开大学 | 美索巴莫磷酸二钾盐的多晶型及其制备方法 |
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ES2865600T3 (es) | 2013-11-12 | 2021-10-15 | Vertex Pharma | Proceso de preparación de composiciones farmacéuticas para el tratamiento de enfermedades mediadas por CFTR |
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JP6494757B2 (ja) | 2014-11-18 | 2019-04-03 | バーテックス ファーマシューティカルズ インコーポレイテッドVertex Pharmaceuticals Incorporated | ハイスループット試験高速液体クロマトグラフィーを行うプロセス |
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- 2000-12-01 EA EA200100874A patent/EA003464B1/ru not_active IP Right Cessation
- 2000-12-01 EP EP00983865A patent/EP1150960B1/de not_active Expired - Lifetime
- 2000-12-01 US US09/728,040 patent/US7476744B2/en not_active Expired - Fee Related
- 2000-12-01 DZ DZ003140A patent/DZ3140A1/xx active
- 2000-12-01 PL PL00349224A patent/PL349224A1/xx not_active Application Discontinuation
- 2000-12-01 WO PCT/US2000/032760 patent/WO2001042222A1/en active IP Right Grant
- 2000-12-01 SK SK1152-2001A patent/SK11522001A3/sk unknown
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- 2000-12-01 NZ NZ514059A patent/NZ514059A/xx unknown
- 2000-12-01 CA CA002362675A patent/CA2362675A1/en not_active Abandoned
- 2000-12-01 SI SI200030663T patent/SI1150960T1/xx unknown
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- 2000-12-01 EP EP05002575A patent/EP1528058A1/de not_active Withdrawn
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- 2000-12-01 DE DE60018040T patent/DE60018040T2/de not_active Expired - Fee Related
- 2000-12-01 AT AT00983865T patent/ATE288897T1/de not_active IP Right Cessation
- 2000-12-06 CZ CZ20013210A patent/CZ20013210A3/cs unknown
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2001
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- 2001-08-09 HR HR20010589A patent/HRP20010589A2/hr not_active Application Discontinuation
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