DE3208506A1 - Verfahren zur herstellung von 6-(d(-)-(alpha)-(4-c(pfeil abwaerts)1(pfeil abwaerts)(pfeil abwaerts)-(pfeil abwaerts)(pfeil abwaerts)4(pfeil abwaerts))-alkyl-2,3-dioxo-1- piperazinocarbonylamino)-phenylacetamido)- penicillansaeuren - Google Patents

Verfahren zur herstellung von 6-(d(-)-(alpha)-(4-c(pfeil abwaerts)1(pfeil abwaerts)(pfeil abwaerts)-(pfeil abwaerts)(pfeil abwaerts)4(pfeil abwaerts))-alkyl-2,3-dioxo-1- piperazinocarbonylamino)-phenylacetamido)- penicillansaeuren

Info

Publication number
DE3208506A1
DE3208506A1 DE19823208506 DE3208506A DE3208506A1 DE 3208506 A1 DE3208506 A1 DE 3208506A1 DE 19823208506 DE19823208506 DE 19823208506 DE 3208506 A DE3208506 A DE 3208506A DE 3208506 A1 DE3208506 A1 DE 3208506A1
Authority
DE
Germany
Prior art keywords
weight
parts
mixture
ampicillin
dioxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
DE19823208506
Other languages
German (de)
English (en)
Other versions
DE3208506C2 (xx
Inventor
Karel F. Belle Mead N.J. Bernady
Donald C. Bloomsbury N.J. Boop
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth Holdings LLC
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of DE3208506A1 publication Critical patent/DE3208506A1/de
Application granted granted Critical
Publication of DE3208506C2 publication Critical patent/DE3208506C2/de
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
DE19823208506 1981-03-30 1982-03-09 Verfahren zur herstellung von 6-(d(-)-(alpha)-(4-c(pfeil abwaerts)1(pfeil abwaerts)(pfeil abwaerts)-(pfeil abwaerts)(pfeil abwaerts)4(pfeil abwaerts))-alkyl-2,3-dioxo-1- piperazinocarbonylamino)-phenylacetamido)- penicillansaeuren Granted DE3208506A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24875481A 1981-03-30 1981-03-30

Publications (2)

Publication Number Publication Date
DE3208506A1 true DE3208506A1 (de) 1982-10-07
DE3208506C2 DE3208506C2 (xx) 1991-05-02

Family

ID=22940531

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19823208506 Granted DE3208506A1 (de) 1981-03-30 1982-03-09 Verfahren zur herstellung von 6-(d(-)-(alpha)-(4-c(pfeil abwaerts)1(pfeil abwaerts)(pfeil abwaerts)-(pfeil abwaerts)(pfeil abwaerts)4(pfeil abwaerts))-alkyl-2,3-dioxo-1- piperazinocarbonylamino)-phenylacetamido)- penicillansaeuren

Country Status (23)

Country Link
JP (1) JPS57165391A (xx)
AT (1) AT381706B (xx)
AU (1) AU544896B2 (xx)
BE (1) BE892586A (xx)
CA (1) CA1200239A (xx)
CH (1) CH654309A5 (xx)
DE (1) DE3208506A1 (xx)
DK (1) DK161079C (xx)
ES (1) ES8306376A1 (xx)
FR (1) FR2502623A1 (xx)
GB (1) GB2095661B (xx)
GR (1) GR76054B (xx)
HK (1) HK23590A (xx)
IE (1) IE52907B1 (xx)
IL (1) IL64981A (xx)
IT (1) IT1148130B (xx)
LU (1) LU84036A1 (xx)
NL (2) NL192453A (xx)
NZ (1) NZ199869A (xx)
PH (1) PH19765A (xx)
PL (1) PL235508A1 (xx)
SE (1) SE452767B (xx)
ZA (1) ZA82674B (xx)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3627581A1 (de) * 1985-08-16 1987-02-19 Dso Pharmachim Verfahren zur herstellung von 6-/d/-/-(alpha)-/4-ethyl-2,3-dioxo-1-piperazinocarbonylamino-(phenylacetamido)-penizillansaeure

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4112090A (en) * 1974-05-09 1978-09-05 Toyama Chemical Co., Ltd. Novel penicillins and cephalosporins and process for producing the same

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4087424A (en) * 1974-05-09 1978-05-02 Toyama Chemical Co., Ltd. Novel penicillins and cephalosporins and process for producing the same
IL47168A (en) * 1974-05-09 1979-07-25 Toyama Chemical Co Ltd Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4112090A (en) * 1974-05-09 1978-09-05 Toyama Chemical Co., Ltd. Novel penicillins and cephalosporins and process for producing the same

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Chem. Abstr. 88, 1978, 105210p *
Yakugaku Zasshi 97, 1977, 980-986 *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3627581A1 (de) * 1985-08-16 1987-02-19 Dso Pharmachim Verfahren zur herstellung von 6-/d/-/-(alpha)-/4-ethyl-2,3-dioxo-1-piperazinocarbonylamino-(phenylacetamido)-penizillansaeure

Also Published As

Publication number Publication date
BE892586A (fr) 1982-09-22
AU7996482A (en) 1982-10-07
JPS57165391A (en) 1982-10-12
DE3208506C2 (xx) 1991-05-02
FR2502623A1 (fr) 1982-10-01
GR76054B (xx) 1984-08-03
IE52907B1 (en) 1988-04-13
GB2095661A (en) 1982-10-06
NL8201301A (nl) 1982-10-18
SE452767B (sv) 1987-12-14
NL192453B (nl) 1997-04-01
CH654309A5 (de) 1986-02-14
DK48282A (da) 1982-10-01
DK161079B (da) 1991-05-27
AT381706B (de) 1986-11-25
NL192453A (xx) 1997-10-01
FR2502623B1 (xx) 1984-12-28
IT1148130B (it) 1986-11-26
AU544896B2 (en) 1985-06-20
GB2095661B (en) 1985-02-27
SE8201998L (sv) 1982-10-01
ES509424A0 (es) 1983-06-01
IT8247962A0 (it) 1982-03-10
IE820746L (en) 1982-09-30
LU84036A1 (de) 1982-07-08
NL192453C (nl) 1997-08-04
NZ199869A (en) 1985-07-31
ZA82674B (en) 1982-12-29
DK161079C (da) 1991-11-04
ES8306376A1 (es) 1983-06-01
PL235508A1 (xx) 1982-12-20
HK23590A (en) 1990-04-06
ATA93082A (de) 1986-04-15
JPH0331716B2 (xx) 1991-05-08
IL64981A (en) 1985-11-29
PH19765A (en) 1986-06-27
CA1200239A (en) 1986-02-04

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Legal Events

Date Code Title Description
8110 Request for examination paragraph 44
D2 Grant after examination
8364 No opposition during term of opposition
V448 Application of spc

Free format text: PRODUCT NAME: PIPERACILLIN/FLUCLOXACILLIN; REGISTRATION NO/DATE: 6402.00.00, 6402.01.00, 6402.02.00, 6402.03.00; 19890705

Spc suppl protection certif: 193 75 107

Filing date: 19930702

V472 Application for supplementary protection certificate rejected

Free format text: PRODUCT NAME: PIPERACILLIN/FLUCLOXACILLIN; REGISTRATION NO/DATE: 6402.00.00, 6402.01.00, 6402.02.00, 6402.03.00; 19890705

Spc suppl protection certif: 193 75 107

Filing date: 19930702