DE2501238C2 - N-(Benzolsulfonyl)-5-0-Desosaminyl-Erythromycylaminderivate und Verfahren zu deren Herstellung - Google Patents

N-(Benzolsulfonyl)-5-0-Desosaminyl-Erythromycylaminderivate und Verfahren zu deren Herstellung

Info

Publication number
DE2501238C2
DE2501238C2 DE2501238A DE2501238A DE2501238C2 DE 2501238 C2 DE2501238 C2 DE 2501238C2 DE 2501238 A DE2501238 A DE 2501238A DE 2501238 A DE2501238 A DE 2501238A DE 2501238 C2 DE2501238 C2 DE 2501238C2
Authority
DE
Germany
Prior art keywords
solution
chloroform
desosaminyl
benzenesulfonyl
erythromycylamine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE2501238A
Other languages
German (de)
English (en)
Other versions
DE2501238A1 (de
Inventor
Slobodan Dr.-Ing. Zagreb Djokic
Gorjana Dipl.-Ing. Radobolja
Zrinka Dr.-Ing. Tamburasev
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pliva Farmaceutika dd
Original Assignee
Pliva Farmaceutska Kemijska Prehrambena I Kozmeticka Industrija dd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva Farmaceutska Kemijska Prehrambena I Kozmeticka Industrija dd filed Critical Pliva Farmaceutska Kemijska Prehrambena I Kozmeticka Industrija dd
Publication of DE2501238A1 publication Critical patent/DE2501238A1/de
Application granted granted Critical
Publication of DE2501238C2 publication Critical patent/DE2501238C2/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE2501238A 1974-01-14 1975-01-14 N-(Benzolsulfonyl)-5-0-Desosaminyl-Erythromycylaminderivate und Verfahren zu deren Herstellung Expired DE2501238C2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
YU97/74A YU35363B (en) 1974-01-14 1974-01-14 Process for obtaining n-(benzene-sulfonyl)-5-0desosaminyl-erythromycilamine derivatives

Publications (2)

Publication Number Publication Date
DE2501238A1 DE2501238A1 (de) 1975-07-17
DE2501238C2 true DE2501238C2 (de) 1982-02-25

Family

ID=25548317

Family Applications (1)

Application Number Title Priority Date Filing Date
DE2501238A Expired DE2501238C2 (de) 1974-01-14 1975-01-14 N-(Benzolsulfonyl)-5-0-Desosaminyl-Erythromycylaminderivate und Verfahren zu deren Herstellung

Country Status (7)

Country Link
US (1) US3939144A (OSRAM)
AT (1) AT333959B (OSRAM)
CA (1) CA1039276A (OSRAM)
DE (1) DE2501238C2 (OSRAM)
FR (1) FR2257302B1 (OSRAM)
GB (1) GB1461032A (OSRAM)
YU (1) YU35363B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK139522C (da) * 1975-04-07 1979-08-20 Thomae Gmbh Dr K Analogifremgangsmaade til fremstilling af 9-iminoalkylamino-erythromyciner eller syreadditionssalte deraf
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4321362A (en) * 1980-06-12 1982-03-23 Eli Lilly And Company De(mycinosyloxy)tylosin and process for its production
US4334019A (en) * 1980-06-12 1982-06-08 Eli Lilly And Company Process for producing de(mycinosyloxy)tylosin
US5075289A (en) * 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
FR2680790B1 (fr) * 1991-08-29 1996-10-31 Roussel Uclaf Nouveaux derives descladinosyles de l'erythromycine, leur procede de preparation et leur application comme medicaments.
FR2677025B1 (fr) * 1991-05-27 1995-04-07 Roussel Uclaf Nouveaux derives descladinosyles de l'erythromycine, leur procede de preparation et leur application comme medicaments.
US20020132782A1 (en) * 2001-01-18 2002-09-19 Zhenkun Ma 9-amino erythromycin derivatives with antibacterial activity
US7582611B2 (en) 2005-05-24 2009-09-01 Pfizer Inc. Motilide compounds
US20070135362A1 (en) * 2005-12-08 2007-06-14 Yaoquan Liu Method for demethylating the 3'-dimethylamino group of erythromycin compounds
AU2007330456B2 (en) * 2006-12-05 2011-03-03 Pfizer Inc. Motilide polymorphs

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1100267A (en) * 1966-10-14 1968-01-24 Pliva Pharm & Chem Works 9-amino-5-o-desosaminyl-3,6,11,12-tetrahydroxy-2,4,6,8,10,12-hexamethylpentadecane-13-olide and 9-amino-3,5,6,11,12-pentahydroxy-2,4,6,8,10,12-hexamethylpentadecane-13-olide

Also Published As

Publication number Publication date
AT333959B (de) 1976-12-27
FR2257302B1 (OSRAM) 1978-07-21
DE2501238A1 (de) 1975-07-17
YU9774A (en) 1980-06-30
GB1461032A (en) 1977-01-13
US3939144A (en) 1976-02-17
ATA21975A (de) 1976-04-15
FR2257302A1 (OSRAM) 1975-08-08
CA1039276A (en) 1978-09-26
YU35363B (en) 1980-12-31

Similar Documents

Publication Publication Date Title
DE2501238C2 (de) N-(Benzolsulfonyl)-5-0-Desosaminyl-Erythromycylaminderivate und Verfahren zu deren Herstellung
DE3140449C2 (de) N-Methyl-11-aza-10-deoxo-10-dihydro-erythromycine A, Verfahren zu ihrer Herstellung sowie ihre Verwendung
DE1643738B1 (de) 7-[3alpha,5alpha-Dihydroxy-2-(3-hydroxyoctenyl-(1))-cyclopentyl]-heptan-1-ol,dessen Tetraacetat und Verfahren zu deren Herstellung
CH646440A5 (de) 11-aza-4-0-cladinosyl-6-0-desosaminyl-15-aethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyloxacyclopentadecan-2-on und dessen derivate sowie ein verfahren zu deren herstellung.
DE2427096A1 (de) 2-deoxystreptamin-aminoglycoside und verfahren zu ihrer herstellung
DE2515629A1 (de) Paromomycin-derivate, verfahren zu ihrer herstellung und arzneimittel
DE2641388C3 (de) 3',4'-Didesoxykanamycin B-N-methansulfonsäuren und deren Alkalimetallsalze sowie diese Verbindungen enthaltende pharmazeutische Präparate
DE2509260B2 (de) a-(23,4,5,6-Penta-O-acetyI- D-gluconyl-thioureido)benzylpenicillin
DE2929058A1 (de) Anorganische salze von trimethylammoniumderivaten der polyenmakrolide, insbesondere anorganische salze von methylestern dieser derivate, und verfahren zu deren herstellung
DE2735455B2 (de) Daunomycinanaloga, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
DE2027699B2 (de) Verfahren zur Herstellung von N-Desalkyl-lincomycin und dessen Analogen
DE3227178C2 (de) 2'-Modifizierte Kanamycine, Verfahren zu deren Herstellung und diese Verbindungen enthaltende antibakterielle Mittel
DE2421488A1 (de) Sulfonylderivate des erythromycins
DE2402200C2 (de) N-(Benzolsulfonyl)-erythromycylaminderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
AT397504B (de) Diosminderivat und verfahren zu dessen herstellung
DE284231C (OSRAM)
DE2900119A1 (de) 4''-desoxy-4''-carbamat- und -dithiocarbamat-derivate des oleandomycins und seine ester, verfahren zu deren herstellung und solche derivate enthaltende arzneimittel
DE1643797A1 (de) Neue Thionocarbamidsaeureester und Verfahren zu ihrer Herstellung
AT241481B (de) Verfahren zur Herstellung von neuen, beispielsweise zur Schädlingsbekämpfung verwendbaren Organophosphorverbindungen
DE2114295A1 (de) Substituierte AEtherderivate des N-Hydroxymethyl-2-pyrrolidinon und Verfahren zu deren Herstellung
DE839940C (de) Verfahren zur Herstellung von organischen Salzen von ª†-Methylmercapto-ª‡-acylaminobuttersaeuren
DE2547738A1 (de) 2-deoxystreptamin-aminoglykoside, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
AT371480B (de) Verfahren zur herstellung von neuen kanamycin a derivaten
AT110280B (de) Verfahren zur Gewinnung von wasserlöslichen Anthrachinonglykosiden aus Drogen.
DE2313845C3 (de) Thiocarbaminsäurederivate und diese enthaltende Arzneimittelzubereitungen

Legal Events

Date Code Title Description
OD Request for examination
D2 Grant after examination
8328 Change in the person/name/address of the agent

Free format text: VON FUENER, A., DIPL.-CHEM. DR.RER.NAT. EBBINGHAUS, D., DIPL.-ING., PAT.-ANW., 8000 MUENCHEN

8339 Ceased/non-payment of the annual fee