DE1935027A1 - Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen - Google Patents

Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen

Info

Publication number
DE1935027A1
DE1935027A1 DE19691935027 DE1935027A DE1935027A1 DE 1935027 A1 DE1935027 A1 DE 1935027A1 DE 19691935027 DE19691935027 DE 19691935027 DE 1935027 A DE1935027 A DE 1935027A DE 1935027 A1 DE1935027 A1 DE 1935027A1
Authority
DE
Germany
Prior art keywords
carbon atoms
general formula
advantageously
methanol
glycosyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19691935027
Other languages
German (de)
English (en)
Inventor
Piskala Dr Alois
Frantisek Sorm
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Czech Academy of Sciences
Original Assignee
Czech Academy of Sciences
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Czech Academy of Sciences filed Critical Czech Academy of Sciences
Publication of DE1935027A1 publication Critical patent/DE1935027A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12—Triazine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Gripping On Spindles (AREA)
DE19691935027 1968-11-12 1969-07-10 Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen Pending DE1935027A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS770868 1968-11-12

Publications (1)

Publication Number Publication Date
DE1935027A1 true DE1935027A1 (de) 1970-06-04

Family

ID=5426669

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19691935027 Pending DE1935027A1 (de) 1968-11-12 1969-07-10 Verfahren zur Herstellung von 1-Glykosyl-5-azacytosinen

Country Status (12)

Country Link
AT (1) AT292205B (cg-RX-API-DMAC7.html)
BE (1) BE732796A (cg-RX-API-DMAC7.html)
CH (1) CH507969A (cg-RX-API-DMAC7.html)
DE (1) DE1935027A1 (cg-RX-API-DMAC7.html)
DK (1) DK128008B (cg-RX-API-DMAC7.html)
ES (1) ES367451A1 (cg-RX-API-DMAC7.html)
FR (1) FR2023018A1 (cg-RX-API-DMAC7.html)
GB (1) GB1227692A (cg-RX-API-DMAC7.html)
IT (1) IT1033029B (cg-RX-API-DMAC7.html)
NL (1) NL6907961A (cg-RX-API-DMAC7.html)
NO (1) NO126626B (cg-RX-API-DMAC7.html)
SE (1) SE350048B (cg-RX-API-DMAC7.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2012888C3 (de) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden
US6943249B2 (en) 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US6887855B2 (en) 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US7038038B2 (en) 2003-03-17 2006-05-02 Pharmion Corporation Synthesis of 5-azacytidine
DK3782612T3 (da) 2008-05-15 2024-01-15 Celgene Corp Orale formuleringer af cytidinanaloger og fremgangsmåder til anvendelse deraf
WO2012135405A1 (en) 2011-03-31 2012-10-04 Pharmion Llc Systhesis of 5-azacytidine

Also Published As

Publication number Publication date
BE732796A (cg-RX-API-DMAC7.html) 1969-10-16
GB1227692A (cg-RX-API-DMAC7.html) 1971-04-07
FR2023018A1 (cg-RX-API-DMAC7.html) 1970-08-07
AT292205B (de) 1971-08-25
NO126626B (cg-RX-API-DMAC7.html) 1973-03-05
NL6907961A (cg-RX-API-DMAC7.html) 1970-05-14
CH507969A (de) 1971-05-31
IT1033029B (it) 1979-07-10
DK128008B (da) 1974-02-18
SE350048B (cg-RX-API-DMAC7.html) 1972-10-16
ES367451A1 (es) 1971-04-01

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