DE102004029784A1 - Neue 2-Benzylaminodihydropteridinone, Verfahren zur deren Herstellung und deren Verwendung als Arzneimittel - Google Patents
Neue 2-Benzylaminodihydropteridinone, Verfahren zur deren Herstellung und deren Verwendung als Arzneimittel Download PDFInfo
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- DE102004029784A1 DE102004029784A1 DE102004029784A DE102004029784A DE102004029784A1 DE 102004029784 A1 DE102004029784 A1 DE 102004029784A1 DE 102004029784 A DE102004029784 A DE 102004029784A DE 102004029784 A DE102004029784 A DE 102004029784A DE 102004029784 A1 DE102004029784 A1 DE 102004029784A1
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- alkyl
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- hydrogen
- optionally substituted
- aryl
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Priority Applications (10)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004029784A DE102004029784A1 (de) | 2004-06-21 | 2004-06-21 | Neue 2-Benzylaminodihydropteridinone, Verfahren zur deren Herstellung und deren Verwendung als Arzneimittel |
| JP2007517147A JP5102021B2 (ja) | 2004-06-21 | 2005-06-15 | 新規２−ベンジルアミノジヒドロプテリジノン、それらを製造する方法及び薬剤としてのそれらの使用 |
| ES05751714T ES2297724T3 (es) | 2004-06-21 | 2005-06-15 | Nuevas 2-bencilaminodihidropteridinonas, procedimiento para su obtencion y su empleo como medicamentos. |
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| EP05751714A EP1761536B1 (de) | 2004-06-21 | 2005-06-15 | Neue 2-benzylaminodihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel |
| AT05751714T ATE382049T1 (de) | 2004-06-21 | 2005-06-15 | Neue 2-benzylaminodihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel |
| CA2571293A CA2571293C (en) | 2004-06-21 | 2005-06-15 | 2-benzylaminodihydropteridinones, method for producing them and use thereof as drugs |
| PCT/EP2005/006404 WO2005123736A1 (de) | 2004-06-21 | 2005-06-15 | Neue 2-benzylaminodihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel |
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| US12/357,731 US7759347B2 (en) | 2004-06-21 | 2009-01-22 | 2-benzylaminodihydropteridinones, process for their manufacture and use thereof as medicaments |
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| US7759485B2 (en) | 2004-08-14 | 2010-07-20 | Boehringer Ingelheim International Gmbh | Process for the manufacture of dihydropteridinones |
| US20060074088A1 (en) | 2004-08-14 | 2006-04-06 | Boehringer Ingelheim International Gmbh | Dihydropteridinones for the treatment of cancer diseases |
| EP1632493A1 (de) | 2004-08-25 | 2006-03-08 | Boehringer Ingelheim Pharma GmbH & Co.KG | Dihydropteridinonderivative, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| EP1630163A1 (de) | 2004-08-25 | 2006-03-01 | Boehringer Ingelheim Pharma GmbH & Co.KG | Dihydropteridinonderivative, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
| CA2575804A1 (en) | 2004-08-26 | 2006-03-02 | Boehringer Ingelheim International Gmbh | Pteridinones used as plk (polo like kinase) inhibitors |
| JP2008510771A (ja) | 2004-08-27 | 2008-04-10 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ジヒドロプテリジノン、その製造方法および医薬薬剤としてのその使用 |
| DE102004058337A1 (de) | 2004-12-02 | 2006-06-14 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Verfahren zur Herstellung von annelierten Piperazin-2-on Derivaten |
| WO2007014838A1 (en) | 2005-08-03 | 2007-02-08 | Boehringer Ingelheim International Gmbh | Dihydropteridinones in the treatment of respiratory diseases |
| US7439358B2 (en) | 2006-02-08 | 2008-10-21 | Boehringer Ingelheim International Gmbh | Specific salt, anhydrous and crystalline form of a dihydropteridione derivative |
| EP2185559A1 (en) | 2007-08-03 | 2010-05-19 | Boehringer Ingelheim International GmbH | Crystalline form of a dihydropteridione derivative |
-
2004
- 2004-06-21 DE DE102004029784A patent/DE102004029784A1/de not_active Withdrawn
-
2005
- 2005-06-15 DE DE502005002356T patent/DE502005002356D1/de not_active Expired - Lifetime
- 2005-06-15 WO PCT/EP2005/006404 patent/WO2005123736A1/de not_active Ceased
- 2005-06-15 AT AT05751714T patent/ATE382049T1/de active
- 2005-06-15 ES ES05751714T patent/ES2297724T3/es not_active Expired - Lifetime
- 2005-06-15 EP EP05751714A patent/EP1761536B1/de not_active Expired - Lifetime
- 2005-06-15 JP JP2007517147A patent/JP5102021B2/ja not_active Expired - Lifetime
- 2005-06-15 CA CA2571293A patent/CA2571293C/en not_active Expired - Lifetime
- 2005-06-21 US US11/157,883 patent/US20060004014A1/en not_active Abandoned
-
2009
- 2009-01-22 US US12/357,731 patent/US7759347B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| CA2571293C (en) | 2013-05-28 |
| ATE382049T1 (de) | 2008-01-15 |
| EP1761536A1 (de) | 2007-03-14 |
| EP1761536B1 (de) | 2007-12-26 |
| JP5102021B2 (ja) | 2012-12-19 |
| DE502005002356D1 (de) | 2008-02-07 |
| US20060004014A1 (en) | 2006-01-05 |
| JP2008503515A (ja) | 2008-02-07 |
| ES2297724T3 (es) | 2008-05-01 |
| WO2005123736A1 (de) | 2005-12-29 |
| WO2005123736A8 (de) | 2006-03-30 |
| US7759347B2 (en) | 2010-07-20 |
| US20090124628A1 (en) | 2009-05-14 |
| CA2571293A1 (en) | 2005-12-29 |
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| 8139 | Disposal/non-payment of the annual fee |