CZ8799A3 - Bicyklické heteroaromatické sloučeniny, způsob jejich výroby a farmaceutický prostředek - Google Patents

Bicyklické heteroaromatické sloučeniny, způsob jejich výroby a farmaceutický prostředek Download PDF

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Publication number
CZ8799A3
CZ8799A3 CZ9987A CZ8799A CZ8799A3 CZ 8799 A3 CZ8799 A3 CZ 8799A3 CZ 9987 A CZ9987 A CZ 9987A CZ 8799 A CZ8799 A CZ 8799A CZ 8799 A3 CZ8799 A3 CZ 8799A3
Authority
CZ
Czechia
Prior art keywords
alkyl
group
compound
furan
pyrido
Prior art date
Application number
CZ9987A
Other languages
Czech (cs)
English (en)
Inventor
George Stuart Cockerill
Malcolm Clive Carter
Stephen Barry Guntrip
Kathryn Jane Smith
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9614756.6A external-priority patent/GB9614756D0/en
Priority claimed from GBGB9625495.8A external-priority patent/GB9625495D0/en
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of CZ8799A3 publication Critical patent/CZ8799A3/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/16—Emollients or protectives, e.g. against radiation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/78—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C07C217/80—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings
    • C07C217/82—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring
    • C07C217/84—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
    • C07C217/86—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings of the same non-condensed six-membered aromatic ring the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/26—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
    • C07C317/36—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring with the nitrogen atoms of the amino groups bound to hydrogen atoms or to carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Toxicology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CZ9987A 1996-07-13 1997-07-11 Bicyklické heteroaromatické sloučeniny, způsob jejich výroby a farmaceutický prostředek CZ8799A3 (cs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9614756.6A GB9614756D0 (en) 1996-07-13 1996-07-13 Heterocyclic compounds
GBGB9625495.8A GB9625495D0 (en) 1996-12-07 1996-12-07 Heterocyclic compounds

Publications (1)

Publication Number Publication Date
CZ8799A3 true CZ8799A3 (cs) 1999-06-16

Family

ID=26309691

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ9987A CZ8799A3 (cs) 1996-07-13 1997-07-11 Bicyklické heteroaromatické sloučeniny, způsob jejich výroby a farmaceutický prostředek

Country Status (22)

Country Link
US (1) US6207669B1 (enExample)
EP (1) EP0912572B1 (enExample)
JP (1) JP2000515136A (enExample)
KR (1) KR20000023813A (enExample)
CN (1) CN1230185A (enExample)
AP (1) AP9901435A0 (enExample)
AR (1) AR007855A1 (enExample)
AT (1) ATE231148T1 (enExample)
AU (1) AU3693697A (enExample)
BR (1) BR9710362A (enExample)
CA (1) CA2260058A1 (enExample)
CZ (1) CZ8799A3 (enExample)
DE (1) DE69718472T2 (enExample)
EA (1) EA199900021A1 (enExample)
ES (1) ES2191187T3 (enExample)
ID (1) ID19430A (enExample)
IS (1) IS4936A (enExample)
NO (1) NO990123L (enExample)
PE (1) PE91098A1 (enExample)
PL (1) PL331154A1 (enExample)
TR (1) TR199900048T2 (enExample)
WO (1) WO1998002437A1 (enExample)

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NO990123D0 (no) 1999-01-12
CA2260058A1 (en) 1998-01-22
CN1230185A (zh) 1999-09-29
IS4936A (is) 1998-12-29
NO990123L (no) 1999-01-13
JP2000515136A (ja) 2000-11-14
EA199900021A1 (ru) 1999-08-26
AR007855A1 (es) 1999-11-24
AU3693697A (en) 1998-02-09
PL331154A1 (en) 1999-06-21
ID19430A (id) 1998-07-09
EP0912572B1 (en) 2003-01-15
EP0912572A1 (en) 1999-05-06
KR20000023813A (en) 2000-04-25
ATE231148T1 (de) 2003-02-15
TR199900048T2 (xx) 1999-04-21
PE91098A1 (es) 1999-01-15
WO1998002437A1 (en) 1998-01-22
ES2191187T3 (es) 2003-09-01
AP9901435A0 (en) 1999-03-31
US6207669B1 (en) 2001-03-27
DE69718472T2 (de) 2003-11-06
DE69718472D1 (de) 2003-02-20
BR9710362A (pt) 1999-08-17

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