CY1949A - Stable salts of 4"-deoxy-4"-epimethylamino avermectin B1a/B1b - Google Patents
Stable salts of 4"-deoxy-4"-epimethylamino avermectin B1a/B1bInfo
- Publication number
- CY1949A CY1949A CY194991A CY194991A CY1949A CY 1949 A CY1949 A CY 1949A CY 194991 A CY194991 A CY 194991A CY 194991 A CY194991 A CY 194991A CY 1949 A CY1949 A CY 1949A
- Authority
- CY
- Cyprus
- Prior art keywords
- acid salt
- deoxy
- epimethylamino
- avermectin
- sec
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Agronomy & Crop Science (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Silicon Polymers (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
- Steroid Compounds (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Fodder In General (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54522990A | 1990-06-28 | 1990-06-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1949A true CY1949A (en) | 1991-06-27 |
Family
ID=24175383
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY194991A CY1949A (en) | 1990-06-28 | 1991-06-27 | Stable salts of 4"-deoxy-4"-epimethylamino avermectin B1a/B1b |
Country Status (21)
Country | Link |
---|---|
US (1) | US5288710A (sv) |
EP (1) | EP0465121B1 (sv) |
JP (1) | JPH0822870B2 (sv) |
KR (1) | KR100224292B1 (sv) |
AT (1) | ATE134377T1 (sv) |
AU (1) | AU641777B2 (sv) |
CA (1) | CA2045864C (sv) |
CY (1) | CY1949A (sv) |
DE (1) | DE69117223T2 (sv) |
DK (1) | DK0465121T3 (sv) |
ES (1) | ES2084110T3 (sv) |
FI (1) | FI97890C (sv) |
GR (1) | GR3019067T3 (sv) |
HK (1) | HK157096A (sv) |
IE (1) | IE71175B1 (sv) |
IL (1) | IL98599A (sv) |
LV (1) | LV5740B4 (sv) |
NO (2) | NO2001007I2 (sv) |
NZ (1) | NZ238705A (sv) |
PT (1) | PT98117B (sv) |
ZA (1) | ZA914961B (sv) |
Families Citing this family (61)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2170099T3 (es) * | 1993-05-26 | 2002-08-01 | Commw Scient Ind Res Org | Composiciones antiparasitarias. |
AU687062B2 (en) * | 1993-05-26 | 1998-02-19 | Commonwealth Scientific And Industrial Research Organisation | Controlled release antiparasitic compositions |
US6486195B1 (en) * | 1993-08-19 | 2002-11-26 | Merck & Co., Inc. | Thermodynamically stable crystal form of 4″-deoxy-4″-epi-methylamino avermectin B1a/B1b benzoic acid salt and processes for its preparation |
ES2139753T3 (es) * | 1993-08-19 | 2000-02-16 | Merck & Co Inc | Forma cristalina termodinamicamente estable de la sal del acido benzoico de la 4''-desoxi-4''-epi-metilamino avermectina b1a/b1b y procedimiento para su preparacion. |
US5362863A (en) * | 1993-09-29 | 1994-11-08 | Merck & Co., Inc. | Process for the preparation of 4"-amino avermectin compounds |
EA002756B1 (ru) * | 1995-11-08 | 2002-08-29 | Мерк Энд Ко., Инк. | Пестицидная композиция в форме растворимых в воде гранул |
AU768262B2 (en) * | 1995-11-08 | 2003-12-04 | Merck Sharp & Dohme Corp. | Pesticidal formulation |
CN1915016B (zh) * | 1995-11-08 | 2010-12-22 | 默沙东公司 | 农药制剂 |
US20050192319A1 (en) * | 1996-09-19 | 2005-09-01 | Albert Boeckh | Spot-on formulations for combating parasites |
US6054140A (en) * | 1997-03-21 | 2000-04-25 | Biogenesis S.A. | Long acting injectable parasiticidal composition and the process for its preparation |
AU1665999A (en) * | 1997-11-14 | 1999-06-07 | Novartis Ag | Pesticidal composition |
JP2001527026A (ja) * | 1997-12-23 | 2001-12-25 | ノバルティス ファーマ アクチエンゲゼルシャフト | 有害生物防除におけるマクロライド類の使用 |
US6486128B1 (en) | 1999-04-08 | 2002-11-26 | Schering-Plough Veterinary Corporation | Method of using emamectin to treat fish parasites |
AR006063A4 (es) * | 1999-04-17 | 1999-08-11 | Romario S R L | Bandeja termica para pizzas |
GB9926887D0 (en) * | 1999-11-12 | 2000-01-12 | Novartis Ag | Organic compounds |
CR6574A (es) * | 2001-02-27 | 2004-10-28 | Syngenta Participations Ag | Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas |
EG23124A (en) | 2001-02-27 | 2004-04-28 | Syngenta Participations Ag | Avermectins substituted in the 4-position having pesticidal properties |
JP4701538B2 (ja) | 2001-05-21 | 2011-06-15 | 住友化学株式会社 | 農業害虫防除剤組成物 |
AR036486A1 (es) | 2001-08-28 | 2004-09-15 | Syngenta Participations Ag | Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion |
DE10203688A1 (de) * | 2002-01-31 | 2003-08-07 | Bayer Cropscience Ag | Synergistische insektizide Mischungen |
DE10207241A1 (de) * | 2002-02-21 | 2003-09-04 | Bayer Cropscience Ag | Synergistische insektizide Mischungen |
DE10207242A1 (de) * | 2002-02-21 | 2003-09-04 | Bayer Cropscience Ag | Synergistische insektizide Mischungen |
CN1642946A (zh) * | 2002-03-22 | 2005-07-20 | 株式会社Lg生命科学 | (2s)-n-{5-[氨基(亚氨基)甲基]-2-噻吩基}甲基-1-{(2r)-2-[(羧甲基)氨基]3,-二苯基丙酰}-2-吡咯烷甲酰胺的马来酸盐及其制备方法 |
AR040073A1 (es) | 2002-05-07 | 2005-03-16 | Syngenta Participations Ag | Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas |
GB0302310D0 (en) | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties |
GB0302308D0 (en) | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties |
GB0320176D0 (en) | 2003-08-28 | 2003-10-01 | Syngenta Participations Ag | Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties |
JP4644254B2 (ja) | 2004-09-23 | 2011-03-02 | シェーリング−プラウ・リミテッド | 新規トリフルオロメタンスルホンアニリドオキシムエーテル誘導体の使用による動物における寄生虫の制御 |
WO2006055565A2 (en) * | 2004-11-19 | 2006-05-26 | Schering-Plough Ltd. | Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives |
AR054380A1 (es) * | 2005-06-09 | 2007-06-20 | Schering Plough Ltd | Control de parasitos en animales con derivados de n- ((feniloxi) fenil) -1,1,1-trifluorometansulfonamida y de n-(fenilsulfanil) fenil) -1,1,1-trifluorometansulfonamida |
US8119667B2 (en) * | 2005-12-29 | 2012-02-21 | Schering-Plough Animal Health Corporation | Carbonates of fenicol antibiotics |
EP1849363A1 (en) * | 2006-03-09 | 2007-10-31 | Cheminova A/S | Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin |
US20070238700A1 (en) * | 2006-04-10 | 2007-10-11 | Winzenberg Kevin N | N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites |
TWI422328B (zh) | 2006-06-19 | 2014-01-11 | Univ California | 結合有殺線蟲之種子塗覆物的生物控制劑 |
FR2906469B1 (fr) * | 2006-09-28 | 2008-11-28 | Galderma Sa | Utilisation de composes de la famille des avermectines pour le traitement de desordres dermatologiques chez l'homme |
US8084643B2 (en) * | 2006-12-13 | 2011-12-27 | Intervet Inc. | Water-soluble prodrugs of florfenicol and its analogs |
CA2672795A1 (en) * | 2006-12-13 | 2008-06-26 | Schering-Plough Ltd. | Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof |
DE102007002872A1 (de) | 2007-01-15 | 2008-07-17 | Alpha-Biocare Gmbh | Verwendung von Avermectin-Derivaten zur Behandlung gegen Parasiten von Fischen |
TWI430995B (zh) | 2007-06-26 | 2014-03-21 | Du Pont | 萘異唑啉無脊椎有害動物控制劑 |
PL2957284T3 (pl) | 2007-06-27 | 2018-08-31 | E. I. Du Pont De Nemours And Company | Sposób zwalczania szkodników zwierzęcych |
TWI556741B (zh) | 2007-08-17 | 2016-11-11 | 英特威特國際股份有限公司 | 異唑啉組成物及其作為抗寄生蟲藥上的應用 |
TWI401023B (zh) | 2008-02-06 | 2013-07-11 | Du Pont | 中離子農藥 |
JP2011529895A (ja) * | 2008-07-30 | 2011-12-15 | インターベツト・インターナシヨナル・ベー・ベー | フロルフェニコール中間体として有用なオキサゾリン保護アミノジオール化合物を調製する方法 |
JP2012520847A (ja) | 2009-03-17 | 2012-09-10 | インターベツト・インターナシヨナル・ベー・ベー | 大環状ラクトン薬物送達システム |
JP2013501063A (ja) | 2009-08-05 | 2013-01-10 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | メソイオン性殺虫剤 |
UA107804C2 (en) | 2009-08-05 | 2015-02-25 | Du Pont | Mixtures of pesticides mezoionnyh |
EP2461684A2 (en) | 2009-08-05 | 2012-06-13 | E. I. du Pont de Nemours and Company | Mesoionic pesticides |
UA110924C2 (uk) | 2009-08-05 | 2016-03-10 | Е. І. Дю Пон Де Немур Енд Компані | Мезоіонні пестициди |
KR102060464B1 (ko) | 2010-05-27 | 2019-12-30 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 4-[5-[3-클로로-5-(트라이플루오로메틸)페닐]-4,5-다이하이드로-5-(트라이플루오로메틸)-3-아이속사졸릴]-n-[2-옥소-2-[(2,2,2-트라이플루오로에틸)아미노]에틸]-1-나프탈렌카르복스아미드의 결정 형태 |
AR081970A1 (es) | 2010-06-24 | 2012-10-31 | Intervet Int Bv | Formulacion inyectable de una lactona macrociclica y levamisol, formulacion y uso veterinario |
EP2629772B1 (en) | 2010-10-20 | 2016-05-18 | Galderma S.A. | Ivermectin for use in the treatment of hemorrhoids |
WO2012087630A1 (en) | 2010-12-20 | 2012-06-28 | E.I. Du Pont De Nemours And Company | Pyridine and pyrimidine compounds for controlling invertebrate |
NZ611476A (en) | 2010-12-27 | 2015-10-30 | Intervet Int Bv | Topical localized isoxazoline formulation |
CN103260620A (zh) | 2010-12-27 | 2013-08-21 | 英特维特国际股份有限公司 | 包含三缩四乙二醇的外用局部异噁唑啉制剂 |
WO2013015993A1 (en) | 2011-07-28 | 2013-01-31 | Syngenta Participations Ag | Methods and compositions for controlling nematode pests |
WO2013158422A1 (en) | 2012-04-17 | 2013-10-24 | E. I. Du Pont De Nemours And Company | Heterocyclic compounds for controlling invertebrate pests |
US9409920B1 (en) * | 2015-06-08 | 2016-08-09 | Rotam Agrochem International Company Limited | Method for purifying emamectin benzoate and compositions comprising the same |
US9643991B2 (en) * | 2015-06-08 | 2017-05-09 | Rotam Agrochem International Company Limited | Process for preparing a novel crystalline form of emamectin benzoate and use the same |
CN107344954B (zh) * | 2017-08-07 | 2020-08-11 | 河北蓝泰化工科技有限公司 | 增效型甲氨基阿维菌素b1或b2的盐及制备方法和应用 |
CN108840893A (zh) * | 2018-07-01 | 2018-11-20 | 李万强 | 一种甲氨基阿维菌素苯甲酸盐的新晶型及其制备方法 |
CN108864230B (zh) * | 2018-07-26 | 2021-05-14 | 河北威远生物化工有限公司 | 一种有机磷基团取代的阿维菌素衍生物及其制备方法和应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4366309A (en) * | 1980-03-14 | 1982-12-28 | Schering Corporation | Derivatives of antibiotic AR-5 components |
US4321361A (en) * | 1980-06-12 | 1982-03-23 | Eli Lilly And Company | Demycinosyltylosin and process for its production |
US4427663A (en) * | 1982-03-16 | 1984-01-24 | Merck & Co., Inc. | 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof |
US4831016A (en) * | 1986-10-31 | 1989-05-16 | Merck & Co., Inc. | Reduced avermectin derivatives |
US4874749A (en) * | 1987-07-31 | 1989-10-17 | Merck & Co., Inc. | 4"-Deoxy-4-N-methylamino avermectin Bla/Blb |
-
1991
- 1991-06-24 IL IL9859991A patent/IL98599A/en not_active IP Right Cessation
- 1991-06-26 NZ NZ238705A patent/NZ238705A/xx not_active IP Right Cessation
- 1991-06-27 KR KR1019910010749A patent/KR100224292B1/ko not_active IP Right Cessation
- 1991-06-27 NO NO2001007C patent/NO2001007I2/no unknown
- 1991-06-27 NO NO912535A patent/NO178339C/no not_active IP Right Cessation
- 1991-06-27 AT AT91305815T patent/ATE134377T1/de not_active IP Right Cessation
- 1991-06-27 IE IE225191A patent/IE71175B1/en not_active IP Right Cessation
- 1991-06-27 CY CY194991A patent/CY1949A/xx unknown
- 1991-06-27 DK DK91305815.2T patent/DK0465121T3/da active
- 1991-06-27 ZA ZA914961A patent/ZA914961B/xx unknown
- 1991-06-27 CA CA002045864A patent/CA2045864C/en not_active Expired - Lifetime
- 1991-06-27 AU AU79392/91A patent/AU641777B2/en not_active Expired
- 1991-06-27 ES ES91305815T patent/ES2084110T3/es not_active Expired - Lifetime
- 1991-06-27 DE DE69117223T patent/DE69117223T2/de not_active Expired - Lifetime
- 1991-06-27 PT PT98117A patent/PT98117B/pt not_active IP Right Cessation
- 1991-06-27 EP EP91305815A patent/EP0465121B1/en not_active Expired - Lifetime
- 1991-06-27 FI FI913137A patent/FI97890C/sv not_active IP Right Cessation
- 1991-06-28 JP JP3252729A patent/JPH0822870B2/ja not_active Expired - Lifetime
-
1992
- 1992-04-02 US US07/862,035 patent/US5288710A/en not_active Expired - Lifetime
-
1995
- 1995-08-31 LV LV950265A patent/LV5740B4/xx unknown
-
1996
- 1996-02-22 GR GR960400308T patent/GR3019067T3/el unknown
- 1996-08-15 HK HK157096A patent/HK157096A/xx not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
HK157096A (en) | Stable salts of 4"-deoxy-4"-epimethylamino avermectin B1A/B1B | |
TW234691B (sv) | ||
EP0427247A3 (en) | Pharmaceutical composition with r-alpha-lipoic acid or s-alpha-lipoic acid as the active ingredient | |
AU2724292A (en) | Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of alpha-d-neuraminic acid | |
EP0990648A4 (en) | DERIVATIVES OF 4-CHINOLOL AND AGRICULTURAL AND GARDENING BACTERICIDES THAT CONTAIN THEM AS AN ACTIVE COMPONENT | |
HUT77333A (hu) | Triazolilszármazékok és ezek sói vagy fémkomplexei, előállításuk és alkalmazásuk, hatóanyagként ezeket a vegyületeket tartalmazó mikrobicid készítmények | |
IL100425A0 (en) | 5-chloroquinoline-8-oxyalkanecarboxylic acid derivatives,processes for their preparation and their use as antidotes for herbicides | |
HUT51218A (en) | Herbicides comprising acylated 1,3-dicarbonyl derivatives as active ingredient and compositions containing antidotes as well | |
DE3168350D1 (en) | Pyridine and pyrazine derivatives, preparation of these compounds, fungicidal agents containing these compounds as active ingredients, and the use of such compounds or agents as fungicides in agriculture and in horticulture | |
MD707C2 (ro) | Derivaţi ai sulfonilureei, procedeu de obţinere a lor, produse intermediare pentru ei, substanţă pe baza lor cu acţiune erbicidă şi de reprimare a creşterii plantelor, procedeu de combatere a buruienilor | |
EP0712853A4 (en) | PYRAZOLE DERIVATIVE | |
GR3018989T3 (en) | Solid glyphosate compositions and their use. | |
IL105577A (en) | Fungicidal compositions containing 3-hydroxy- 5-methylisoxazole or salts thereof, methods for the preparation thereof and their use | |
ZA881430B (sv) | ||
DE3471587D1 (en) | Derivatives of benzoic acid, process for their preparation and their use in disinfecting and conserving medicaments | |
IL108997A0 (en) | Heterotricyclically substituted phenyl-cyclohexane-carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them | |
HU896150D0 (en) | Herbicide compositions containing pyrazoles derivatives as active ingredients | |
IL103417A (en) | Alkyl 5- 2-(2, 5-dialkoxyphenyl) ethyl9-2-hydroxybenzoates their preparation and pharmaceutical compositions containing them | |
GB2000973A (en) | Pesticides | |
IL89959A (en) | 1-dimethylcarbamoyl-1 -3-substituted-5- substituted-1h-1,2,4- triazoles and their use as insecticides | |
GR3035058T3 (en) | Use of derivatives of beta-naphthoquinone for inhibiting platelet aggregation. | |
HU912233D0 (en) | Herbicide preparations containing cyclohexenone derivatives as active agents and 1,8-naphtalene-dicarbonic acid anhydrides as antidotes | |
NO952511D0 (no) | Analogifremgangsmåte for fremstilling av terapeutisk aktive, stabile salter av 4''-deoksy-4''-epi-metylaminoavermectin B1a/B1b |