CY1122518T1 - Καινοφανεις προσδετες υποδοχεα οιστρογονου - Google Patents

Καινοφανεις προσδετες υποδοχεα οιστρογονου

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Publication number
CY1122518T1
CY1122518T1 CY20191101088T CY191101088T CY1122518T1 CY 1122518 T1 CY1122518 T1 CY 1122518T1 CY 20191101088 T CY20191101088 T CY 20191101088T CY 191101088 T CY191101088 T CY 191101088T CY 1122518 T1 CY1122518 T1 CY 1122518T1
Authority
CY
Cyprus
Prior art keywords
estrogen receptor
receptor agents
novel estrogen
novel
carbamate
Prior art date
Application number
CY20191101088T
Other languages
English (en)
Inventor
Aiping Cheng
Neeraj Garg
Lars KRÜGER
Joakim LÖFSTEDT
Eva Koch
Konrad Koehler
Lars Hagberg
Daniel NÖTEBERG
Original Assignee
Karo Pharma Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Karo Pharma Ab filed Critical Karo Pharma Ab
Publication of CY1122518T1 publication Critical patent/CY1122518T1/el

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
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    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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Abstract

Οι ενώσεις του τύπου (I) ή ένας φαρμακευτικά αποδεκτός εστέρας, αμίδιο, καρβαμιδικός εστέρας ή άλατός τους, συμπεριλαμβανομένου ενός άλατος ενός τέτοιου εστέρα, αμιδίου ή καρβαμιδικού εστέρα όπου τα R1 έως R9 έχουν έννοιες όπως ορίζονται στην Προδιαγραφή, είναι χρήσιμα ως προσδέτες υποδοχέα οιστρογόνου.
CY20191101088T 2011-08-04 2019-10-17 Καινοφανεις προσδετες υποδοχεα οιστρογονου CY1122518T1 (el)

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