CY1120802T1 - Συνθεση - Google Patents

Συνθεση

Info

Publication number
CY1120802T1
CY1120802T1 CY181101125T CY181101125T CY1120802T1 CY 1120802 T1 CY1120802 T1 CY 1120802T1 CY 181101125 T CY181101125 T CY 181101125T CY 181101125 T CY181101125 T CY 181101125T CY 1120802 T1 CY1120802 T1 CY 1120802T1
Authority
CY
Cyprus
Prior art keywords
compound
treatment
allergic
specific
composition
Prior art date
Application number
CY181101125T
Other languages
English (en)
Inventor
Claire Louise Ambery
Christopher David Edwards
Original Assignee
Glaxosmithkline Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Llc filed Critical Glaxosmithkline Llc
Publication of CY1120802T1 publication Critical patent/CY1120802T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/28—Oxygen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/007—Pulmonary tract; Aromatherapy
    • A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/12—Aerosols; Foams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Otolaryngology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Η ένωση (Ι) και φαρμακευτικώς αποδεκτά άλατα αυτής, είναι επαγωγείς ανθρώπινης ιντερφερόνης. Συγκεκριμένες, διακριτές και ειδικές δοσολογίες ένωσης (Ι) μπορεί να είναι ιδιαιτέρως χρήσιμες στην θεραπεία διαφόρων διαταραχών, για παράδειγμα στην θεραπεία αλλεργικών ασθενειών και άλλων φλεγμονωδών καταστάσεων, για παράδειγμα αλλεργικής ρινίτιδας και αλλεργικού άσθματος.
CY181101125T 2011-07-22 2018-10-31 Συνθεση CY1120802T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161510624P 2011-07-22 2011-07-22
PCT/EP2012/064139 WO2013014052A1 (en) 2011-07-22 2012-07-19 Composition

Publications (1)

Publication Number Publication Date
CY1120802T1 true CY1120802T1 (el) 2019-12-11

Family

ID=46581948

Family Applications (1)

Application Number Title Priority Date Filing Date
CY181101125T CY1120802T1 (el) 2011-07-22 2018-10-31 Συνθεση

Country Status (19)

Country Link
US (2) US10112946B2 (el)
EP (1) EP2734186B1 (el)
JP (1) JP2014520874A (el)
KR (1) KR101916928B1 (el)
CN (1) CN103841958A (el)
AU (2) AU2012289042A1 (el)
BR (1) BR112014001425A2 (el)
CA (1) CA2841361A1 (el)
CY (1) CY1120802T1 (el)
DK (1) DK2734186T3 (el)
ES (1) ES2693122T3 (el)
HR (1) HRP20181667T1 (el)
LT (1) LT2734186T (el)
PL (1) PL2734186T3 (el)
PT (1) PT2734186T (el)
RS (1) RS57995B1 (el)
RU (1) RU2631482C2 (el)
SI (1) SI2734186T1 (el)
WO (1) WO2013014052A1 (el)

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UA103195C2 (uk) 2008-08-11 2013-09-25 Глаксосмитклайн Ллк Похідні пурину для застосування у лікуванні алергій, запальних та інфекційних захворювань
RU2631482C2 (ru) 2011-07-22 2017-09-22 ГЛАКСОСМИТКЛАЙН ЭлЭлСи Композиция
WO2014031815A1 (en) 2012-08-24 2014-02-27 Glaxosmithkline Llc Pyrazolopyrimidine compounds
KR20150085081A (ko) 2012-11-20 2015-07-22 글락소스미스클라인 엘엘씨 신규 화합물
WO2014081645A1 (en) 2012-11-20 2014-05-30 Glaxosmithkline Llc Novel compounds
EP2922550B1 (en) 2012-11-20 2017-04-19 Glaxosmithkline LLC Novel compounds

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Also Published As

Publication number Publication date
AU2012289042A1 (en) 2014-03-13
PL2734186T3 (pl) 2019-01-31
EP2734186B1 (en) 2018-09-12
US20190023707A1 (en) 2019-01-24
PT2734186T (pt) 2018-12-17
DK2734186T3 (en) 2019-01-07
RU2013157398A (ru) 2015-08-27
US10112946B2 (en) 2018-10-30
JP2014520874A (ja) 2014-08-25
KR20140049001A (ko) 2014-04-24
ES2693122T3 (es) 2018-12-07
AU2016202513B2 (en) 2018-03-22
HRP20181667T1 (hr) 2018-12-14
RU2631482C2 (ru) 2017-09-22
WO2013014052A1 (en) 2013-01-31
BR112014001425A2 (pt) 2017-11-21
CA2841361A1 (en) 2013-01-31
US20140288099A1 (en) 2014-09-25
CN103841958A (zh) 2014-06-04
SI2734186T1 (sl) 2018-11-30
RS57995B1 (sr) 2019-01-31
KR101916928B1 (ko) 2018-11-08
LT2734186T (lt) 2018-12-10
EP2734186A1 (en) 2014-05-28

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