CY1114869T1 - Παραγωγα 5-αμινο-2-(1-υδροξυ-αιθυλο)-τετραϋδροπυρανιου - Google Patents
Παραγωγα 5-αμινο-2-(1-υδροξυ-αιθυλο)-τετραϋδροπυρανιουInfo
- Publication number
- CY1114869T1 CY1114869T1 CY20131101136T CY131101136T CY1114869T1 CY 1114869 T1 CY1114869 T1 CY 1114869T1 CY 20131101136 T CY20131101136 T CY 20131101136T CY 131101136 T CY131101136 T CY 131101136T CY 1114869 T1 CY1114869 T1 CY 1114869T1
- Authority
- CY
- Cyprus
- Prior art keywords
- tethydropyranium
- aythyl
- hydroxy
- amino
- production
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D497/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Η εφεύρεση αφορά σε αντιβακτηριακές ενώσεις του τύπου Ι, όπου το R1 παριστάνει αλκοξύ (ειδικά μεθοξύ), το R2 παριστάνει Η ή F, έκαστο από τα R3, R4, R5 και R6 παριστάνει ανεξάρτητα Η ή D, το V παριστάνει CΗ και το W παριστάνει CH ή Ν ή το V παριστάνει Ν και το W παριστάνει CH, το Υ παριστάνει CH ή Ν, το Ζ παριστάνει Ο, S ή CΗ2, και το Α παριστάνει, CΗ2, CH2CH2 ή CD2CD2, και άλατα τέτοιων ενώσεων.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IB2008055261 | 2008-12-12 | ||
EP09796819.2A EP2376497B1 (en) | 2008-12-12 | 2009-12-11 | 5-amino-2-(1-hydroxy-ethyl)-tetrahydropyran derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1114869T1 true CY1114869T1 (el) | 2016-12-14 |
Family
ID=41723046
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20131101136T CY1114869T1 (el) | 2008-12-12 | 2013-12-18 | Παραγωγα 5-αμινο-2-(1-υδροξυ-αιθυλο)-τετραϋδροπυρανιου |
Country Status (28)
Country | Link |
---|---|
US (1) | US8211890B2 (el) |
EP (1) | EP2376497B1 (el) |
JP (1) | JP4955835B2 (el) |
KR (1) | KR101297450B1 (el) |
CN (1) | CN102232078B (el) |
AR (1) | AR074604A1 (el) |
AU (1) | AU2009325902B2 (el) |
BR (1) | BRPI0924081A2 (el) |
CA (1) | CA2744456C (el) |
CL (1) | CL2011001413A1 (el) |
CY (1) | CY1114869T1 (el) |
DK (1) | DK2376497T3 (el) |
ES (1) | ES2435596T3 (el) |
HK (1) | HK1162478A1 (el) |
HR (1) | HRP20140010T1 (el) |
IL (1) | IL213432A (el) |
MA (1) | MA32956B1 (el) |
MX (1) | MX2011005905A (el) |
MY (1) | MY159183A (el) |
NZ (1) | NZ593891A (el) |
PL (1) | PL2376497T3 (el) |
PT (1) | PT2376497E (el) |
RU (1) | RU2525541C2 (el) |
SG (1) | SG172088A1 (el) |
SI (1) | SI2376497T1 (el) |
TW (1) | TWI426076B (el) |
WO (1) | WO2010067332A1 (el) |
ZA (1) | ZA201105095B (el) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR076222A1 (es) | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen |
WO2012164498A1 (en) | 2011-05-31 | 2012-12-06 | Actelion Pharmaceuticals Ltd | New synthetic intermediates for manufacturing antibiotics |
AU2012275499A1 (en) * | 2011-06-27 | 2013-12-19 | Kyorin Pharmaceutical Co., Ltd. | Bridged bicyclic compounds for the treatment of bacterial infections |
WO2013038374A1 (en) | 2011-09-16 | 2013-03-21 | Actelion Pharmaceuticals Ltd | Process for manufacturing a synthetic intermediate |
AR089929A1 (es) | 2012-02-10 | 2014-10-01 | Actelion Pharmaceuticals Ltd | Proceso para manufacturar un derivado de naftiridina |
AR090844A1 (es) | 2012-04-27 | 2014-12-10 | Actelion Pharmaceuticals Ltd | Proceso para elaborar derivados de naftiridina |
TW201722965A (zh) * | 2015-08-16 | 2017-07-01 | 葛蘭素史密斯克藍智慧財產發展有限公司 | 用於抗菌應用之化合物 |
TW201833120A (zh) | 2017-02-17 | 2018-09-16 | 瑞士商愛杜西亞製藥有限公司 | 芳基噁唑啶酮抗生素化合物 |
KR20200037830A (ko) | 2017-08-09 | 2020-04-09 | 데날리 테라퓨틱스 인크. | 화합물, 조성물 및 방법 |
PL3676297T3 (pl) * | 2017-09-01 | 2023-12-11 | Denali Therapeutics Inc. | Związki, kompozycje i sposoby |
TW202045164A (zh) | 2019-02-13 | 2020-12-16 | 美商戴納立製藥公司 | 化合物、組合物及方法 |
MA54959A (fr) | 2019-02-13 | 2021-12-22 | Denali Therapeutics Inc | Composés, compositions et procédés |
Family Cites Families (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SU1095611A1 (ru) * | 1982-09-10 | 2007-06-27 | Краснодарский ордена Трудового Красного Знамени политехнический институт | Хлорид 5-хлорметил-2-этил-8-метил-4Н-м-диоксино-(4,5-с)-пиридиния, обладающий антимикробной активностью |
EP0646115B1 (en) * | 1991-03-28 | 2003-01-22 | Eisai Co., Ltd. | Heterocyclic-cyclic amine derivatives |
GB9822450D0 (en) | 1998-10-14 | 1998-12-09 | Smithkline Beecham Plc | Medicaments |
GB0101577D0 (en) | 2001-01-22 | 2001-03-07 | Smithkline Beecham Plc | Compounds |
GB0112834D0 (en) | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
EP1470125A1 (en) * | 2002-01-29 | 2004-10-27 | Glaxo Group Limited | Aminopiperidine derivatives |
AR040336A1 (es) * | 2002-06-26 | 2005-03-30 | Glaxo Group Ltd | Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto |
TW200427688A (en) | 2002-12-18 | 2004-12-16 | Glaxo Group Ltd | Antibacterial agents |
DE10316081A1 (de) | 2003-04-08 | 2004-10-21 | Morphochem AG Aktiengesellschaft für kombinatorische Chemie | Neue Verbindungen mit antibakterieller Aktivität |
US7160888B2 (en) | 2003-08-22 | 2007-01-09 | Warner Lambert Company Llc | [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia |
JP2008505920A (ja) | 2004-07-08 | 2008-02-28 | グラクソ グループ リミテッド | 抗菌剤 |
JP4887297B2 (ja) * | 2004-09-24 | 2012-02-29 | アクテリオン ファーマシューティカルズ リミテッド | 新規二環式抗生物質 |
WO2006046552A1 (ja) | 2004-10-27 | 2006-05-04 | Toyama Chemical Co., Ltd. | 新規な含窒素複素環化合物およびその塩 |
CN101258157A (zh) * | 2005-05-24 | 2008-09-03 | 阿斯利康(瑞典)有限公司 | 具有抗菌活性的氨基哌啶喹啉及其氮杂等构类似物 |
WO2007016610A2 (en) * | 2005-08-02 | 2007-02-08 | Glaxo Group Limited | Antibacterial agents |
NZ567315A (en) | 2005-10-21 | 2011-01-28 | Glaxo Group Ltd | Peri condensed tricyclic compounds useful as antibacterial agents |
JP2009520779A (ja) | 2005-12-22 | 2009-05-28 | グラクソ グループ リミテッド | 複素環化合物、その製造およびその抗菌剤としての使用 |
DE102005062889A1 (de) | 2005-12-29 | 2007-07-05 | Robert Bosch Gmbh | Elektrische Null-Kraft-Steckvorrichtung |
EP1981881B1 (en) | 2006-01-26 | 2011-12-07 | Actelion Pharmaceuticals Ltd. | Tetrahydropyrane antibiotics |
JP2009529525A (ja) * | 2006-03-10 | 2009-08-20 | アクテリオン ファーマシューティカルズ リミテッド | 抗菌性の化合物 |
WO2007115947A1 (en) | 2006-04-06 | 2007-10-18 | Glaxo Group Limited | Pyrrolo-quinoxalinone derivatives as antibacterials |
GB0613208D0 (en) | 2006-07-03 | 2006-08-09 | Glaxo Group Ltd | Compounds |
EP1992628A1 (en) | 2007-05-18 | 2008-11-19 | Glaxo Group Limited | Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones |
CL2008001003A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
ES2370123T3 (es) * | 2007-06-15 | 2011-12-12 | Actelion Pharmaceuticals Ltd. | Derivados de 3-amino-6-(1-aminoetil)-tetrahidropirano. |
BRPI0820394A2 (pt) | 2007-11-26 | 2015-05-19 | Toyama Chemical Co Ltd | Composto, método para produzir um composto, derivado do ácido kójico, e, agente antibacteriano. |
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2009
- 2009-12-11 MX MX2011005905A patent/MX2011005905A/es active IP Right Grant
- 2009-12-11 EP EP09796819.2A patent/EP2376497B1/en active Active
- 2009-12-11 MY MYPI2011002646A patent/MY159183A/en unknown
- 2009-12-11 RU RU2011128550/04A patent/RU2525541C2/ru not_active IP Right Cessation
- 2009-12-11 NZ NZ593891A patent/NZ593891A/xx not_active IP Right Cessation
- 2009-12-11 DK DK09796819.2T patent/DK2376497T3/da active
- 2009-12-11 KR KR1020117015370A patent/KR101297450B1/ko active IP Right Grant
- 2009-12-11 AR ARP090104821A patent/AR074604A1/es not_active Application Discontinuation
- 2009-12-11 WO PCT/IB2009/055689 patent/WO2010067332A1/en active Application Filing
- 2009-12-11 AU AU2009325902A patent/AU2009325902B2/en not_active Ceased
- 2009-12-11 MA MA34003A patent/MA32956B1/fr unknown
- 2009-12-11 PT PT97968192T patent/PT2376497E/pt unknown
- 2009-12-11 JP JP2011540318A patent/JP4955835B2/ja active Active
- 2009-12-11 SG SG2011042611A patent/SG172088A1/en unknown
- 2009-12-11 TW TW098142582A patent/TWI426076B/zh not_active IP Right Cessation
- 2009-12-11 ES ES09796819T patent/ES2435596T3/es active Active
- 2009-12-11 US US13/139,179 patent/US8211890B2/en not_active Expired - Fee Related
- 2009-12-11 PL PL09796819T patent/PL2376497T3/pl unknown
- 2009-12-11 SI SI200930791T patent/SI2376497T1/sl unknown
- 2009-12-11 CA CA2744456A patent/CA2744456C/en active Active
- 2009-12-11 CN CN200980148242.2A patent/CN102232078B/zh active Active
- 2009-12-11 BR BRPI0924081A patent/BRPI0924081A2/pt active Search and Examination
-
2011
- 2011-06-09 IL IL213432A patent/IL213432A/en not_active IP Right Cessation
- 2011-06-10 CL CL2011001413A patent/CL2011001413A1/es unknown
- 2011-07-11 ZA ZA2011/05095A patent/ZA201105095B/en unknown
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2012
- 2012-03-16 HK HK12102672.7A patent/HK1162478A1/xx not_active IP Right Cessation
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2013
- 2013-12-18 CY CY20131101136T patent/CY1114869T1/el unknown
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2014
- 2014-01-07 HR HRP20140010AT patent/HRP20140010T1/hr unknown
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