MA32956B1 - Derives de 5-amino-2-(1-hydroxyethyl)-tetrahydropyrane - Google Patents
Derives de 5-amino-2-(1-hydroxyethyl)-tetrahydropyraneInfo
- Publication number
- MA32956B1 MA32956B1 MA34003A MA34003A MA32956B1 MA 32956 B1 MA32956 B1 MA 32956B1 MA 34003 A MA34003 A MA 34003A MA 34003 A MA34003 A MA 34003A MA 32956 B1 MA32956 B1 MA 32956B1
- Authority
- MA
- Morocco
- Prior art keywords
- hydroxyethyl
- amino
- tetrahydropyrane
- derivatives
- tetrahydropyrane derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D497/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D497/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having oxygen and sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D497/04—Ortho-condensed systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
L'INVENTION PORTE SUR DES COMPOSÉS ANTIBACTÉRIENS DE FORMULE I, DANS LAQUELLE R1 REPRÉSENTE UN GROUPE ALCOXY (NOTAMMENT MÉTHOXY); R2 REPRÉSENTE H OU F; CHACUN DE R3, R4, R5 ET R6 REPRÉSENTE INDÉPENDAMMENT H OU D; V REPRÉSENTE CH ET W REPRÉSENTE CH OU N, OU V REPRÉSENTE N ET W REPRÉSENTE CH; Y REPRÉSENTE CH OU N; Z REPRÉSENTE O, S OU CH2; ET A REPRÉSENTE CH2, CH2CH2 OU CD2CD2; ET SUR DES SELS DE TELS COMPOSÉS.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IB2008055261 | 2008-12-12 | ||
PCT/IB2009/055689 WO2010067332A1 (fr) | 2008-12-12 | 2009-12-11 | Dérivés de 5-amino-2-(1-hydroxyéthyl)tétrahydropyrane |
Publications (1)
Publication Number | Publication Date |
---|---|
MA32956B1 true MA32956B1 (fr) | 2012-01-02 |
Family
ID=41723046
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA34003A MA32956B1 (fr) | 2008-12-12 | 2009-12-11 | Derives de 5-amino-2-(1-hydroxyethyl)-tetrahydropyrane |
Country Status (28)
Country | Link |
---|---|
US (1) | US8211890B2 (fr) |
EP (1) | EP2376497B1 (fr) |
JP (1) | JP4955835B2 (fr) |
KR (1) | KR101297450B1 (fr) |
CN (1) | CN102232078B (fr) |
AR (1) | AR074604A1 (fr) |
AU (1) | AU2009325902B2 (fr) |
BR (1) | BRPI0924081A2 (fr) |
CA (1) | CA2744456C (fr) |
CL (1) | CL2011001413A1 (fr) |
CY (1) | CY1114869T1 (fr) |
DK (1) | DK2376497T3 (fr) |
ES (1) | ES2435596T3 (fr) |
HK (1) | HK1162478A1 (fr) |
HR (1) | HRP20140010T1 (fr) |
IL (1) | IL213432A (fr) |
MA (1) | MA32956B1 (fr) |
MX (1) | MX2011005905A (fr) |
MY (1) | MY159183A (fr) |
NZ (1) | NZ593891A (fr) |
PL (1) | PL2376497T3 (fr) |
PT (1) | PT2376497E (fr) |
RU (1) | RU2525541C2 (fr) |
SG (1) | SG172088A1 (fr) |
SI (1) | SI2376497T1 (fr) |
TW (1) | TWI426076B (fr) |
WO (1) | WO2010067332A1 (fr) |
ZA (1) | ZA201105095B (fr) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR076222A1 (es) | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen |
EP2748163B1 (fr) | 2011-05-31 | 2016-04-20 | Actelion Pharmaceuticals Ltd. | Procédé pour la préparation des produits intermédiares utiles dans la fabrication d'antibiotiques |
CA2840060A1 (fr) * | 2011-06-27 | 2013-01-03 | Kyorin Pharmaceutical Co., Ltd. | Composes bicycliques pontes pour le traitement des infections bacteriennes |
WO2013038374A1 (fr) | 2011-09-16 | 2013-03-21 | Actelion Pharmaceuticals Ltd | Procédé de préparation d'un intermédiaire de synthèse |
AR089929A1 (es) | 2012-02-10 | 2014-10-01 | Actelion Pharmaceuticals Ltd | Proceso para manufacturar un derivado de naftiridina |
AR090844A1 (es) * | 2012-04-27 | 2014-12-10 | Actelion Pharmaceuticals Ltd | Proceso para elaborar derivados de naftiridina |
UY36851A (es) * | 2015-08-16 | 2017-03-31 | Glaxosmithkline Ip Dev Ltd | Compuestos para uso en aplicaciones antibacterianas |
TW201833120A (zh) | 2017-02-17 | 2018-09-16 | 瑞士商愛杜西亞製藥有限公司 | 芳基噁唑啶酮抗生素化合物 |
IL301709A (en) | 2017-08-09 | 2023-05-01 | Denali Therapeutics Inc | Compounds, preparations and methods |
FI3676297T3 (fi) * | 2017-09-01 | 2023-08-08 | Denali Therapeutics Inc | Yhdisteitä, koostumuksia ja menetelmiä |
CR20210426A (es) | 2019-02-13 | 2021-09-30 | Denali Therapeutics Inc | Compuestos, composiciones y métodos |
Family Cites Families (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SU1095611A1 (ru) * | 1982-09-10 | 2007-06-27 | Краснодарский ордена Трудового Красного Знамени политехнический институт | Хлорид 5-хлорметил-2-этил-8-метил-4Н-м-диоксино-(4,5-с)-пиридиния, обладающий антимикробной активностью |
BR9205811A (pt) * | 1991-03-28 | 1994-06-28 | Pfizer | Derivados heterociclicos de aminas ciclicas |
GB9822450D0 (en) | 1998-10-14 | 1998-12-09 | Smithkline Beecham Plc | Medicaments |
GB0101577D0 (en) | 2001-01-22 | 2001-03-07 | Smithkline Beecham Plc | Compounds |
GB0112834D0 (en) | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
WO2003064421A1 (fr) * | 2002-01-29 | 2003-08-07 | Glaxo Group Limited | Derives aminopiperidine |
AR040336A1 (es) * | 2002-06-26 | 2005-03-30 | Glaxo Group Ltd | Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto |
AR042486A1 (es) | 2002-12-18 | 2005-06-22 | Glaxo Group Ltd | Compuesto de quinolina y naftiridina halosustituido en la posicion 3, procedimiento para preparar el compuesto, composicion farmaceutica que lo comprende y su uso para preparar dicha composicion . |
DE10316081A1 (de) | 2003-04-08 | 2004-10-21 | Morphochem AG Aktiengesellschaft für kombinatorische Chemie | Neue Verbindungen mit antibakterieller Aktivität |
US7160888B2 (en) | 2003-08-22 | 2007-01-09 | Warner Lambert Company Llc | [1,8]naphthyridin-2-ones and related compounds for the treatment of schizophrenia |
JP2008505920A (ja) | 2004-07-08 | 2008-02-28 | グラクソ グループ リミテッド | 抗菌剤 |
WO2006032466A2 (fr) * | 2004-09-24 | 2006-03-30 | Actelion Pharmaceuticals Ltd | Nouveaux antibiotiques bicycliques |
WO2006046552A1 (fr) | 2004-10-27 | 2006-05-04 | Toyama Chemical Co., Ltd. | Nouveaux composés hétérocycliques azotés et sels desdits composés |
US20090131444A1 (en) * | 2005-05-24 | 2009-05-21 | Astrazeneca Ab | Aminopiperidine Quinolines and Their Azaisosteric Analogues with Antibacterial Activity |
WO2007016610A2 (fr) * | 2005-08-02 | 2007-02-08 | Glaxo Group Limited | Agents antibactériens |
DE602006012535D1 (de) | 2005-10-21 | 2010-04-08 | Glaxo Group Ltd | Peri-kondensierte tricyclische verbindungen verwendbar als antibakterielle mittel |
ATE465163T1 (de) | 2005-12-22 | 2010-05-15 | Glaxo Group Ltd | Heterocyclische verbindungen, ihre herstellung und ihre verwendung als antibakterielle mittel |
DE102005062889A1 (de) | 2005-12-29 | 2007-07-05 | Robert Bosch Gmbh | Elektrische Null-Kraft-Steckvorrichtung |
EP1981881B1 (fr) * | 2006-01-26 | 2011-12-07 | Actelion Pharmaceuticals Ltd. | Antibiotiques de type tétrahydropyranne |
WO2007105154A2 (fr) * | 2006-03-10 | 2007-09-20 | Actelion Pharmaceuticals Ltd | Composés antibiotiques |
US7709483B2 (en) | 2006-04-06 | 2010-05-04 | Glaxo Group Limited | Pyrrolo-quinoxalinone derivatives as antibacterials |
GB0613208D0 (en) | 2006-07-03 | 2006-08-09 | Glaxo Group Ltd | Compounds |
EP1992628A1 (fr) | 2007-05-18 | 2008-11-19 | Glaxo Group Limited | Dérivés et analogues de N-éthylquinolones et N-éthylazaquinolones |
CL2008001003A1 (es) | 2007-04-11 | 2008-10-17 | Actelion Pharmaceuticals Ltd | Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana. |
MX2009013254A (es) * | 2007-06-15 | 2010-01-25 | Actelion Pharmaceuticals Ltd | Derivados 3-amino-6(1-amino-etil)-tetrahidropirano. |
JP5491195B2 (ja) | 2007-11-26 | 2014-05-14 | 富山化学工業株式会社 | 新規なナフチリジン誘導体1水和物およびその製造法 |
-
2009
- 2009-12-11 SI SI200930791T patent/SI2376497T1/sl unknown
- 2009-12-11 AR ARP090104821A patent/AR074604A1/es not_active Application Discontinuation
- 2009-12-11 US US13/139,179 patent/US8211890B2/en active Active
- 2009-12-11 CN CN200980148242.2A patent/CN102232078B/zh active Active
- 2009-12-11 MX MX2011005905A patent/MX2011005905A/es active IP Right Grant
- 2009-12-11 CA CA2744456A patent/CA2744456C/fr active Active
- 2009-12-11 DK DK09796819.2T patent/DK2376497T3/da active
- 2009-12-11 PT PT97968192T patent/PT2376497E/pt unknown
- 2009-12-11 KR KR1020117015370A patent/KR101297450B1/ko active IP Right Grant
- 2009-12-11 PL PL09796819T patent/PL2376497T3/pl unknown
- 2009-12-11 JP JP2011540318A patent/JP4955835B2/ja active Active
- 2009-12-11 TW TW098142582A patent/TWI426076B/zh not_active IP Right Cessation
- 2009-12-11 RU RU2011128550/04A patent/RU2525541C2/ru not_active IP Right Cessation
- 2009-12-11 AU AU2009325902A patent/AU2009325902B2/en not_active Ceased
- 2009-12-11 SG SG2011042611A patent/SG172088A1/en unknown
- 2009-12-11 MA MA34003A patent/MA32956B1/fr unknown
- 2009-12-11 BR BRPI0924081A patent/BRPI0924081A2/pt active Search and Examination
- 2009-12-11 ES ES09796819T patent/ES2435596T3/es active Active
- 2009-12-11 EP EP09796819.2A patent/EP2376497B1/fr active Active
- 2009-12-11 NZ NZ593891A patent/NZ593891A/xx not_active IP Right Cessation
- 2009-12-11 MY MYPI2011002646A patent/MY159183A/en unknown
- 2009-12-11 WO PCT/IB2009/055689 patent/WO2010067332A1/fr active Application Filing
-
2011
- 2011-06-09 IL IL213432A patent/IL213432A/en not_active IP Right Cessation
- 2011-06-10 CL CL2011001413A patent/CL2011001413A1/es unknown
- 2011-07-11 ZA ZA2011/05095A patent/ZA201105095B/en unknown
-
2012
- 2012-03-16 HK HK12102672.7A patent/HK1162478A1/xx not_active IP Right Cessation
-
2013
- 2013-12-18 CY CY20131101136T patent/CY1114869T1/el unknown
-
2014
- 2014-01-07 HR HRP20140010AT patent/HRP20140010T1/hr unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MA32956B1 (fr) | Derives de 5-amino-2-(1-hydroxyethyl)-tetrahydropyrane | |
ECSP099091A (es) | Profarmaco de compuesto de cinamida | |
CY1112467T1 (el) | Παραγωγα 1-θειο-d-γλυκιτολης | |
NO20071642L (no) | N-Benzensulfonylsubstituerte anilino-pyrimidinanaloger | |
CR9830A (es) | Compuestos de amino-5-[4-(difluorometoxi)fenil]-5-fenilimidazolona para la inhibicion de la b-secretasa | |
ECSP099818A (es) | Procesos para la preparacion de pirazoles | |
EA200801608A1 (ru) | Производные бензимидазолонкарбоновой кислоты | |
MX337588B (es) | Metodo para preparar derivados de 5-haloalquil-4,5-dihidroisoxasol . | |
CY1111628T1 (el) | Υποκατεστημενες ενωσεις δικυκλολακταμης | |
ME01992B (fr) | Composes diarylhydantoines | |
CY1114452T1 (el) | Ενωσεις πυρρολιου | |
DK1817300T3 (da) | Forstærkere af glutamat-receptorer | |
CY1115767T1 (el) | 1η-κιναζολινο-2,4-διονες | |
GT200500296A (es) | Sintesis asimetrica de derivados del dehidrobenzofurano | |
EA200801365A1 (ru) | Замещенные 5-фенил-3,6-дигидро-2-оксо-6h-1,3,4-тиадиазины | |
UY31750A (es) | Compuestos y composiciones como inhibidores de quinasa | |
CY1113716T1 (el) | Νεα μεθοδος συνθεσης της αγομελατινης | |
MX344529B (es) | Derivados antibioticos de 2 - oxo -oxazolidin - 3, 5 -diilo. | |
UA117151C2 (uk) | N-ациліміногетероциклічні сполуки | |
EA200801366A1 (ru) | Производные 3,6-дигидро-2-оксо-6н-1,3,4-тиадиазина | |
ATE517869T1 (de) | Herstellung substituierter morphinan-6-one und salzen und zwischenprodukten davon | |
EA200900946A1 (ru) | Новый способ синтеза агомелатина | |
CR11463A (es) | Compuestos de piridilmetil-sulfonamida | |
MY149400A (en) | Bridged six-membered ring compounds | |
EA200800070A1 (ru) | Производные 2-(1h-индолилсульфанил)ариламина |