UY31750A - Compuestos y composiciones como inhibidores de quinasa - Google Patents
Compuestos y composiciones como inhibidores de quinasaInfo
- Publication number
- UY31750A UY31750A UY0001031750A UY31750A UY31750A UY 31750 A UY31750 A UY 31750A UY 0001031750 A UY0001031750 A UY 0001031750A UY 31750 A UY31750 A UY 31750A UY 31750 A UY31750 A UY 31750A
- Authority
- UY
- Uruguay
- Prior art keywords
- compositions
- compounds
- quinasa
- inhibitors
- quinasa inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
La invención se rediere a composiciones de triazina y pirimidina y mètodos para utilizar las composiciones de la Fórmula (1) o (2): donde R1, R2, R3, R4, R5, X Y, Z1, Ph, B m, n son como se los definió anteriormente.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US4311108P | 2008-04-07 | 2008-04-07 | |
US9588308P | 2008-09-10 | 2008-09-10 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY31750A true UY31750A (es) | 2009-12-14 |
Family
ID=40786670
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001031750A UY31750A (es) | 2008-04-07 | 2009-04-03 | Compuestos y composiciones como inhibidores de quinasa |
Country Status (13)
Country | Link |
---|---|
US (1) | US8518931B2 (es) |
EP (1) | EP2271645A1 (es) |
JP (1) | JP5214799B2 (es) |
KR (1) | KR20110002080A (es) |
CN (1) | CN102056925A (es) |
AR (1) | AR071300A1 (es) |
AU (1) | AU2009233963B2 (es) |
BR (1) | BRPI0910979A2 (es) |
CA (1) | CA2720944C (es) |
EA (1) | EA018484B1 (es) |
MX (1) | MX2010011069A (es) |
UY (1) | UY31750A (es) |
WO (1) | WO2009126514A1 (es) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI389893B (zh) | 2007-07-06 | 2013-03-21 | Astellas Pharma Inc | 二(芳胺基)芳基化合物 |
CA2723961C (en) | 2008-05-21 | 2017-03-21 | Ariad Pharmaceuticals, Inc. | Phosphorous derivatives as kinase inhibitors |
US9273077B2 (en) | 2008-05-21 | 2016-03-01 | Ariad Pharmaceuticals, Inc. | Phosphorus derivatives as kinase inhibitors |
PL2428508T3 (pl) | 2009-05-08 | 2016-05-31 | Astellas Pharma Inc | Diaminoheterocykliczny związek karboksyamidowy |
WO2012097478A1 (en) * | 2011-01-21 | 2012-07-26 | Abbott Laboratories | Bicyclic carboxamide inhibitors of kinases |
CN103501612B (zh) | 2011-05-04 | 2017-03-29 | 阿里亚德医药股份有限公司 | 抑制表皮生长因子受体导致的癌症中细胞增殖的化合物 |
WO2013169401A1 (en) | 2012-05-05 | 2013-11-14 | Ariad Pharmaceuticals, Inc. | Compounds for inhibiting cell proliferation in egfr-driven cancers |
EP2867233A1 (en) | 2012-07-03 | 2015-05-06 | Aurigene Discovery Technologies Limited | 3-(PYRAZOLYL)-1H-PYRROLO[2,3-b]PYRIDINE DERIVATIVES AS KINASE INHIBITORS |
CN104854101B (zh) * | 2012-11-06 | 2018-05-01 | 上海复尚慧创医药研究有限公司 | Alk激酶抑制剂 |
US9611283B1 (en) | 2013-04-10 | 2017-04-04 | Ariad Pharmaceuticals, Inc. | Methods for inhibiting cell proliferation in ALK-driven cancers |
CN103570728B (zh) * | 2013-11-12 | 2015-12-30 | 山东大学 | 一种取代吡唑并[1,5-a]嘧啶类衍生物及其制备方法与应用 |
CA2940918C (en) * | 2014-03-27 | 2023-10-24 | Janssen Pharmaceutica Nv | Substituted 4,5,6,7-tetrahydro-pyrazolo[1,5-.alpha.]pyrazine derivatives and 5,6,7,8-tetrahydro-4h-pyrazolo[1,5-.alpha.][1,4]diazepine derivatives as ros1 inhibitors |
EP3778604A1 (en) * | 2015-02-13 | 2021-02-17 | Dana Farber Cancer Institute, Inc. | Lrrk2 inhibitors and methods of making and using the same |
JP7216705B2 (ja) | 2017-07-28 | 2023-02-02 | ニンバス ラクシュミ, インコーポレイテッド | Tyk2阻害剤およびその使用方法 |
CN110483526B (zh) * | 2019-09-09 | 2021-10-01 | 辽宁大学 | 含芳基腙结构的吡唑并[1,5-a]嘧啶类衍生物及其应用 |
GB201915618D0 (en) | 2019-10-28 | 2019-12-11 | Univ Oslo | ALK inhibitors for treatment of ALK-negative cancer and antibody-mediated diseases |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NL7406641A (es) | 1973-05-22 | 1974-11-26 | ||
EP1345941A1 (fr) | 2000-12-20 | 2003-09-24 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | Inhibiteurs de kinases dependantes des cylines (cdk) et de la glycogene synthase kinase-3 (gsk-3) |
FR2842809A1 (fr) | 2002-07-26 | 2004-01-30 | Greenpharma Sas | NOUVELLES PYRAZOLO[1,5-a]-1,3,5-TRIAZINES SUBSTITUEES ET LEURS ANALOGUES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, UTILISATION A TITRE DE MEDICAMENT ET PROCEDES POUR LEUR PREPARATION |
KR20050033659A (ko) * | 2002-09-04 | 2005-04-12 | 쉐링 코포레이션 | 사이클린 의존성 키나제 억제제로서의 피라졸로[1,5-a]피리미딘 화합물 |
EP1599482A4 (en) * | 2003-02-28 | 2008-10-01 | Teijin Pharma Ltd | PYRAZOLO1,5-A PYRIMIDINE DERIVATIVES |
GB0305559D0 (en) * | 2003-03-11 | 2003-04-16 | Teijin Ltd | Compounds |
US20070179161A1 (en) * | 2003-03-31 | 2007-08-02 | Vernalis (Cambridge) Limited. | Pyrazolopyrimidine compounds and their use in medicine |
US20070060595A1 (en) * | 2003-10-10 | 2007-03-15 | Toshio Yoshizawa | Novel fused heterocyclic compound and use thereof |
PE20051128A1 (es) | 2004-02-25 | 2006-01-16 | Schering Corp | Pirazolotriazinas como inhibidores de quinasa |
JP2006160628A (ja) | 2004-12-03 | 2006-06-22 | Ishihara Sangyo Kaisha Ltd | アデノシンA2a受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物 |
JP2008524330A (ja) * | 2004-12-21 | 2008-07-10 | シェーリング コーポレイション | ピラゾロ[1,5−A]ピリミジンアデノシンA2a受容体アンタゴニスト |
US7723336B2 (en) | 2005-09-22 | 2010-05-25 | Bristol-Myers Squibb Company | Fused heterocyclic compounds useful as kinase modulators |
US7517882B2 (en) * | 2006-09-18 | 2009-04-14 | Polaris Group | Protein kinase inhibitors |
WO2008057402A2 (en) | 2006-11-02 | 2008-05-15 | Cytovia, Inc. | N-aryl-isoxazolopyrimidin-4-amines and related compounds as activators of caspases and inducers of apoptosis and the use thereof |
-
2009
- 2009-04-03 US US12/936,193 patent/US8518931B2/en not_active Expired - Fee Related
- 2009-04-03 UY UY0001031750A patent/UY31750A/es not_active Application Discontinuation
- 2009-04-03 EP EP09731237A patent/EP2271645A1/en not_active Withdrawn
- 2009-04-03 MX MX2010011069A patent/MX2010011069A/es not_active Application Discontinuation
- 2009-04-03 CN CN2009801210269A patent/CN102056925A/zh active Pending
- 2009-04-03 BR BRPI0910979A patent/BRPI0910979A2/pt not_active IP Right Cessation
- 2009-04-03 AU AU2009233963A patent/AU2009233963B2/en not_active Ceased
- 2009-04-03 JP JP2011504085A patent/JP5214799B2/ja not_active Expired - Fee Related
- 2009-04-03 CA CA2720944A patent/CA2720944C/en not_active Expired - Fee Related
- 2009-04-03 KR KR1020107024934A patent/KR20110002080A/ko not_active Application Discontinuation
- 2009-04-03 EA EA201001596A patent/EA018484B1/ru not_active IP Right Cessation
- 2009-04-03 WO PCT/US2009/039380 patent/WO2009126514A1/en active Application Filing
- 2009-04-07 AR ARP090101228A patent/AR071300A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
CA2720944A1 (en) | 2009-10-15 |
JP2011516554A (ja) | 2011-05-26 |
JP5214799B2 (ja) | 2013-06-19 |
AR071300A1 (es) | 2010-06-09 |
EA018484B1 (ru) | 2013-08-30 |
CN102056925A (zh) | 2011-05-11 |
MX2010011069A (es) | 2010-11-12 |
CA2720944C (en) | 2012-12-18 |
US8518931B2 (en) | 2013-08-27 |
BRPI0910979A2 (pt) | 2016-01-05 |
EA201001596A1 (ru) | 2011-04-29 |
KR20110002080A (ko) | 2011-01-06 |
US20110190264A1 (en) | 2011-08-04 |
AU2009233963B2 (en) | 2011-10-06 |
WO2009126514A1 (en) | 2009-10-15 |
WO2009126514A8 (en) | 2010-10-21 |
AU2009233963A1 (en) | 2009-10-15 |
EP2271645A1 (en) | 2011-01-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20181025 |