CS276093B6 - Process for preparing novel derivatives of imidazole - Google Patents
Process for preparing novel derivatives of imidazole Download PDFInfo
- Publication number
- CS276093B6 CS276093B6 CS88891A CS89188A CS276093B6 CS 276093 B6 CS276093 B6 CS 276093B6 CS 88891 A CS88891 A CS 88891A CS 89188 A CS89188 A CS 89188A CS 276093 B6 CS276093 B6 CS 276093B6
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- tert
- hydroxy
- compound
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C07D233/61—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms not forming part of a nitro radical, attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epoxy Resins (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH107387 | 1987-03-20 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CS8800891A2 CS8800891A2 (en) | 1990-09-12 |
| CS276093B6 true CS276093B6 (en) | 1992-04-15 |
Family
ID=4201822
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS88891A CS276093B6 (en) | 1987-03-20 | 1988-02-12 | Process for preparing novel derivatives of imidazole |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US4908363A (hu) |
| EP (1) | EP0283857B1 (hu) |
| JP (1) | JPS63253070A (hu) |
| KR (1) | KR880011117A (hu) |
| CN (1) | CN1016169B (hu) |
| AT (1) | ATE73777T1 (hu) |
| AU (1) | AU613349B2 (hu) |
| CS (1) | CS276093B6 (hu) |
| DE (1) | DE3869163D1 (hu) |
| DK (1) | DK59888A (hu) |
| ES (1) | ES2032482T3 (hu) |
| FI (1) | FI880813A (hu) |
| GR (1) | GR3004729T3 (hu) |
| HU (1) | HU201312B (hu) |
| IL (1) | IL85725A (hu) |
| MC (1) | MC1919A1 (hu) |
| MX (1) | MX10721A (hu) |
| NO (1) | NO170215C (hu) |
| NZ (1) | NZ223862A (hu) |
| PT (1) | PT87025B (hu) |
| SU (1) | SU1657057A3 (hu) |
| YU (1) | YU46444B (hu) |
| ZA (1) | ZA881810B (hu) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5073566A (en) * | 1989-11-30 | 1991-12-17 | Eli Lilly And Company | Angiotensin ii antagonist 1,3-imidazoles and use thereas |
| US5401851A (en) * | 1992-06-03 | 1995-03-28 | Eli Lilly And Company | Angiotensin II antagonists |
| US5612360A (en) * | 1992-06-03 | 1997-03-18 | Eli Lilly And Company | Angiotensin II antagonists |
| US5574057A (en) * | 1993-02-03 | 1996-11-12 | University Of Utah Research Foundation | Naamidine A extracted from sea sponges and methods for its use as an anti-tumor agent |
| US5523310A (en) * | 1994-12-05 | 1996-06-04 | Hoffmann-La Roche Inc. | 1,2,3-triazole derivatives |
| AU1383200A (en) | 1998-11-23 | 2000-06-13 | F. Hoffmann-La Roche Ag | Synthesis of anti-inflammatory (1,2,3)triazoles |
| DE10132896A1 (de) * | 2001-07-06 | 2003-01-16 | Bayer Cropscience Ag | Heterocyclische Amidderivate |
| WO2003010143A1 (en) * | 2001-07-26 | 2003-02-06 | Samsung Electronics Co., Ltd. | Dialkylhydroxybenzoic acid derivatives containing metal chelating groups and their therapeutic uses |
| EP1431292A1 (en) * | 2002-12-16 | 2004-06-23 | Laboratoire Theramex | 1-N-phenylamino-1H-imidazole derivatives as aromatase inhibitors |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3152228C1 (de) * | 1980-07-31 | 1985-07-18 | Vadim Michajlovič Frjazino Moskovskaja oblast' Šošin | 2,2'-Azoimidazolderivate,Verfahren zu ihrer Herstellung und ihre Verwendung zur Herstellung eines fluessigkristallinen Materials |
| DE3674054D1 (de) * | 1985-04-26 | 1990-10-18 | Hoffmann La Roche | 1,3-disubstituierte imidazoliumsalze. |
| ZW6687A1 (en) * | 1986-05-13 | 1987-12-02 | Hoffmann La Roche | 1,3-disubstituted imidazolium salts |
| MW7087A1 (en) * | 1986-10-03 | 1988-05-11 | Hoffmann La Roche | 1,3-disubstituted imidazolium salts |
| KR890700582A (ko) * | 1987-03-20 | 1989-04-25 | 사무엘 에스. 블라이트 | 살진균성 아미노트리아졸 및 아미노이미다졸 |
-
1988
- 1988-02-05 DK DK059888A patent/DK59888A/da not_active Application Discontinuation
- 1988-02-12 CS CS88891A patent/CS276093B6/cs unknown
- 1988-02-22 FI FI880813A patent/FI880813A/fi not_active Application Discontinuation
- 1988-03-01 YU YU40388A patent/YU46444B/sh unknown
- 1988-03-09 AT AT88103746T patent/ATE73777T1/de active
- 1988-03-09 ES ES198888103746T patent/ES2032482T3/es not_active Expired - Lifetime
- 1988-03-09 DE DE8888103746T patent/DE3869163D1/de not_active Expired - Fee Related
- 1988-03-09 EP EP88103746A patent/EP0283857B1/de not_active Expired - Lifetime
- 1988-03-10 MX MX1072188A patent/MX10721A/es unknown
- 1988-03-11 NZ NZ223862A patent/NZ223862A/xx unknown
- 1988-03-14 ZA ZA881810A patent/ZA881810B/xx unknown
- 1988-03-14 IL IL85725A patent/IL85725A/xx unknown
- 1988-03-15 US US07/169,207 patent/US4908363A/en not_active Expired - Fee Related
- 1988-03-16 HU HU881238A patent/HU201312B/hu not_active IP Right Cessation
- 1988-03-17 MC MC881959A patent/MC1919A1/xx unknown
- 1988-03-18 PT PT87025A patent/PT87025B/pt not_active IP Right Cessation
- 1988-03-18 SU SU884355836A patent/SU1657057A3/ru active
- 1988-03-18 JP JP63063734A patent/JPS63253070A/ja active Pending
- 1988-03-18 NO NO881199A patent/NO170215C/no unknown
- 1988-03-19 CN CN88101452A patent/CN1016169B/zh not_active Expired
- 1988-03-19 KR KR1019880002924A patent/KR880011117A/ko not_active Application Discontinuation
- 1988-03-21 AU AU13532/88A patent/AU613349B2/en not_active Ceased
-
1992
- 1992-05-27 GR GR920401077T patent/GR3004729T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR880011117A (ko) | 1988-10-26 |
| MX10721A (es) | 1993-09-01 |
| AU1353288A (en) | 1988-09-22 |
| YU46444B (sh) | 1993-10-20 |
| HUT49581A (en) | 1989-10-30 |
| JPS63253070A (ja) | 1988-10-20 |
| PT87025B (pt) | 1992-06-30 |
| YU40388A (en) | 1990-02-28 |
| FI880813A0 (fi) | 1988-02-22 |
| CN1016169B (zh) | 1992-04-08 |
| NO170215C (no) | 1992-09-23 |
| SU1657057A3 (ru) | 1991-06-15 |
| PT87025A (pt) | 1988-04-01 |
| NZ223862A (en) | 1990-08-28 |
| FI880813A (fi) | 1988-09-21 |
| US4908363A (en) | 1990-03-13 |
| IL85725A (en) | 1991-12-12 |
| AU613349B2 (en) | 1991-08-01 |
| EP0283857B1 (de) | 1992-03-18 |
| NO881199D0 (no) | 1988-03-18 |
| ZA881810B (en) | 1988-09-20 |
| DK59888A (da) | 1988-09-21 |
| EP0283857A1 (de) | 1988-09-28 |
| NO170215B (no) | 1992-06-15 |
| CN88101452A (zh) | 1988-10-05 |
| DK59888D0 (da) | 1988-02-05 |
| GR3004729T3 (hu) | 1993-04-28 |
| HU201312B (en) | 1990-10-28 |
| CS8800891A2 (en) | 1990-09-12 |
| DE3869163D1 (de) | 1992-04-23 |
| ES2032482T3 (es) | 1993-02-16 |
| NO881199L (no) | 1988-09-21 |
| ATE73777T1 (de) | 1992-04-15 |
| IL85725A0 (en) | 1988-08-31 |
| MC1919A1 (fr) | 1989-04-06 |
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