CS262692B2 - Process for preparing new derivatives of 1h,3h-pyrrolo-/1,2-c/thiazole - Google Patents

Process for preparing new derivatives of 1h,3h-pyrrolo-/1,2-c/thiazole Download PDF

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Publication number
CS262692B2
CS262692B2 CS875013A CS501387A CS262692B2 CS 262692 B2 CS262692 B2 CS 262692B2 CS 875013 A CS875013 A CS 875013A CS 501387 A CS501387 A CS 501387A CS 262692 B2 CS262692 B2 CS 262692B2
Authority
CS
Czechoslovakia
Prior art keywords
total
temperature
kpa
pyridyl
pyrrolo
Prior art date
Application number
CS875013A
Other languages
Czech (cs)
English (en)
Other versions
CS501387A2 (en
Inventor
Jean-Louis Fabre
Claude James
Daniel Lave
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Priority to CS88215A priority Critical patent/CS262700B2/cs
Publication of CS501387A2 publication Critical patent/CS501387A2/cs
Publication of CS262692B2 publication Critical patent/CS262692B2/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Steroid Compounds (AREA)
CS875013A 1986-07-04 1987-07-02 Process for preparing new derivatives of 1h,3h-pyrrolo-/1,2-c/thiazole CS262692B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS88215A CS262700B2 (cs) 1987-07-02 1988-01-12 Způsob výroby nového derivátu 1H, 3H-pyrrolo(l,2-e]thiazolu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8609728A FR2601015B1 (fr) 1986-07-04 1986-07-04 Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
CS501387A2 CS501387A2 (en) 1988-08-16
CS262692B2 true CS262692B2 (en) 1989-03-14

Family

ID=9337075

Family Applications (1)

Application Number Title Priority Date Filing Date
CS875013A CS262692B2 (en) 1986-07-04 1987-07-02 Process for preparing new derivatives of 1h,3h-pyrrolo-/1,2-c/thiazole

Country Status (28)

Country Link
US (1) US4783472A (de)
EP (1) EP0253711B1 (de)
JP (1) JPS6322589A (de)
KR (1) KR880001681A (de)
AT (1) ATE53037T1 (de)
AU (1) AU597996B2 (de)
BG (2) BG47498A3 (de)
CA (1) CA1294966C (de)
CS (1) CS262692B2 (de)
DD (1) DD263772A5 (de)
DE (1) DE3762861D1 (de)
DK (1) DK340087A (de)
ES (1) ES2015070B3 (de)
FI (1) FI84727C (de)
FR (1) FR2601015B1 (de)
GR (1) GR3000502T3 (de)
HU (1) HU198727B (de)
IE (1) IE60743B1 (de)
IL (1) IL83066A (de)
MA (1) MA21027A1 (de)
MX (1) MX173398B (de)
NO (1) NO170419C (de)
NZ (1) NZ220929A (de)
PL (2) PL149903B1 (de)
PT (1) PT85235B (de)
SU (2) SU1528323A3 (de)
TN (1) TNSN87083A1 (de)
ZA (1) ZA874814B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2617484B1 (fr) * 1987-07-02 1989-10-20 Rhone Poulenc Sante Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2644456B1 (fr) * 1989-03-17 1991-07-05 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
JP3061631B2 (ja) * 1989-10-11 2000-07-10 山之内製薬株式会社 新規なヘテロ環化合物およびその製造法
FR2662606A1 (fr) * 1990-06-01 1991-12-06 Rhone Poulenc Sante Compositions pharmaceutiques pour le traitement de la fibrillation ventriculaire, du syndrome de menace de l'infarctus du myocarde et de l'angine de poitrine contenant le n-(benzoyl-3 phenyl) (pyridyl-3)-3 1h,3h-pyrrolo[1,2-c]thiazolecarboxamide-7.
FR2687574B1 (fr) * 1992-02-25 1995-05-05 Rhone Poulenc Rorer Sa Nouvelle application therapeutique de derives du pyridylpyrrolothiazole carboxamide.
GB9207645D0 (en) * 1992-04-08 1992-05-27 Smithkline Beecham Corp Methods
AU2002367023A1 (en) * 2001-12-21 2003-07-30 Cytokinetics, Inc. Compositions and methods for treating heart failure
JP2010518014A (ja) 2007-01-31 2010-05-27 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害剤として有用な２−アミノピリジン誘導体
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
JP5631310B2 (ja) 2008-07-23 2014-11-26 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ 三環式ピラゾロピリジンキナーゼ阻害剤
EP2318407B1 (de) 2008-07-23 2013-01-02 Vertex Pharmaceuticals Incorporated Pyrazolpyridine als kinaseinhibitoren
CA2732765A1 (en) * 2008-08-06 2010-02-11 Vertex Pharmaceuticals Incorporated Aminopyridine kinase inhibitors
WO2010129668A1 (en) 2009-05-06 2010-11-11 Vertex Pharmaceuticals Incorporated Pyrazolopyridines
MX2012008643A (es) 2010-01-27 2013-02-26 Vertex Pharma Inhibidores de cinasas de pirazolopiridinas.
US9067932B2 (en) 2010-01-27 2015-06-30 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
CN102869663A (zh) 2010-01-27 2013-01-09 沃泰克斯药物股份有限公司 吡唑并吡嗪激酶抑制剂
KR102608281B1 (ko) * 2022-07-27 2023-12-01 김규현 감자를 이용한 맥주 제조 방법 및 이에 의해 제조된 감자 맥주

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2541280B1 (fr) * 1983-01-13 1985-06-21 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent
US4500532A (en) * 1983-03-03 1985-02-19 Usv Pharmaceutical Corporation 1-(Substituted aminoalkyl)-1,4-dihydropyridines
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
IL83066A (en) 1991-01-31
FI84727C (fi) 1992-01-10
PL266582A1 (en) 1988-09-01
NO170419B (no) 1992-07-06
IE60743B1 (en) 1994-08-10
MA21027A1 (fr) 1988-04-01
CA1294966C (fr) 1992-01-28
ES2015070B3 (es) 1990-08-01
FR2601015B1 (fr) 1988-08-05
FI872931A0 (fi) 1987-07-02
CS501387A2 (en) 1988-08-16
SU1528323A3 (ru) 1989-12-07
NO872779D0 (no) 1987-07-02
ATE53037T1 (de) 1990-06-15
DE3762861D1 (de) 1990-06-28
ZA874814B (en) 1988-03-30
SU1588284A3 (ru) 1990-08-23
PT85235B (pt) 1990-03-30
IL83066A0 (en) 1987-12-31
BG47498A3 (bg) 1990-07-16
EP0253711B1 (de) 1990-05-23
BG47038A3 (bg) 1990-04-16
PT85235A (fr) 1987-08-01
US4783472A (en) 1988-11-08
IE871767L (en) 1988-01-04
DD263772A5 (de) 1989-01-11
HU198727B (en) 1989-11-28
PL149434B1 (en) 1990-02-28
TNSN87083A1 (fr) 1990-01-01
AU597996B2 (en) 1990-06-14
MX173398B (es) 1994-02-28
NO170419C (no) 1992-10-14
NZ220929A (en) 1989-09-27
PL149903B1 (en) 1990-03-31
FI872931A7 (fi) 1988-01-05
MX7191A (es) 1993-10-01
GR3000502T3 (en) 1991-07-31
AU7504787A (en) 1988-01-07
DK340087D0 (da) 1987-07-02
JPS6322589A (ja) 1988-01-30
HUT44791A (en) 1988-04-28
DK340087A (da) 1988-01-05
KR880001681A (ko) 1988-04-26
FR2601015A1 (fr) 1988-01-08
NO872779L (no) 1988-01-05
FI84727B (fi) 1991-09-30
EP0253711A1 (de) 1988-01-20

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