CS235972B2 - Method of new azinorifamycines production - Google Patents

Method of new azinorifamycines production Download PDF

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Publication number
CS235972B2
CS235972B2 CS828107A CS810782A CS235972B2 CS 235972 B2 CS235972 B2 CS 235972B2 CS 828107 A CS828107 A CS 828107A CS 810782 A CS810782 A CS 810782A CS 235972 B2 CS235972 B2 CS 235972B2
Authority
CS
Czechoslovakia
Prior art keywords
delta
carbon atoms
group
alkyl
formula
Prior art date
Application number
CS828107A
Other languages
Czech (cs)
English (en)
Inventor
Giovanni Franceschi
Leonardo Marsili
Aurora Sanfilippo
Sergio Vioglio
Original Assignee
Parmitalia Carlo Erba S P A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Parmitalia Carlo Erba S P A filed Critical Parmitalia Carlo Erba S P A
Publication of CS235972B2 publication Critical patent/CS235972B2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CS828107A 1981-11-17 1982-11-15 Method of new azinorifamycines production CS235972B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8134549 1981-11-17

Publications (1)

Publication Number Publication Date
CS235972B2 true CS235972B2 (en) 1985-05-15

Family

ID=10525927

Family Applications (1)

Application Number Title Priority Date Filing Date
CS828107A CS235972B2 (en) 1981-11-17 1982-11-15 Method of new azinorifamycines production

Country Status (32)

Country Link
US (1) US4447432A (da)
JP (1) JPS5892682A (da)
KR (1) KR880001284B1 (da)
AT (1) AT376222B (da)
AU (1) AU553727B2 (da)
BE (1) BE895020A (da)
CA (1) CA1205074A (da)
CH (1) CH657619A5 (da)
CS (1) CS235972B2 (da)
DE (1) DE3241764A1 (da)
DK (1) DK157873C (da)
ES (1) ES517153A0 (da)
FI (1) FI73436C (da)
FR (1) FR2516514A1 (da)
GB (2) GB2110677B (da)
GR (1) GR76790B (da)
HK (1) HK74687A (da)
HU (1) HU186160B (da)
IE (1) IE54153B1 (da)
IL (1) IL67263A (da)
IT (1) IT1224111B (da)
MX (1) MX157130A (da)
NL (1) NL8204330A (da)
NO (1) NO167290C (da)
NZ (1) NZ202495A (da)
PH (1) PH17897A (da)
PT (1) PT75850A (da)
SE (1) SE453506B (da)
SG (1) SG34787G (da)
SU (1) SU1378783A3 (da)
YU (1) YU44034B (da)
ZA (1) ZA828387B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1201963B (it) * 1983-03-24 1989-02-02 Prodotti Antibiotici Spa Derivati delle rifamicine e procedimento per la loro preparazione
GB8308166D0 (en) * 1983-03-24 1983-05-05 Erba Farmitalia Preparation of azinomethyl-rifamycins
US4560509A (en) * 1983-11-16 1985-12-24 Eli Lilly And Company Antibiotic A39079 factor S-1
GB8408924D0 (en) * 1984-04-06 1984-05-16 Dobfar Spa 3-azinomethyl rifamycins
US4956373A (en) * 1989-01-31 1990-09-11 Farmitalia Carlo Erba S.R.L Pharmaceutical composition comprising 3-(N-piperidinomethyl-azino) methylrifamycin S as active ingredient
JPH02215716A (ja) * 1989-02-08 1990-08-28 Farmitalia Carlo Erba Spa 3―(n―ピペリジノメチル―アジノ)メチルリファマイシンsを活性成分として含有する薬剤組成物
JP3202960B2 (ja) * 1998-02-17 2001-08-27 大塚化学株式会社 ハロゲン化剤及び水酸基のハロゲン化方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR208F (da) * 1964-07-31
GB1336399A (en) * 1971-06-24 1973-11-07 Lepetit Spa 3-formylrifamycin sv derivatives
BE794298A (fr) * 1972-01-19 1973-05-16 Lepetit Spa Derives d'imidazole de rifamycine et leur preparation
AR205434A1 (es) * 1972-03-27 1976-05-07 Lepetit Spa Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv
CH605974A5 (en) * 1973-09-28 1978-10-13 Ciba Geigy Ag 3-(4-Substd.-1-piperazinyl) rifamycin S and SV derivs
JPS5128640A (da) * 1974-09-03 1976-03-11 Matsushita Electric Ind Co Ltd
GB1478563A (en) * 1975-03-05 1977-07-06 Lepetit Spa Rifamycin derivatives
IT1135270B (it) * 1980-04-12 1986-08-20 Erba Farmitalia 3-amidino-ansamicine

Also Published As

Publication number Publication date
MX157130A (es) 1988-10-28
NO167290C (no) 1991-10-23
FI73436C (fi) 1987-10-09
FI823902L (fi) 1983-05-18
GR76790B (da) 1984-09-04
FI823902A0 (fi) 1982-11-12
BE895020A (fr) 1983-05-16
CH657619A5 (it) 1986-09-15
NO167290B (no) 1991-07-15
NL8204330A (nl) 1983-06-16
FR2516514A1 (fr) 1983-05-20
KR840002401A (ko) 1984-07-02
GB2110677B (en) 1985-02-13
IL67263A0 (en) 1983-03-31
DK157873C (da) 1990-08-06
AT376222B (de) 1984-10-25
DE3241764C2 (da) 1990-05-23
NZ202495A (en) 1985-10-11
HK74687A (en) 1987-10-23
GB2119365A (en) 1983-11-16
NO823812L (no) 1983-05-18
YU44034B (en) 1990-02-28
GB2119365B (en) 1985-02-27
CA1205074A (en) 1986-05-27
IT8224224A0 (it) 1982-11-12
IT1224111B (it) 1990-09-26
PH17897A (en) 1985-01-25
DE3241764A1 (de) 1983-05-26
HU186160B (en) 1985-06-28
ES8401766A1 (es) 1984-01-01
IE54153B1 (en) 1989-07-05
DK507282A (da) 1983-05-18
PT75851A (pt) 1982-12-01
IE822725L (en) 1983-05-17
DK157873B (da) 1990-02-26
SG34787G (en) 1987-07-24
ATA414982A (de) 1984-03-15
GB2110677A (en) 1983-06-22
ZA828387B (en) 1984-06-27
JPH0235758B2 (da) 1990-08-13
US4447432A (en) 1984-05-08
AU9041382A (en) 1983-05-26
IL67263A (en) 1985-12-31
KR880001284B1 (ko) 1988-07-18
YU255482A (en) 1984-12-31
SU1378783A3 (ru) 1988-02-28
AU553727B2 (en) 1986-07-24
JPS5892682A (ja) 1983-06-02
SE453506B (sv) 1988-02-08
PT75850A (fr) 1982-12-01
FI73436B (fi) 1987-06-30
FR2516514B1 (da) 1984-03-23
SE8206499D0 (sv) 1982-11-15
ES517153A0 (es) 1984-01-01
SE8206499L (sv) 1983-05-18

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