CS213305B2 - Method of making the 2-amino or 2-thiosubstituted derivatives of 4,5-diphenyloxazole - Google Patents

Method of making the 2-amino or 2-thiosubstituted derivatives of 4,5-diphenyloxazole Download PDF

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Publication number
CS213305B2
CS213305B2 CS797044A CS704479A CS213305B2 CS 213305 B2 CS213305 B2 CS 213305B2 CS 797044 A CS797044 A CS 797044A CS 704479 A CS704479 A CS 704479A CS 213305 B2 CS213305 B2 CS 213305B2
Authority
CS
Czechoslovakia
Prior art keywords
diphenyl
amino
solution
chloride
aminooxazole
Prior art date
Application number
CS797044A
Other languages
Czech (cs)
English (en)
Inventor
Walter Marconi
Francesco Bartoli
Franco Morisi
Francesco Pittalis
Original Assignee
Eni Ente Naz Idrocarb
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eni Ente Naz Idrocarb filed Critical Eni Ente Naz Idrocarb
Publication of CS213305B2 publication Critical patent/CS213305B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/46—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/48—Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
CS797044A 1978-10-17 1979-10-17 Method of making the 2-amino or 2-thiosubstituted derivatives of 4,5-diphenyloxazole CS213305B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT28825/78A IT1099996B (it) 1978-10-17 1978-10-17 Derivati del 4,5-difenil-ossazolo 2-ammino o 2-tio sostituiti e procedimento per il loro ottenimento

Publications (1)

Publication Number Publication Date
CS213305B2 true CS213305B2 (en) 1982-04-09

Family

ID=11224263

Family Applications (1)

Application Number Title Priority Date Filing Date
CS797044A CS213305B2 (en) 1978-10-17 1979-10-17 Method of making the 2-amino or 2-thiosubstituted derivatives of 4,5-diphenyloxazole

Country Status (22)

Country Link
US (1) US4591596A (xx)
JP (1) JPS5589271A (xx)
AU (1) AU533275B2 (xx)
BE (1) BE879440A (xx)
CA (1) CA1122221A (xx)
CH (1) CH645364A5 (xx)
CS (1) CS213305B2 (xx)
DD (1) DD146598A5 (xx)
DE (1) DE2942050C2 (xx)
DK (1) DK151880C (xx)
FR (1) FR2439191A1 (xx)
GB (1) GB2036006B (xx)
HU (1) HU181426B (xx)
IL (1) IL58458A (xx)
IT (1) IT1099996B (xx)
LU (1) LU81788A1 (xx)
NL (1) NL7907661A (xx)
NO (1) NO793322L (xx)
SE (1) SE446533B (xx)
SU (1) SU982540A3 (xx)
YU (1) YU41184B (xx)
ZA (1) ZA795525B (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1099996B (it) * 1978-10-17 1985-09-28 Anic Spa Derivati del 4,5-difenil-ossazolo 2-ammino o 2-tio sostituiti e procedimento per il loro ottenimento
WO2005039590A1 (en) * 2003-10-21 2005-05-06 Inspire Pharmaceuticals, Inc. Non-nucleotide compositions and method for treating pain
WO2021029826A1 (en) 2019-08-09 2021-02-18 Zuru (Singapore) Pte. Ltd. Gummy confectionery-coated non-edible container
USD1012421S1 (en) 2020-08-07 2024-01-30 Zuru (Singapore) Pte. Ltd. Confectionery

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1538009A (fr) * 1966-08-10 1968-08-30 Serono Ist Farm 4, 5-diphényl-oxazols 2-amino-substitués et les procédés de préparation par synthèse propres à les obtenir
CH506548A (de) * 1966-08-10 1971-04-30 Serono Ist Farm Verfahren zur Herstellung von 2-aminsubstituiertem 4,5-Diphenyl-Oxazol
DE2129012A1 (de) * 1971-06-11 1973-01-04 Merck Patent Gmbh Azol-derivate
DE2428249C3 (de) * 1973-07-09 1978-12-14 Serna Ag, Glarus (Schweiz) Verfahren zur Herstellung von
GB1497536A (en) * 1973-12-17 1978-01-12 Lilly Industries Ltd 2-acylaminooxazoles methods for their preparation and their use
GB1507032A (en) * 1974-08-06 1978-04-12 Serono Lab 2-thiol-4,5-diphenyloxazole s-derivatives
IT1085524B (it) * 1977-03-22 1985-05-28 Snam Progetti Materiali e fibre porose biocompatibili in grado di inglobare sostanze di interesse biologico e metodi per il loro ottenimento
IT1099996B (it) * 1978-10-17 1985-09-28 Anic Spa Derivati del 4,5-difenil-ossazolo 2-ammino o 2-tio sostituiti e procedimento per il loro ottenimento

Also Published As

Publication number Publication date
AU5171279A (en) 1980-04-24
SU982540A3 (ru) 1982-12-15
HU181426B (en) 1983-07-28
ZA795525B (en) 1980-10-29
CA1122221A (en) 1982-04-20
US4591596A (en) 1986-05-27
JPS5589271A (en) 1980-07-05
SE446533B (sv) 1986-09-22
DK151880B (da) 1988-01-11
GB2036006A (en) 1980-06-25
LU81788A1 (fr) 1980-01-24
GB2036006B (en) 1983-01-06
IL58458A0 (en) 1980-01-31
NL7907661A (nl) 1980-04-21
FR2439191A1 (fr) 1980-05-16
AU533275B2 (en) 1983-11-17
IT7828825A0 (it) 1978-10-17
YU41184B (en) 1986-12-31
BE879440A (fr) 1980-04-16
FR2439191B1 (xx) 1982-06-18
IT1099996B (it) 1985-09-28
SE7908532L (sv) 1980-04-18
DE2942050C2 (de) 1986-12-04
DK151880C (da) 1988-06-06
IL58458A (en) 1983-06-15
DE2942050A1 (de) 1980-04-24
CH645364A5 (it) 1984-09-28
DK436879A (da) 1980-04-18
YU250379A (en) 1983-04-30
NO793322L (no) 1980-04-18
JPH0231072B2 (xx) 1990-07-11
DD146598A5 (de) 1981-02-18

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