CS207671B2 - Method of making the piperazinylchinazoline derivatives - Google Patents

Method of making the piperazinylchinazoline derivatives Download PDF

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Publication number
CS207671B2
CS207671B2 CS787166A CS716678A CS207671B2 CS 207671 B2 CS207671 B2 CS 207671B2 CS 787166 A CS787166 A CS 787166A CS 716678 A CS716678 A CS 716678A CS 207671 B2 CS207671 B2 CS 207671B2
Authority
CS
Czechoslovakia
Prior art keywords
carbon atoms
formula
group
different
alkoxy
Prior art date
Application number
CS787166A
Other languages
Czech (cs)
English (en)
Inventor
Simon F Campbell
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Priority to CS801183A priority Critical patent/CS207672B2/cs
Publication of CS207671B2 publication Critical patent/CS207671B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/20—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CS787166A 1977-11-05 1978-11-02 Method of making the piperazinylchinazoline derivatives CS207671B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS801183A CS207672B2 (cs) 1977-11-05 1980-02-20 Způsob výroby piperazinylchinazolinových derivátů

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4612877 1977-11-05

Publications (1)

Publication Number Publication Date
CS207671B2 true CS207671B2 (en) 1981-08-31

Family

ID=10439957

Family Applications (2)

Application Number Title Priority Date Filing Date
CS787166A CS207671B2 (en) 1977-11-05 1978-11-02 Method of making the piperazinylchinazoline derivatives
CS913544A CS354491A3 (en) 1977-11-05 1991-11-22 4-amino-2-/piperazin-1-yl/ or /homopiperazin-1-yl/quinazoline derivatives, process of their preparation and use

Family Applications After (1)

Application Number Title Priority Date Filing Date
CS913544A CS354491A3 (en) 1977-11-05 1991-11-22 4-amino-2-/piperazin-1-yl/ or /homopiperazin-1-yl/quinazoline derivatives, process of their preparation and use

Country Status (36)

Country Link
JP (1) JPS5498792A (enrdf_load_stackoverflow)
AR (2) AR219562A1 (enrdf_load_stackoverflow)
AT (1) AT365186B (enrdf_load_stackoverflow)
AU (1) AU509329B2 (enrdf_load_stackoverflow)
BE (1) BE871771A (enrdf_load_stackoverflow)
CA (1) CA1088059A (enrdf_load_stackoverflow)
CH (1) CH643255A5 (enrdf_load_stackoverflow)
CS (2) CS207671B2 (enrdf_load_stackoverflow)
DD (1) DD139850A5 (enrdf_load_stackoverflow)
DE (1) DE2847623C2 (enrdf_load_stackoverflow)
DK (1) DK154082C (enrdf_load_stackoverflow)
EG (1) EG13594A (enrdf_load_stackoverflow)
ES (2) ES474805A1 (enrdf_load_stackoverflow)
FI (1) FI64366C (enrdf_load_stackoverflow)
FR (1) FR2407929A1 (enrdf_load_stackoverflow)
GR (1) GR81514B (enrdf_load_stackoverflow)
HK (1) HK94284A (enrdf_load_stackoverflow)
HU (1) HU176306B (enrdf_load_stackoverflow)
IE (1) IE47888B1 (enrdf_load_stackoverflow)
IL (1) IL55857A (enrdf_load_stackoverflow)
IN (1) IN148828B (enrdf_load_stackoverflow)
IT (1) IT1100919B (enrdf_load_stackoverflow)
KE (1) KE3350A (enrdf_load_stackoverflow)
LU (2) LU80470A1 (enrdf_load_stackoverflow)
MY (1) MY8500286A (enrdf_load_stackoverflow)
NL (2) NL174549C (enrdf_load_stackoverflow)
NO (1) NO150158C (enrdf_load_stackoverflow)
NZ (1) NZ188813A (enrdf_load_stackoverflow)
PH (1) PH13966A (enrdf_load_stackoverflow)
PL (2) PL119419B1 (enrdf_load_stackoverflow)
PT (1) PT68735A (enrdf_load_stackoverflow)
SE (1) SE437518B (enrdf_load_stackoverflow)
SU (1) SU816403A3 (enrdf_load_stackoverflow)
UA (1) UA8324A1 (enrdf_load_stackoverflow)
YU (2) YU40204B (enrdf_load_stackoverflow)
ZA (1) ZA786184B (enrdf_load_stackoverflow)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985002617A1 (en) * 1983-12-14 1985-06-20 Takeda Chemical Industries. Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1985004658A1 (en) * 1984-04-04 1985-10-24 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepine derivatives and their preparation
WO1986002644A1 (en) * 1984-11-01 1986-05-09 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
EP0849265A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von Doxazosin-Mesylat (Form II)
EP0849264A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von doxazosinmesylat (Form I)
EP0849266B8 (de) * 1996-12-20 2007-10-03 Heumann PCS GmbH Neue polymorphe Form von Doxazosinmesylat (Form III)
TW448155B (en) * 1999-03-29 2001-08-01 Dev Center Biotechnology Method for producing amide compounds and quinazolin derivatives
EP1403263B1 (en) * 2002-09-27 2005-06-22 Council of Scientific and Industrial Research Process for the preparation of N-(2,3-dihydrobenzo 1,4 dioxin-2-carbonyl) piperazine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3635979A (en) * 1969-09-29 1972-01-18 Pfizer Certain 6- and/or 7-alkoxy-substituted-2 4-bis(disubstituted amino) quinazolines
US3669968A (en) * 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines

Also Published As

Publication number Publication date
SE7811382L (sv) 1979-05-06
JPS5498792A (en) 1979-08-03
IL55857A0 (en) 1979-01-31
BE871771A (fr) 1979-05-03
LU88331I2 (fr) 1994-05-04
NL930062I2 (nl) 1993-11-16
DK154082B (da) 1988-10-10
IL55857A (en) 1982-07-30
NZ188813A (en) 1980-10-08
HU176306B (en) 1981-01-28
AU509329B2 (en) 1980-05-08
PT68735A (en) 1978-12-01
PL119419B1 (en) 1981-12-31
DD139850A5 (de) 1980-01-23
JPS5625233B2 (enrdf_load_stackoverflow) 1981-06-11
PL210681A1 (enrdf_load_stackoverflow) 1979-11-05
AT365186B (de) 1981-12-28
IN148828B (enrdf_load_stackoverflow) 1981-06-27
KE3350A (en) 1983-12-16
EG13594A (en) 1982-03-31
FI783347A7 (fi) 1979-05-06
DK428678A (da) 1979-05-06
IE782179L (en) 1979-05-05
ES480121A0 (es) 1980-07-16
ATA784378A (de) 1981-05-15
YU255378A (en) 1983-06-30
IT1100919B (it) 1985-09-28
CS354491A3 (en) 1992-06-17
PH13966A (en) 1980-11-12
SE437518B (sv) 1985-03-04
NL174549B (nl) 1984-02-01
DK154082C (da) 1989-02-27
DE2847623C2 (de) 1983-06-01
AU4132278A (en) 1979-05-17
AR223015A1 (es) 1981-07-15
FR2407929B1 (enrdf_load_stackoverflow) 1981-02-27
ES474805A1 (es) 1980-01-16
YU38683A (en) 1983-06-30
CA1088059A (en) 1980-10-21
UA8324A1 (uk) 1996-03-29
AR219562A1 (es) 1980-08-29
MY8500286A (en) 1985-12-31
NO150158C (no) 1984-08-29
NO150158B (no) 1984-05-21
NO783705L (no) 1979-05-08
IE47888B1 (en) 1984-07-11
SU816403A3 (ru) 1981-03-23
YU40204B (en) 1985-08-31
CH643255A5 (en) 1984-05-30
FR2407929A1 (fr) 1979-06-01
DE2847623A1 (de) 1979-05-23
HK94284A (en) 1984-12-07
NL930062I1 (nl) 1993-09-01
FI64366C (fi) 1983-11-10
PL119586B1 (en) 1982-01-30
NL7810909A (nl) 1979-05-08
ES8308559A1 (es) 1980-07-16
LU80470A1 (fr) 1980-06-05
GR81514B (enrdf_load_stackoverflow) 1984-12-11
FI64366B (fi) 1983-07-29
ZA786184B (en) 1979-10-31
YU40419B (en) 1985-12-31
IT7829434A0 (it) 1978-11-03
NL174549C (nl) 1984-07-02

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