CO4480098A1 - Formulaciones de danofloxacina inyectable que comprenden un compuesto de cinc con un disolvente complementario . - Google Patents

Formulaciones de danofloxacina inyectable que comprenden un compuesto de cinc con un disolvente complementario .

Info

Publication number
CO4480098A1
CO4480098A1 CO96066993A CO96066993A CO4480098A1 CO 4480098 A1 CO4480098 A1 CO 4480098A1 CO 96066993 A CO96066993 A CO 96066993A CO 96066993 A CO96066993 A CO 96066993A CO 4480098 A1 CO4480098 A1 CO 4480098A1
Authority
CO
Colombia
Prior art keywords
conforming
complementary solvent
danofloxacin
complementary
solvent
Prior art date
Application number
CO96066993A
Other languages
English (en)
Inventor
Wayne Alan Boettner
Peter Connor Canning
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21735307&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO4480098(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of CO4480098A1 publication Critical patent/CO4480098A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4995Pyrazines or piperazines forming part of bridged ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Organic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

SOLUCIONES FARMACEUTICAS ACUOSAS ADECUADAS PARA INYECCION EN UN HUESPED, QUE TIENEN MEJORADA LA TOLERANCIA EN EL SITIO DE LA INYECCION, COMPRENDEN DANOFLOXACINA O SUS SALES FARMACEUTICAMENTE ACEP- TABLES Y UN COMPUESTO DE MAGNESIO O DE CINC. EL COMPUESTO DE CINC REQUIERE ADEMAS LA PRESENCIA DE UN DISOLVENTE COMPLEMENTARIO. ADECUADA EN UN HUESPED, QUE COMPRENDE DANOFLOXACI- NA O UNA DE SUS SALES FARMACEUTICAMENTE ACEPTABLES EN UNA CANTIDAD SUFICIENTE PARA EL TRATAMIENTO DE INFECCIONES BACTERIANAS Y, (1) UN COMPUESTO DE MAGNESIO O, (2) UN COMPUESTO DE CINC MEZCLADO CON UN DISOLVENTE COMPLEMENTARIO, ESTANDO PRESENTES DICHOS COMPUESTOS Y DICHO DISOLVENTE COMPLEMENTA- RIO EN CANTIDADES QUE SON SUFICIENTES PARA MEJORAR LA TOLERANCIA EN EL SITIO DE LA INYECCION. UNA CONFORME A LA REIVINDICACION 1, EN LA QUE DI- CHO COMPUESTO DE MAGNESIO ESTA PRESENTE JUNTO CON UN DISOLVENTE COMPLEMENTARIO. UNA CONFORME A LA REIVINDICACION 1 O 2, EN LA QUE DICHO DISOLVENTE COMPLEMENTARIO ES AL MENOS UNO DE 2-PIRROLIDONA, PROPILENGLICOL, POLIETILENGLICOL Y N-METIL PIRROLIDONA, CADA UNO DE ELLOS OPCIONAL- MENTE JUNTO CON POLIVINILPIRROLIDONA. UNA CONFORME A UNA CUALQUIERA DE LAS REIVINDICA- CIONES 1, 2 O 3, EN LA QUE DICHA SOLUCION CONTIENE ADEMAS UN ANTIOXIDANTE. UNA CONFORME A LA REIVINDICACION 4, EN LA QUE DI- CHO ANTIOXIDANTE ES FORMALDEHIDO SULFOXILATO SODI- CO.
CO96066993A 1995-12-21 1996-12-20 Formulaciones de danofloxacina inyectable que comprenden un compuesto de cinc con un disolvente complementario . CO4480098A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US905295P 1995-12-21 1995-12-21

Publications (1)

Publication Number Publication Date
CO4480098A1 true CO4480098A1 (es) 1997-07-09

Family

ID=21735307

Family Applications (1)

Application Number Title Priority Date Filing Date
CO96066993A CO4480098A1 (es) 1995-12-21 1996-12-20 Formulaciones de danofloxacina inyectable que comprenden un compuesto de cinc con un disolvente complementario .

Country Status (42)

Country Link
US (1) US5811130A (es)
EP (1) EP0868183B1 (es)
JP (1) JP3416145B2 (es)
KR (1) KR100402570B1 (es)
CN (1) CN1104899C (es)
AP (1) AP706A (es)
AR (1) AR005147A1 (es)
AT (1) ATE212551T1 (es)
AU (1) AU709474B2 (es)
BG (1) BG63933B1 (es)
BR (1) BR9612230A (es)
CA (1) CA2239352C (es)
CO (1) CO4480098A1 (es)
CZ (1) CZ293747B6 (es)
DE (1) DE69618987T2 (es)
DK (1) DK0868183T3 (es)
DZ (1) DZ2146A1 (es)
EG (1) EG24071A (es)
ES (1) ES2167609T3 (es)
GT (1) GT199600098A (es)
HR (1) HRP960607B1 (es)
HU (1) HU227918B1 (es)
IL (1) IL124454A (es)
IS (1) IS2010B (es)
MA (1) MA24035A1 (es)
MX (1) MX9805026A (es)
MY (1) MY117109A (es)
NO (1) NO315734B1 (es)
NZ (2) NZ501160A (es)
OA (1) OA10697A (es)
PE (1) PE25798A1 (es)
PL (1) PL186795B1 (es)
PT (1) PT868183E (es)
RS (1) RS49523B (es)
RU (1) RU2141827C1 (es)
SI (1) SI0868183T1 (es)
SK (1) SK284412B6 (es)
TN (1) TNSN96163A1 (es)
TW (1) TW449475B (es)
UA (1) UA56151C2 (es)
WO (1) WO1997023217A1 (es)
ZA (1) ZA9610780B (es)

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ID21415A (id) * 1997-12-05 1999-06-10 Upjohn Co Senyawa-senyawa antibiotik magnesium quinolon
US6017948A (en) * 1998-10-30 2000-01-25 Supergen, Inc. Water-miscible pharmaceutical compositions
DE19937115A1 (de) 1999-08-06 2001-02-08 Bayer Ag Wäßrige Arzneimittelformulierung von Moxifloxacin oder Salzen davon
DE19937116A1 (de) * 1999-08-06 2001-02-08 Bayer Ag Moxifloxacin Kochsalzformulierung
WO2001051089A1 (de) * 2000-01-13 2001-07-19 Merck Patent Gmbh Pharmazeutische zubereitungen enthaltend 2-pyrrolidon als lösungsvermittler
CA2433037C (en) * 2000-12-28 2010-12-21 Takeda Chemical Industries, Ltd. Sustained-release preparation
AU2003247793A1 (en) * 2002-06-26 2004-01-19 Pharmacia Corporation Stable liquid parenteral parecoxib formulation
KR20070029280A (ko) * 2004-07-02 2007-03-13 다이이찌 세이야꾸 가부시기가이샤 퀴놀론 함유 의약 조성물
WO2006125132A2 (en) * 2005-05-18 2006-11-23 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
US8524735B2 (en) 2005-05-18 2013-09-03 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
FR2896416B1 (fr) 2006-01-24 2010-08-13 Vetoquinol Composition anti-infectieuse comprenant un compose de type pyrido (3,2,1-ij)-benzoxadiazine
HUE037773T2 (hu) * 2006-02-10 2018-09-28 Pari Pharma Gmbh Porlasztott antibiotikumok inhalációs terápiához
US20070197548A1 (en) 2006-02-17 2007-08-23 Murthy Yerramilli V S Fluoroquinolone compositions
DE102006010642A1 (de) * 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
DE102006010643A1 (de) 2006-03-08 2007-09-13 Bayer Healthcare Aktiengesellschaft Arzneimittel enthaltend Fluorchinolone
MX2007009796A (es) 2007-08-14 2009-02-25 Cell Therapy And Technology S Gel conteniendo pirfenidona.
KR20110091510A (ko) 2008-10-07 2011-08-11 엠펙스 파마슈티컬즈, 인코포레이티드 약동학 개선을 위한 에어로졸 플루오로퀴놀론 제형
CN102325532B (zh) 2008-10-07 2015-06-17 Mpex医药有限公司 用于减轻肺部炎症的左氧氟沙星吸入剂
ES2739979T3 (es) 2009-09-04 2020-02-05 Horizon Orphan Llc Uso de levofloxacino en aerosol para el tratamiento de la fibrosis quística
MX2011007675A (es) 2011-07-19 2012-07-11 Cell Therapy And Technology S A De C V Procedimiento para la fabricacion de una composicion farmaceutica en forma de tabletas de liberacion prolongada conteniendo pirfenidona y su aplicacion en la regresion de la insuficiencia renal cronica, contractura capsular mamaria y fibrosis hepatica humanas.
MX346763B (es) 2012-03-28 2017-03-31 Cell Therapy And Tech S A De C V Composición tópica semisólida conteniendo pirfenidona y dialil óxido de disulfuro modificado (odd-m) para eliminar o prevenir el acné.
MX356551B (es) 2012-08-23 2018-06-04 Grupo Medifarma S A De C V Star Composición antiséptica, antiseborreica y exfoliante para eliminar o prevenir el acné.
EP3305294A4 (en) 2015-06-02 2019-02-20 Kyorin Pharmaceutical Co., Ltd. AQUEOUS MEDICINE
US10406149B2 (en) 2015-06-02 2019-09-10 Kyorin Pharmaceutical Co., Ltd. Aqueous liquid formulation
US10206917B2 (en) 2015-06-02 2019-02-19 Kyorin Pharmaceutical Co., Ltd. Aqueous drug
ES2886088T3 (es) * 2017-02-13 2021-12-16 Bayer Animal Health Gmbh Composición líquida que contiene pradofloxacina
MX366086B (es) 2017-08-15 2019-06-27 Cell Therapy And Tech S A De C V Composicion topica semisolida conteniendo un agente antimicrobiano y pirfenidona para el tratamiento de daños cronicos de la piel.

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US523505A (en) * 1894-07-24 Island
DE3517709A1 (de) * 1985-01-05 1986-07-10 Bayer Ag Basische zubereitungen von chinoloncarbonsaeuren
JPS63188626A (ja) * 1987-01-30 1988-08-04 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸の可溶化方法
DE3902079A1 (de) * 1988-04-15 1989-10-26 Bayer Ag I.m. injektionsformen von gyrase-inhibitoren
ATE150973T1 (de) * 1989-12-29 1997-04-15 Abbott Lab Chinoloncarbonsäure-metallionsäurekomplexe
US5084276A (en) * 1990-01-05 1992-01-28 Abbott Laboratories Quinolone carboxylic acid compositions with polymeric additive to reduce vein irritation
EP0443381B2 (en) * 1990-02-14 1997-10-22 Takeda Chemical Industries, Ltd. Effervescent composition, its production and use
FR2665635A1 (fr) * 1990-08-10 1992-02-14 Merck Sharp & Dohme Composition pharmaceutique fluide a base d'un complexe metallique et son procede de preparation.
US5082863A (en) * 1990-08-29 1992-01-21 Schering Corporation Pharmaceutical composition of florfenicol
US5235054A (en) * 1992-07-15 1993-08-10 Pfizer Inc. 3-carboxaldehyde substituted quinolines and naphthyridines
JPH0782141A (ja) * 1993-09-17 1995-03-28 Tanabe Seiyaku Co Ltd 動物用注射剤

Also Published As

Publication number Publication date
ZA9610780B (en) 1998-06-22
HUP9903726A2 (hu) 2000-04-28
JPH11501331A (ja) 1999-02-02
DE69618987D1 (de) 2002-03-14
AU7328996A (en) 1997-07-17
NO982842L (no) 1998-06-19
HU227918B1 (en) 2012-06-28
CZ293747B6 (cs) 2004-07-14
AR005147A1 (es) 1999-04-14
BG102542A (en) 1999-06-30
WO1997023217A1 (en) 1997-07-03
US5811130A (en) 1998-09-22
PE25798A1 (es) 1998-05-21
IS4755A (is) 1998-05-25
EP0868183A1 (en) 1998-10-07
YU69096A (sh) 1999-06-15
HRP960607A2 (en) 1998-06-30
HRP960607B1 (en) 2002-06-30
IL124454A0 (en) 1998-12-06
PT868183E (pt) 2002-06-28
EG24071A (en) 2008-05-11
SK80798A3 (en) 1999-09-10
CN1205636A (zh) 1999-01-20
TW449475B (en) 2001-08-11
ES2167609T3 (es) 2002-05-16
NZ320545A (en) 2000-03-27
MX9805026A (es) 1998-09-30
HUP9903726A3 (en) 2001-01-29
NZ501160A (en) 2001-10-26
KR19990076617A (ko) 1999-10-15
CA2239352C (en) 2002-06-04
IS2010B (is) 2005-05-13
MA24035A1 (fr) 1997-07-01
NO315734B1 (no) 2003-10-20
DE69618987T2 (de) 2002-11-21
PL186795B1 (pl) 2004-02-27
DK0868183T3 (da) 2002-03-25
RS49523B (sr) 2006-10-27
PL328001A1 (en) 1999-01-04
CZ193098A3 (cs) 1999-05-12
BG63933B1 (bg) 2003-07-31
NO982842D0 (no) 1998-06-19
MY117109A (en) 2004-05-31
KR100402570B1 (ko) 2003-12-18
BR9612230A (pt) 1999-07-13
EP0868183B1 (en) 2002-01-30
RU2141827C1 (ru) 1999-11-27
ATE212551T1 (de) 2002-02-15
SI0868183T1 (en) 2002-04-30
OA10697A (en) 2001-05-04
DZ2146A1 (fr) 2002-10-23
AP9600898A0 (en) 1997-01-31
AP706A (en) 1998-12-04
AU709474B2 (en) 1999-08-26
CA2239352A1 (en) 1997-07-03
TNSN96163A1 (fr) 2005-03-15
IL124454A (en) 2003-10-31
SK284412B6 (sk) 2005-03-04
GT199600098A (es) 1998-06-12
JP3416145B2 (ja) 2003-06-16
UA56151C2 (uk) 2003-05-15
CN1104899C (zh) 2003-04-09

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