TNSN96163A1 - Formulations injectables de quinolones - Google Patents

Formulations injectables de quinolones

Info

Publication number
TNSN96163A1
TNSN96163A1 TNTNSN96163A TNSN96163A TNSN96163A1 TN SN96163 A1 TNSN96163 A1 TN SN96163A1 TN TNSN96163 A TNTNSN96163 A TN TNSN96163A TN SN96163 A TNSN96163 A TN SN96163A TN SN96163 A1 TNSN96163 A1 TN SN96163A1
Authority
TN
Tunisia
Prior art keywords
quinolones
injectable formulations
injection
danofloxacin
magnesium
Prior art date
Application number
TNTNSN96163A
Other languages
English (en)
Inventor
Alan Boettner Wayne
Connor Canning Pter
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21735307&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TNSN96163(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of TNSN96163A1 publication Critical patent/TNSN96163A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4995Pyrazines or piperazines forming part of bridged ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Abstract

L'INVENTION CONCERNE DES SOLUTIONS PHARMACEUTIQUES ACQUEUSES APTES A L'INJECTION. CES SOLUTIONS COMPRENNENT DE LA DANOFLOXACINE OU UN DE SES SELS PHARMACEUTIQUEMENT ACCEPTABLES ET UN COMPOSE DE MAGNESIUM OU DE ZINC EN PRESENCE D'UN CO-SOLVANT. APPLICATION : TRAITEMENT D'INFECTIONS BACTERIENNES PAR INJECTION SOUS-CUTANEE, AVEC UNE TOLERANCE AMELIOREE AU SITE D'INJECTION.
TNTNSN96163A 1995-12-21 1996-12-18 Formulations injectables de quinolones TNSN96163A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US905295P 1995-12-21 1995-12-21

Publications (1)

Publication Number Publication Date
TNSN96163A1 true TNSN96163A1 (fr) 2005-03-15

Family

ID=21735307

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN96163A TNSN96163A1 (fr) 1995-12-21 1996-12-18 Formulations injectables de quinolones

Country Status (42)

Country Link
US (1) US5811130A (fr)
EP (1) EP0868183B1 (fr)
JP (1) JP3416145B2 (fr)
KR (1) KR100402570B1 (fr)
CN (1) CN1104899C (fr)
AP (1) AP706A (fr)
AR (1) AR005147A1 (fr)
AT (1) ATE212551T1 (fr)
AU (1) AU709474B2 (fr)
BG (1) BG63933B1 (fr)
BR (1) BR9612230A (fr)
CA (1) CA2239352C (fr)
CO (1) CO4480098A1 (fr)
CZ (1) CZ293747B6 (fr)
DE (1) DE69618987T2 (fr)
DK (1) DK0868183T3 (fr)
DZ (1) DZ2146A1 (fr)
EG (1) EG24071A (fr)
ES (1) ES2167609T3 (fr)
GT (1) GT199600098A (fr)
HR (1) HRP960607B1 (fr)
HU (1) HU227918B1 (fr)
IL (1) IL124454A (fr)
IS (1) IS2010B (fr)
MA (1) MA24035A1 (fr)
MX (1) MX9805026A (fr)
MY (1) MY117109A (fr)
NO (1) NO315734B1 (fr)
NZ (2) NZ501160A (fr)
OA (1) OA10697A (fr)
PE (1) PE25798A1 (fr)
PL (1) PL186795B1 (fr)
PT (1) PT868183E (fr)
RS (1) RS49523B (fr)
RU (1) RU2141827C1 (fr)
SI (1) SI0868183T1 (fr)
SK (1) SK284412B6 (fr)
TN (1) TNSN96163A1 (fr)
TW (1) TW449475B (fr)
UA (1) UA56151C2 (fr)
WO (1) WO1997023217A1 (fr)
ZA (1) ZA9610780B (fr)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ID21415A (id) * 1997-12-05 1999-06-10 Upjohn Co Senyawa-senyawa antibiotik magnesium quinolon
US6017948A (en) * 1998-10-30 2000-01-25 Supergen, Inc. Water-miscible pharmaceutical compositions
DE19937116A1 (de) * 1999-08-06 2001-02-08 Bayer Ag Moxifloxacin Kochsalzformulierung
DE19937115A1 (de) 1999-08-06 2001-02-08 Bayer Ag Wäßrige Arzneimittelformulierung von Moxifloxacin oder Salzen davon
EP1255565A1 (fr) * 2000-01-13 2002-11-13 MERCK PATENT GmbH Compositions pharmaceutiques contenant de la 2-pyrrolidone en tant qu'agent de solubilisation
EP1356809A4 (fr) * 2000-12-28 2008-05-14 Takeda Pharmaceutical Preparations a liberation soutenue
EP1524997A1 (fr) * 2002-06-26 2005-04-27 Pharmacia Corporation Formulation de parecoxib liquide stable administree par voie parenterale
CA2572167A1 (fr) * 2004-07-02 2006-01-12 Daiichi Pharmaceutical Co., Ltd. Composition medicinale contenant de la quinolone
DK1901749T3 (en) * 2005-05-18 2016-10-24 Raptor Pharmaceuticals Inc Aerosolized fluoroquinolones AND USES THEREOF
US8524734B2 (en) 2005-05-18 2013-09-03 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
FR2896416B1 (fr) 2006-01-24 2010-08-13 Vetoquinol Composition anti-infectieuse comprenant un compose de type pyrido (3,2,1-ij)-benzoxadiazine
MX2008010222A (es) * 2006-02-10 2008-10-17 Pari Pharma Gmbh Antibioticos nebulizados para terapia de inhalacion.
US20070197548A1 (en) 2006-02-17 2007-08-23 Murthy Yerramilli V S Fluoroquinolone compositions
DE102006010642A1 (de) * 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
DE102006010643A1 (de) * 2006-03-08 2007-09-13 Bayer Healthcare Aktiengesellschaft Arzneimittel enthaltend Fluorchinolone
MX2007009796A (es) 2007-08-14 2009-02-25 Cell Therapy And Technology S Gel conteniendo pirfenidona.
KR20110091510A (ko) 2008-10-07 2011-08-11 엠펙스 파마슈티컬즈, 인코포레이티드 약동학 개선을 위한 에어로졸 플루오로퀴놀론 제형
CA2739893C (fr) 2008-10-07 2016-10-04 Mpex Pharmaceuticals, Inc. Inhalation de levofloxacine pour reduire une inflammation des poumons
RU2015130524A (ru) 2009-09-04 2018-12-21 Раптор Фармасьютикалз Инк. Применение левофлоксацина в форме аэрозоля для лечения муковисцидоза
MX2011007675A (es) 2011-07-19 2012-07-11 Cell Therapy And Technology S A De C V Procedimiento para la fabricacion de una composicion farmaceutica en forma de tabletas de liberacion prolongada conteniendo pirfenidona y su aplicacion en la regresion de la insuficiencia renal cronica, contractura capsular mamaria y fibrosis hepatica humanas.
MX346763B (es) 2012-03-28 2017-03-31 Cell Therapy And Tech S A De C V Composición tópica semisólida conteniendo pirfenidona y dialil óxido de disulfuro modificado (odd-m) para eliminar o prevenir el acné.
MX356551B (es) 2012-08-23 2018-06-04 Grupo Medifarma S A De C V Star Composición antiséptica, antiseborreica y exfoliante para eliminar o prevenir el acné.
CA2987879A1 (fr) 2015-06-02 2016-12-08 Kyorin Pharmaceutical Co., Ltd. Medicament aqueux
WO2016195020A1 (fr) 2015-06-02 2016-12-08 杏林製薬株式会社 Médicament aqueux
CA2988092A1 (fr) 2015-06-02 2016-12-08 Kyorin Pharmaceutical Co., Ltd. Formulation liquide aqueuse
WO2018146194A1 (fr) * 2017-02-13 2018-08-16 Bayer Animal Health Gmbh Composition liquide contenant de la pradofloxacine
MX366086B (es) 2017-08-15 2019-06-27 Cell Therapy And Tech S A De C V Composicion topica semisolida conteniendo un agente antimicrobiano y pirfenidona para el tratamiento de daños cronicos de la piel.

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3517709A1 (de) * 1985-01-05 1986-07-10 Bayer Ag Basische zubereitungen von chinoloncarbonsaeuren
JPS63188626A (ja) * 1987-01-30 1988-08-04 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸の可溶化方法
DE3902079A1 (de) * 1988-04-15 1989-10-26 Bayer Ag I.m. injektionsformen von gyrase-inhibitoren
CA2072366C (fr) * 1989-12-29 2002-08-20 Laman A. Al-Razzak Complexes d'acide carboxylique d'une quinolone-ion d'un metal-acide
US5084276A (en) * 1990-01-05 1992-01-28 Abbott Laboratories Quinolone carboxylic acid compositions with polymeric additive to reduce vein irritation
DE69102900T3 (de) * 1990-02-14 1998-04-09 Takeda Chemical Industries Ltd Brausemischung, deren Herstellung sowie Verwendung.
FR2665635A1 (fr) * 1990-08-10 1992-02-14 Merck Sharp & Dohme Composition pharmaceutique fluide a base d'un complexe metallique et son procede de preparation.
US5082863A (en) * 1990-08-29 1992-01-21 Schering Corporation Pharmaceutical composition of florfenicol
US5235054A (en) * 1992-07-15 1993-08-10 Pfizer Inc. 3-carboxaldehyde substituted quinolines and naphthyridines
JPH0782141A (ja) * 1993-09-17 1995-03-28 Tanabe Seiyaku Co Ltd 動物用注射剤

Also Published As

Publication number Publication date
HUP9903726A3 (en) 2001-01-29
KR19990076617A (ko) 1999-10-15
ES2167609T3 (es) 2002-05-16
IS2010B (is) 2005-05-13
PE25798A1 (es) 1998-05-21
JP3416145B2 (ja) 2003-06-16
DZ2146A1 (fr) 2002-10-23
HU227918B1 (en) 2012-06-28
CO4480098A1 (es) 1997-07-09
DE69618987T2 (de) 2002-11-21
AP706A (en) 1998-12-04
AU709474B2 (en) 1999-08-26
NO315734B1 (no) 2003-10-20
SK284412B6 (sk) 2005-03-04
NO982842L (no) 1998-06-19
MX9805026A (es) 1998-09-30
CZ193098A3 (cs) 1999-05-12
JPH11501331A (ja) 1999-02-02
BG102542A (en) 1999-06-30
NZ320545A (en) 2000-03-27
KR100402570B1 (ko) 2003-12-18
ATE212551T1 (de) 2002-02-15
PL328001A1 (en) 1999-01-04
TW449475B (en) 2001-08-11
CZ293747B6 (cs) 2004-07-14
BG63933B1 (bg) 2003-07-31
EG24071A (en) 2008-05-11
CA2239352A1 (fr) 1997-07-03
IL124454A0 (en) 1998-12-06
CN1104899C (zh) 2003-04-09
HUP9903726A2 (hu) 2000-04-28
OA10697A (en) 2001-05-04
IL124454A (en) 2003-10-31
CA2239352C (fr) 2002-06-04
HRP960607B1 (en) 2002-06-30
YU69096A (sh) 1999-06-15
DE69618987D1 (de) 2002-03-14
UA56151C2 (uk) 2003-05-15
SK80798A3 (en) 1999-09-10
BR9612230A (pt) 1999-07-13
EP0868183A1 (fr) 1998-10-07
RS49523B (sr) 2006-10-27
US5811130A (en) 1998-09-22
HRP960607A2 (en) 1998-06-30
WO1997023217A1 (fr) 1997-07-03
NZ501160A (en) 2001-10-26
SI0868183T1 (en) 2002-04-30
MY117109A (en) 2004-05-31
NO982842D0 (no) 1998-06-19
AU7328996A (en) 1997-07-17
GT199600098A (es) 1998-06-12
IS4755A (is) 1998-05-25
DK0868183T3 (da) 2002-03-25
ZA9610780B (en) 1998-06-22
PL186795B1 (pl) 2004-02-27
AR005147A1 (es) 1999-04-14
CN1205636A (zh) 1999-01-20
RU2141827C1 (ru) 1999-11-27
AP9600898A0 (en) 1997-01-31
PT868183E (pt) 2002-06-28
EP0868183B1 (fr) 2002-01-30
MA24035A1 (fr) 1997-07-01

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