CN1742007A - 甾族激素核受体的吲哚衍生物调控剂 - Google Patents
甾族激素核受体的吲哚衍生物调控剂 Download PDFInfo
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- CN1742007A CN1742007A CNA2004800026858A CN200480002685A CN1742007A CN 1742007 A CN1742007 A CN 1742007A CN A2004800026858 A CNA2004800026858 A CN A2004800026858A CN 200480002685 A CN200480002685 A CN 200480002685A CN 1742007 A CN1742007 A CN 1742007A
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- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US44194703P | 2003-01-22 | 2003-01-22 | |
| US60/441,947 | 2003-01-22 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1742007A true CN1742007A (zh) | 2006-03-01 |
Family
ID=32825176
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA2004800026858A Pending CN1742007A (zh) | 2003-01-22 | 2004-01-20 | 甾族激素核受体的吲哚衍生物调控剂 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20060235222A1 (enExample) |
| EP (1) | EP1597254A1 (enExample) |
| JP (1) | JP2007500253A (enExample) |
| CN (1) | CN1742007A (enExample) |
| AU (1) | AU2004207740A1 (enExample) |
| BR (1) | BRPI0406883A (enExample) |
| CA (1) | CA2511806A1 (enExample) |
| MX (1) | MXPA05007857A (enExample) |
| WO (1) | WO2004067529A1 (enExample) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI582080B (zh) * | 2012-07-19 | 2017-05-11 | 默沙東藥廠 | 礦皮質素受體拮抗劑 |
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| DE102004021637A1 (de) * | 2004-05-03 | 2005-12-01 | Merck Patent Gmbh | Dihydrobenzothiophene |
| EP1632491A1 (en) * | 2004-08-30 | 2006-03-08 | Laboratorios Del Dr. Esteve, S.A. | Substituted indole compounds and their use as 5-HT6 receptor modulators |
| WO2006101454A1 (en) * | 2005-03-21 | 2006-09-28 | S*Bio Pte Ltd | Benzothiophene derivatives: preparation and pharmaceutical applications |
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| GEP20115239B (en) | 2006-10-31 | 2011-06-10 | Pfizer Prod Inc | Pyrazoline compounds as mineralocorticoid receptor antagonists |
| JP2010138072A (ja) * | 2007-03-29 | 2010-06-24 | Dainippon Sumitomo Pharma Co Ltd | 新規な縮合ピロール誘導体 |
| KR20090018593A (ko) | 2007-08-17 | 2009-02-20 | 주식회사 엘지생명과학 | 세포괴사 저해제로서의 인돌 및 인다졸 화합물 |
| DE102008030207A1 (de) | 2008-06-25 | 2009-12-31 | Bayer Schering Pharma Aktiengesellschaft | Substituierte 7-Sulfanylmethyl-, 7-Sulfinylmethyl- und 7-Sulfonylmethyl-Indole und ihre Verwendung |
| DE102008030206A1 (de) | 2008-06-25 | 2009-12-31 | Bayer Schering Pharma Aktiengesellschaft | 3-Cyanoalky- und 3-Hydroxyalkyl-Indole und ihre Verwendung |
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| WO2011137220A1 (en) * | 2010-04-28 | 2011-11-03 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Small molecule neuropeptide s antagonists for the treatment of addictive disorders, mood, anxiety and sleep disorders |
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| US10414760B2 (en) | 2016-11-29 | 2019-09-17 | Angion Biomedica Corp. | Cytochrome P450 inhibitors and uses thereof |
| EP2576544A4 (en) * | 2010-06-01 | 2013-09-11 | Angion Biomedica Corp | INHIBITORS OF CYTOCHROMES P450 AND USES THEREOF |
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| AU2015301891B2 (en) | 2014-08-11 | 2019-12-05 | Angion Biomedica Corporation | Cytochrome P450 inhibitors and uses thereof |
| US10189819B2 (en) | 2014-12-10 | 2019-01-29 | Merck Sharp & Dohme, Corp. | Factor IXa inhibitors |
| EP3240778A4 (en) | 2014-12-31 | 2018-07-11 | Angion Biomedica Corp. | Methods and agents for treating disease |
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| TN2018000020A1 (en) * | 2015-07-20 | 2019-07-08 | Genzyme Corp | Colony stimulating factor-1 receptor (csf-1r) inhibitors. |
| JP2024500919A (ja) | 2020-12-23 | 2024-01-10 | ジェンザイム・コーポレーション | 重水素化コロニー刺激因子-1受容体(csf-1r)阻害剤 |
| WO2024229040A1 (en) * | 2023-05-01 | 2024-11-07 | Seed Therapeutics, Inc | Heteroaromatic indolesulfonamides |
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| DE2750283C2 (de) * | 1977-11-10 | 1985-08-22 | Bayer Ag, 5090 Leverkusen | Druck- und wärmeempfindliches Aufzeichnungsmaterial |
| JPS62503194A (ja) * | 1985-07-03 | 1987-12-17 | ポラロイド コ−ポレ−シヨン | カラー拡散転写写真フィルム単位 |
| US5041547A (en) * | 1986-08-28 | 1991-08-20 | Appleton Papers Inc. | Chromogenic substituted 4,7-diazaphthalides |
| GB9609641D0 (en) * | 1996-05-09 | 1996-07-10 | Pfizer Ltd | Compounds useful in therapy |
| CN1492863A (zh) * | 2000-12-22 | 2004-04-28 | 作为5-羟色胺-6配基的杂环基烷基-吲哚或氮杂吲哚化合物 |
-
2004
- 2004-01-20 CN CNA2004800026858A patent/CN1742007A/zh active Pending
- 2004-01-20 JP JP2006536489A patent/JP2007500253A/ja active Pending
- 2004-01-20 US US10/542,621 patent/US20060235222A1/en not_active Abandoned
- 2004-01-20 MX MXPA05007857A patent/MXPA05007857A/es unknown
- 2004-01-20 WO PCT/US2004/000017 patent/WO2004067529A1/en not_active Ceased
- 2004-01-20 AU AU2004207740A patent/AU2004207740A1/en not_active Abandoned
- 2004-01-20 CA CA002511806A patent/CA2511806A1/en not_active Abandoned
- 2004-01-20 EP EP04703558A patent/EP1597254A1/en not_active Withdrawn
- 2004-01-20 BR BR0406883-1A patent/BRPI0406883A/pt not_active IP Right Cessation
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI582080B (zh) * | 2012-07-19 | 2017-05-11 | 默沙東藥廠 | 礦皮質素受體拮抗劑 |
| CN109678862A (zh) * | 2018-08-08 | 2019-04-26 | 青岛科技大学 | 一种多取代二苯乙烯基吲哚衍生物的制备方法 |
| CN109678862B (zh) * | 2018-08-08 | 2021-04-27 | 青岛科技大学 | 一种多取代二苯乙烯基吲哚衍生物的制备方法 |
| CN109293550A (zh) * | 2018-11-23 | 2019-02-01 | 南京林业大学 | 一种含三氟甲基3,6’-非对称双吲哚化合物及其合成方法 |
| CN109293550B (zh) * | 2018-11-23 | 2020-09-25 | 南京林业大学 | 一种含三氟甲基3,6’-非对称双吲哚化合物及其合成方法 |
| CN115894330A (zh) * | 2022-09-06 | 2023-04-04 | 吉林医药学院 | 一种1-乙酰基-1h-吲哚-3-基乙酸酯衍生物的合成方法和应用 |
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004207740A1 (en) | 2004-08-12 |
| CA2511806A1 (en) | 2004-08-12 |
| US20060235222A1 (en) | 2006-10-19 |
| JP2007500253A (ja) | 2007-01-11 |
| WO2004067529A1 (en) | 2004-08-12 |
| BRPI0406883A (pt) | 2006-01-03 |
| MXPA05007857A (es) | 2005-10-18 |
| EP1597254A1 (en) | 2005-11-23 |
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