BRPI0406883A - Composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto - Google Patents

Composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto

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Publication number
BRPI0406883A
BRPI0406883A BR0406883-1A BRPI0406883A BRPI0406883A BR PI0406883 A BRPI0406883 A BR PI0406883A BR PI0406883 A BRPI0406883 A BR PI0406883A BR PI0406883 A BRPI0406883 A BR PI0406883A
Authority
BR
Brazil
Prior art keywords
compound
treating
disorder
pharmaceutical composition
formula
Prior art date
Application number
BR0406883-1A
Other languages
English (en)
Portuguese (pt)
Inventor
Michael Gregory Bell
Konstantinos Gavardinas
Douglas Linn Gernert
Timothy Alan Grese
Prabhakar Kondaji Jadhav
Peter Ambrose Lander
Mitchell Irvin Steinberg
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BRPI0406883A publication Critical patent/BRPI0406883A/pt

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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • AHUMAN NECESSITIES
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    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
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    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
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    • C07D333/62Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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  • Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Diabetes (AREA)
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  • Physical Education & Sports Medicine (AREA)
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  • Obesity (AREA)
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  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
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  • Transplantation (AREA)
  • Oncology (AREA)
  • Vascular Medicine (AREA)
BR0406883-1A 2003-01-22 2004-01-20 Composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto BRPI0406883A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US44194703P 2003-01-22 2003-01-22
PCT/US2004/000017 WO2004067529A1 (en) 2003-01-22 2004-01-20 Indole-derivative modulators of steroid hormone nuclear receptors

Publications (1)

Publication Number Publication Date
BRPI0406883A true BRPI0406883A (pt) 2006-01-03

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BR0406883-1A BRPI0406883A (pt) 2003-01-22 2004-01-20 Composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto

Country Status (9)

Country Link
US (1) US20060235222A1 (enExample)
EP (1) EP1597254A1 (enExample)
JP (1) JP2007500253A (enExample)
CN (1) CN1742007A (enExample)
AU (1) AU2004207740A1 (enExample)
BR (1) BRPI0406883A (enExample)
CA (1) CA2511806A1 (enExample)
MX (1) MXPA05007857A (enExample)
WO (1) WO2004067529A1 (enExample)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1723105B1 (en) 2004-03-03 2013-05-15 Eli Lilly And Company Bicyclic substituted indole-derivative steroid hormone nuclear receptor modulators
DE102004021637A1 (de) * 2004-05-03 2005-12-01 Merck Patent Gmbh Dihydrobenzothiophene
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