CN1703221A - 作为黑皮质素受体配体用于治疗肥胖症的2－烷基－(2－氨基－3－芳基－丙酰基)哌嗪衍生物及相关化合物 - Google Patents

作为黑皮质素受体配体用于治疗肥胖症的2－烷基－(2－氨基－3－芳基－丙酰基)哌嗪衍生物及相关化合物 Download PDF

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Publication number
CN1703221A
CN1703221A CNA2003801009342A CN200380100934A CN1703221A CN 1703221 A CN1703221 A CN 1703221A CN A2003801009342 A CNA2003801009342 A CN A2003801009342A CN 200380100934 A CN200380100934 A CN 200380100934A CN 1703221 A CN1703221 A CN 1703221A
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Prior art keywords
methyl
piperazine
propiono
base
fluorophenyl
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Pending
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CNA2003801009342A
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English (en)
Chinese (zh)
Inventor
F·H·艾伯蒂诺
X·田
W·A·马佐
A·－O·科尔森
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Procter and Gamble Ltd
Procter and Gamble Co
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Procter and Gamble Ltd
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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    • C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
CNA2003801009342A 2002-10-23 2003-10-22 作为黑皮质素受体配体用于治疗肥胖症的2－烷基－(2－氨基－3－芳基－丙酰基)哌嗪衍生物及相关化合物 Pending CN1703221A (zh)

Applications Claiming Priority (2)

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US42057802P 2002-10-23 2002-10-23
US60/420,578 2002-10-23

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CN1703221A true CN1703221A (zh) 2005-11-30

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CNA2003801009342A Pending CN1703221A (zh) 2002-10-23 2003-10-22 作为黑皮质素受体配体用于治疗肥胖症的2－烷基－(2－氨基－3－芳基－丙酰基)哌嗪衍生物及相关化合物

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CN (1) CN1703221A (US07132539-20061107-C00059.png)
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US7132539B2 (en) 2006-11-07
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EP1556361A2 (en) 2005-07-27
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CA2501231A1 (en) 2004-05-06
RU2005111967A (ru) 2006-01-20
US20050010031A1 (en) 2005-01-13
PL376702A1 (pl) 2006-01-09
BR0315614A (pt) 2005-08-30
KR20050072445A (ko) 2005-07-11
MXPA05004378A (es) 2005-07-05
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AU2003286557A1 (en) 2004-05-13
AR043054A1 (es) 2005-07-13

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