CN1671694A - 作为激酶抑制剂的二吲哚基－顺丁烯二酰亚胺衍生物 - Google Patents

作为激酶抑制剂的二吲哚基－顺丁烯二酰亚胺衍生物 Download PDF

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Publication number
CN1671694A
CN1671694A CNA038184788A CN03818478A CN1671694A CN 1671694 A CN1671694 A CN 1671694A CN A038184788 A CNA038184788 A CN A038184788A CN 03818478 A CN03818478 A CN 03818478A CN 1671694 A CN1671694 A CN 1671694A
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alkyl
aryl
compound
hydrogen
following radicals
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Chinese (zh)
Inventor
H·－C·张
B·E·玛利亚诺夫
H·叶
B·R·康维
K·德马雷斯特
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Janssen Pharmaceutica NV
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Janssen Pharmaceutica NV
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Hospice & Palliative Care (AREA)
  • Endocrinology (AREA)
  • Transplantation (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Ophthalmology & Optometry (AREA)
CNA038184788A 2002-06-05 2003-06-04 作为激酶抑制剂的二吲哚基－顺丁烯二酰亚胺衍生物 Pending CN1671694A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38593502P 2002-06-05 2002-06-05
US60/385,935 2002-06-05

Publications (1)

Publication Number Publication Date
CN1671694A true CN1671694A (zh) 2005-09-21

Family

ID=29736126

Family Applications (1)

Application Number Title Priority Date Filing Date
CNA038184788A Pending CN1671694A (zh) 2002-06-05 2003-06-04 作为激酶抑制剂的二吲哚基－顺丁烯二酰亚胺衍生物

Country Status (14)

Country Link
US (1) US6987110B2 (https=)
EP (1) EP1513830A1 (https=)
JP (1) JP2005531609A (https=)
KR (1) KR20050008787A (https=)
CN (1) CN1671694A (https=)
AU (1) AU2003238874A1 (https=)
BR (1) BR0311821A (https=)
CA (1) CA2488602A1 (https=)
CR (1) CR7606A (https=)
IL (1) IL165515A0 (https=)
MX (1) MXPA04012188A (https=)
NO (1) NO20045699L (https=)
RU (1) RU2004135382A (https=)
WO (1) WO2003104222A1 (https=)

Cited By (1)

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CN109535158A (zh) * 2016-04-26 2019-03-29 浙江工业大学 一种双芳基马来酰亚胺类化合物及其药学上可接受的盐及其制备方法和应用

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NO20045699L (no) 2005-01-28
EP1513830A1 (en) 2005-03-16
BR0311821A (pt) 2005-04-05
IL165515A0 (en) 2006-01-15
US6987110B2 (en) 2006-01-17
AU2003238874A1 (en) 2003-12-22
RU2004135382A (ru) 2005-06-27
KR20050008787A (ko) 2005-01-21
CA2488602A1 (en) 2003-12-18
US20040059113A1 (en) 2004-03-25
CR7606A (es) 2009-01-16

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