CN1390143A - 两亲型前药 - Google Patents
两亲型前药 Download PDFInfo
- Publication number
- CN1390143A CN1390143A CN00815508A CN00815508A CN1390143A CN 1390143 A CN1390143 A CN 1390143A CN 00815508 A CN00815508 A CN 00815508A CN 00815508 A CN00815508 A CN 00815508A CN 1390143 A CN1390143 A CN 1390143A
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- Prior art keywords
- prodrug
- etoposide
- oligomer
- chemical compound
- peg
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- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
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-
1999
- 1999-12-31 US US09/474,915 patent/US6713454B1/en not_active Expired - Fee Related
-
2000
- 2000-09-07 AU AU75756/00A patent/AU7575600A/en not_active Abandoned
- 2000-09-07 CZ CZ2002928A patent/CZ2002928A3/cs unknown
- 2000-09-07 NZ NZ517681A patent/NZ517681A/en unknown
- 2000-09-07 MX MXPA02002712A patent/MXPA02002712A/es unknown
- 2000-09-07 HU HU0204110A patent/HUP0204110A3/hu unknown
- 2000-09-07 CN CN00815508A patent/CN1390143A/zh active Pending
- 2000-09-07 RU RU2002109595/14A patent/RU2002109595A/ru not_active Application Discontinuation
- 2000-09-07 IL IL14855800A patent/IL148558A0/xx unknown
- 2000-09-07 WO PCT/US2000/024520 patent/WO2001019406A2/en not_active Application Discontinuation
- 2000-09-07 KR KR1020027003276A patent/KR20020059398A/ko not_active Application Discontinuation
- 2000-09-07 EP EP00964949A patent/EP1212099A2/en not_active Withdrawn
- 2000-09-07 CA CA002384645A patent/CA2384645A1/en not_active Abandoned
- 2000-09-07 PL PL00354261A patent/PL354261A1/xx not_active Application Discontinuation
- 2000-09-07 JP JP2001523037A patent/JP2003509385A/ja active Pending
- 2000-09-07 BR BR0013948-3A patent/BR0013948A/pt not_active IP Right Cessation
-
2002
- 2002-03-12 NO NO20021213A patent/NO20021213L/no not_active Application Discontinuation
-
2004
- 2004-03-24 US US10/808,044 patent/US7119074B2/en not_active Expired - Fee Related
- 2004-03-29 US US10/811,760 patent/US20040253206A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| PL354261A1 (en) | 2003-12-29 |
| KR20020059398A (ko) | 2002-07-12 |
| US7119074B2 (en) | 2006-10-10 |
| CZ2002928A3 (cs) | 2002-09-11 |
| NO20021213L (no) | 2002-05-13 |
| US20040180840A1 (en) | 2004-09-16 |
| RU2002109595A (ru) | 2003-11-27 |
| BR0013948A (pt) | 2002-05-14 |
| AU7575600A (en) | 2001-04-17 |
| HUP0204110A2 (hu) | 2003-04-28 |
| CA2384645A1 (en) | 2001-03-22 |
| WO2001019406A3 (en) | 2002-01-17 |
| JP2003509385A (ja) | 2003-03-11 |
| HUP0204110A3 (en) | 2003-08-28 |
| MXPA02002712A (es) | 2003-10-14 |
| NO20021213D0 (no) | 2002-03-12 |
| US6713454B1 (en) | 2004-03-30 |
| WO2001019406A2 (en) | 2001-03-22 |
| EP1212099A2 (en) | 2002-06-12 |
| IL148558A0 (en) | 2002-09-12 |
| US20040253206A1 (en) | 2004-12-16 |
| NZ517681A (en) | 2004-01-30 |
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