CN1149209C - 与多巴胺d3受体具有亲和力的三唑化合物 - Google Patents

与多巴胺d3受体具有亲和力的三唑化合物 Download PDF

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Publication number
CN1149209C
CN1149209C CNB008049424A CN00804942A CN1149209C CN 1149209 C CN1149209 C CN 1149209C CN B008049424 A CNB008049424 A CN B008049424A CN 00804942 A CN00804942 A CN 00804942A CN 1149209 C CN1149209 C CN 1149209C
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propyl
methyl
phenyl
cyano
methoxy
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CN1345319A (zh
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D
D·斯塔克
�ױ�
H·J·特雷贝
L·翁格
-
B·纽曼－舒尔茨
�ķ�ͺ�
K·布卢姆巴赫
D·舍贝
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BASF SE
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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  • Organic Chemistry (AREA)
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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychology (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CNB008049424A 1999-01-12 2000-01-12 与多巴胺d3受体具有亲和力的三唑化合物 Expired - Fee Related CN1149209C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19900811 1999-01-12
DE19900811.6 1999-01-12

Publications (2)

Publication Number Publication Date
CN1345319A CN1345319A (zh) 2002-04-17
CN1149209C true CN1149209C (zh) 2004-05-12

Family

ID=7894006

Family Applications (3)

Application Number Title Priority Date Filing Date
CNB008049432A Expired - Fee Related CN1267430C (zh) 1999-01-12 2000-01-12 与多巴胺d3受体具有亲和力的三唑化合物
CN00804933A Pending CN1347414A (zh) 1999-01-12 2000-01-12 对多巴胺d3受体具有亲和力的三唑化合物
CNB008049424A Expired - Fee Related CN1149209C (zh) 1999-01-12 2000-01-12 与多巴胺d3受体具有亲和力的三唑化合物

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Application Number Title Priority Date Filing Date
CNB008049432A Expired - Fee Related CN1267430C (zh) 1999-01-12 2000-01-12 与多巴胺d3受体具有亲和力的三唑化合物
CN00804933A Pending CN1347414A (zh) 1999-01-12 2000-01-12 对多巴胺d3受体具有亲和力的三唑化合物

Country Status (28)

Country Link
US (3) US6602867B1 (enExample)
EP (3) EP1140908B1 (enExample)
JP (3) JP4615125B2 (enExample)
KR (3) KR100775720B1 (enExample)
CN (3) CN1267430C (enExample)
AR (3) AR022229A1 (enExample)
AT (3) ATE424398T1 (enExample)
AU (3) AU773047B2 (enExample)
BG (2) BG65086B1 (enExample)
BR (2) BR0007500A (enExample)
CA (3) CA2359952A1 (enExample)
CO (3) CO5150182A1 (enExample)
CZ (2) CZ303926B6 (enExample)
DE (3) DE50015802D1 (enExample)
ES (2) ES2334326T3 (enExample)
HK (1) HK1045311B (enExample)
HR (1) HRP20010590A2 (enExample)
HU (2) HUP0200522A3 (enExample)
ID (2) ID29930A (enExample)
IL (3) IL144136A0 (enExample)
NO (2) NO20013444L (enExample)
NZ (2) NZ512864A (enExample)
PL (2) PL201889B1 (enExample)
SK (2) SK9852001A3 (enExample)
TR (2) TR200102026T2 (enExample)
TW (1) TWI274750B (enExample)
WO (3) WO2000042037A1 (enExample)
ZA (2) ZA200106585B (enExample)

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KR20030045187A (ko) * 2000-11-14 2003-06-09 스미스클라인비이참피이엘시이 도파민 ｄ₃수용체 조절제 (정신병 치료제)로서 유용한테트라히드로벤즈아제핀 유도체
HU227543B1 (en) * 2001-09-28 2011-08-29 Richter Gedeon Nyrt N-[4-(2-piperazin- and 2-piperidin-1-yl-ethyl)-cyclohexyl]-sulfon- and sulfamides, process for their preparation, their use and pharmaceutical compositions containing them
GB0130219D0 (en) * 2001-12-18 2002-02-06 Pfizer Ltd Compounds for the treatment of sexual dysfunction
WO2003062205A1 (en) * 2001-12-21 2003-07-31 Smithkline Beecham P.L.C. 7-sulfonyl-3-benzazepine derivatives as modulators of the dopamine receptor and their use for the treatment of cns disorders
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KR20050054084A (ko) * 2003-12-03 2005-06-10 한국전자통신연구원 수신 환경에 기반한 위성 상태 데이터 분배 기능을 가지는위성관제 시스템 및 그 방법
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DE102004027358A1 (de) 2004-06-04 2005-12-29 Abbott Gmbh & Co. Kg Pyrimidinverbindungen und ihre Verwendung
GB0413879D0 (en) * 2004-06-21 2004-07-21 Glaxo Group Ltd Compounds
GB0414795D0 (en) * 2004-07-01 2004-08-04 Glaxo Group Ltd Compounds
ATE452134T1 (de) * 2004-08-09 2010-01-15 Abbott Gmbh & Co Kg Zur behandlung von auf eine modulation des dopamin-d3-rezeptors ansprechende erkrankungen geeignete 4-piperazinylpyrimidinverbindungen
CA2577060A1 (en) * 2004-08-13 2006-02-23 Amgen Inc. Substituted benzofused heterocycles
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